AU2002247886A1 - Process for preparing hydroxypyrrolidinyl ethylamine compounds useful as kappa agonists - Google Patents

Process for preparing hydroxypyrrolidinyl ethylamine compounds useful as kappa agonists

Info

Publication number
AU2002247886A1
AU2002247886A1 AU2002247886A AU2002247886A AU2002247886A1 AU 2002247886 A1 AU2002247886 A1 AU 2002247886A1 AU 2002247886 A AU2002247886 A AU 2002247886A AU 2002247886 A AU2002247886 A AU 2002247886A AU 2002247886 A1 AU2002247886 A1 AU 2002247886A1
Authority
AU
Australia
Prior art keywords
hydroxypyrrolidinyl
preparing
compounds useful
kappa agonists
ethylamine compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2002247886A
Inventor
Brian Michael Andresen
Michel Andre Couturier
Keith Michael Devries
Fumitaka Ito
John Lloyd Tucker
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Products Inc
Original Assignee
Pfizer Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Publication of AU2002247886A1 publication Critical patent/AU2002247886A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/12—Oxygen or sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
AU2002247886A 2001-04-30 2002-03-25 Process for preparing hydroxypyrrolidinyl ethylamine compounds useful as kappa agonists Abandoned AU2002247886A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US28742801P 2001-04-30 2001-04-30
US60/287,428 2001-04-30
US31400601P 2001-08-21 2001-08-21
US60/314,006 2001-08-21
PCT/IB2002/000924 WO2002088082A2 (en) 2001-04-30 2002-03-25 Process for preparing hydroxypyrrolidinyl ethylamine compounds useful as kappa agonists

Publications (1)

Publication Number Publication Date
AU2002247886A1 true AU2002247886A1 (en) 2002-11-11

Family

ID=26964447

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2002247886A Abandoned AU2002247886A1 (en) 2001-04-30 2002-03-25 Process for preparing hydroxypyrrolidinyl ethylamine compounds useful as kappa agonists

Country Status (7)

Country Link
US (1) US6624313B2 (en)
EP (1) EP1461317A2 (en)
JP (1) JP2005508851A (en)
AU (1) AU2002247886A1 (en)
CA (1) CA2445874A1 (en)
MX (1) MXPA03009927A (en)
WO (1) WO2002088082A2 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1478622A1 (en) * 2002-02-28 2004-11-24 Pfizer Products Inc. Crystalline anhydrous and monohydrate benzoate salts of (2's,3s)-3-hydroxy-n- 2 n-methyl-n-4-(n-propylamino-carbonyl)phenyl]amino-2-phenyl -ethylpyrrolidine
WO2004039785A1 (en) * 2002-11-01 2004-05-13 Pfizer Products Inc. Process for the preparation of pyrrolidinyl ethylamine compounds via a copper-mediated aryl amination

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8618188D0 (en) 1986-07-25 1986-09-03 Ici Plc Diamine compounds
DE4034785A1 (en) 1990-11-02 1992-05-07 Merck Patent Gmbh 1- (2-arylethyl) pyrrolidine
IL117440A0 (en) 1995-03-31 1996-07-23 Pfizer Pyrrolidinyl hydroxamic acid compounds and their production process
TNSN97092A1 (en) * 1996-09-18 1999-12-31 Agouron Pharma Metal protein enzyme inhibitors and pharmaceutical formulations containing these inhibitors and their pharmacological use and methods and intermediates useful for preparing the aforementioned formulations.
EP0982297A3 (en) * 1998-08-24 2001-08-01 Pfizer Products Inc. Process for the preparation of hydroxy-pyrrolidinyl hydroxamic acid derivatives being opioid kappa receptor agonists

Also Published As

Publication number Publication date
CA2445874A1 (en) 2002-11-07
US20020161241A1 (en) 2002-10-31
US6624313B2 (en) 2003-09-23
WO2002088082A3 (en) 2004-05-21
JP2005508851A (en) 2005-04-07
MXPA03009927A (en) 2004-01-29
WO2002088082A2 (en) 2002-11-07
EP1461317A2 (en) 2004-09-29

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase