AU2002325882A1 - Phenyl derivatives as factor Xa inhibitors - Google Patents
Phenyl derivatives as factor Xa inhibitorsInfo
- Publication number
- AU2002325882A1 AU2002325882A1 AU2002325882A AU2002325882A AU2002325882A1 AU 2002325882 A1 AU2002325882 A1 AU 2002325882A1 AU 2002325882 A AU2002325882 A AU 2002325882A AU 2002325882 A AU2002325882 A AU 2002325882A AU 2002325882 A1 AU2002325882 A1 AU 2002325882A1
- Authority
- AU
- Australia
- Prior art keywords
- inhibitors
- factor
- phenyl derivatives
- phenyl
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 108010074860 Factor Xa Proteins 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 230000002401 inhibitory effect Effects 0.000 title 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 title 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10139060.2 | 2001-08-08 | ||
| DE10139060A DE10139060A1 (en) | 2001-08-08 | 2001-08-08 | New bicyclic benzene derivatives useful as factor Xa and VIIa inhibitors, e.g. for treating thrombosis, myocardial infarct, arteriosclerosis, inflammation, stroke, angina, restenosis and tumors |
| PCT/EP2002/007798 WO2003013531A1 (en) | 2001-08-08 | 2002-07-12 | Phenyl derivatives as factor xa inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2002325882A1 true AU2002325882A1 (en) | 2003-06-19 |
| AU2002325882B2 AU2002325882B2 (en) | 2007-05-17 |
Family
ID=7694867
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2002325882A Ceased AU2002325882B2 (en) | 2001-08-08 | 2002-07-12 | Phenyl derivatives as factor Xa inhibitors |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US7902223B2 (en) |
| EP (1) | EP1414456B1 (en) |
| JP (1) | JP4409941B2 (en) |
| KR (1) | KR20040020061A (en) |
| CN (1) | CN1538845A (en) |
| AT (1) | ATE538792T1 (en) |
| AU (1) | AU2002325882B2 (en) |
| BR (1) | BR0211737A (en) |
| CA (1) | CA2456717C (en) |
| DE (1) | DE10139060A1 (en) |
| ES (1) | ES2377497T3 (en) |
| HU (1) | HUP0401405A2 (en) |
| MX (1) | MXPA04001121A (en) |
| PL (1) | PL367960A1 (en) |
| RU (1) | RU2004106784A (en) |
| WO (1) | WO2003013531A1 (en) |
| ZA (1) | ZA200401800B (en) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10238002A1 (en) * | 2002-08-20 | 2004-03-04 | Merck Patent Gmbh | benzimidazole derivatives |
| AU2003279735A1 (en) * | 2002-10-02 | 2004-04-23 | Bristol-Myers Squibb Company | Lactam-containing diaminoalkyl, beta-aminoacids, alpha-aminoacids and derivatives thereof as factor xa inhibitors |
| JP2006517589A (en) * | 2003-02-11 | 2006-07-27 | ブリストル−マイヤーズ スクイブ カンパニー | Benzeneacetamide compounds useful as serine protease inhibitors |
| WO2004072101A2 (en) | 2003-02-11 | 2004-08-26 | Bristol-Myers Squibb Company | Phenylglycine derivatives useful as serine protease inhibitors |
| TW200505894A (en) | 2003-08-08 | 2005-02-16 | Yamanouchi Pharma Co Ltd | Tetrahydro-2H-thiopyran-4-carboxamide derivative |
| DE602006016566D1 (en) | 2005-01-10 | 2010-10-14 | Bristol Myers Squibb Co | PHENYLGLYCINAMIDE DERIVATIVES USED AS ANTICOAGULANTS |
| WO2007002313A2 (en) * | 2005-06-24 | 2007-01-04 | Bristol-Myers Squibb Company | Phenylglycinamide and pyridylglycinamide derivatives useful as anticoagulants |
| EP1917245A1 (en) | 2005-08-21 | 2008-05-07 | Abbott GmbH & Co. KG | Heterocyclic compounds and their use as binding partners for 5-ht5 receptors |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3279880A (en) | 1965-07-12 | 1966-10-18 | Eastman Kodak Co | Polyester textile material dyed with 1-hydroxy-4-n-p-(2'-pyrrolidonyl-1-) phenyl-amino anthraquinones |
| US4208202A (en) | 1977-04-15 | 1980-06-17 | Ciba-Geigy Corporation | N-Phenyl-substituted N-heterocyclic compounds, their preparation and use in agents for regulating plant growth |
| ZA928276B (en) | 1991-10-31 | 1993-05-06 | Daiichi Seiyaku Co | Aromatic amidine derivates and salts thereof. |
| IL115420A0 (en) | 1994-09-26 | 1995-12-31 | Zeneca Ltd | Aminoheterocyclic derivatives |
| US5612353A (en) | 1995-06-07 | 1997-03-18 | Rhone-Poulenc Rorer Pharmaceuticals Inc. | Substituted (sulfinic acid, sulfonic acid, sulfonylamino or sulfinylamino) N-[(aminoiminomethyl)phenylalkyl]-azaheterocyclylamide compounds |
| DE19530996A1 (en) | 1995-08-23 | 1997-02-27 | Boehringer Mannheim Gmbh | Cyclic guanidines, process for their preparation and pharmaceuticals |
| NZ336162A (en) | 1996-12-23 | 2000-09-29 | Du Pont Pharm Co | pyrrole, tetrazole or pyrazole derivatives useful as factor Xa inhibitors |
| EP1181270A2 (en) | 1999-05-24 | 2002-02-27 | Cor Therapeutics, Inc. | Inhibitors of factor xa |
| WO2000071512A1 (en) | 1999-05-24 | 2000-11-30 | Cor Therapeutics, Inc. | INHIBITORS OF FACTOR Xa |
| CA2374793A1 (en) | 1999-05-24 | 2000-11-30 | Penglie Zhang | Inhibitors of factor xa |
| WO2000071516A2 (en) | 1999-05-24 | 2000-11-30 | Cor Therapeutics, Inc. | INHIBITORS OF FACTOR Xa |
| DE10102322A1 (en) * | 2001-01-19 | 2002-07-25 | Merck Patent Gmbh | New disubstituted and trisubstituted benzene derivatives useful as coagulation inhibitors for the treatment of thromboembolic diseases |
-
2001
- 2001-08-08 DE DE10139060A patent/DE10139060A1/en not_active Withdrawn
-
2002
- 2002-07-12 CN CNA028154827A patent/CN1538845A/en active Pending
- 2002-07-12 EP EP02760242A patent/EP1414456B1/en not_active Expired - Lifetime
- 2002-07-12 MX MXPA04001121A patent/MXPA04001121A/en unknown
- 2002-07-12 RU RU2004106784/04A patent/RU2004106784A/en not_active Application Discontinuation
- 2002-07-12 WO PCT/EP2002/007798 patent/WO2003013531A1/en active IP Right Grant
- 2002-07-12 CA CA2456717A patent/CA2456717C/en not_active Expired - Fee Related
- 2002-07-12 ES ES02760242T patent/ES2377497T3/en not_active Expired - Lifetime
- 2002-07-12 AT AT02760242T patent/ATE538792T1/en active
- 2002-07-12 KR KR10-2003-7016957A patent/KR20040020061A/en not_active Application Discontinuation
- 2002-07-12 JP JP2003518540A patent/JP4409941B2/en not_active Expired - Fee Related
- 2002-07-12 AU AU2002325882A patent/AU2002325882B2/en not_active Ceased
- 2002-07-12 BR BR0211737-1A patent/BR0211737A/en not_active IP Right Cessation
- 2002-07-12 PL PL02367960A patent/PL367960A1/en unknown
- 2002-07-12 HU HU0401405A patent/HUP0401405A2/en unknown
- 2002-07-12 US US10/486,238 patent/US7902223B2/en not_active Expired - Fee Related
-
2004
- 2004-03-04 ZA ZA200401800A patent/ZA200401800B/en unknown
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