AU2001291852A1 - A process for producing 3,4-dihydro naphthyridinone analogs - Google Patents
A process for producing 3,4-dihydro naphthyridinone analogsInfo
- Publication number
- AU2001291852A1 AU2001291852A1 AU2001291852A AU9185201A AU2001291852A1 AU 2001291852 A1 AU2001291852 A1 AU 2001291852A1 AU 2001291852 A AU2001291852 A AU 2001291852A AU 9185201 A AU9185201 A AU 9185201A AU 2001291852 A1 AU2001291852 A1 AU 2001291852A1
- Authority
- AU
- Australia
- Prior art keywords
- dihydro
- producing
- naphthyridinone
- analogs
- naphthyridinone analogs
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/06—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom
- C07D213/08—Preparation by ring-closure
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/06—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom
- C07D213/08—Preparation by ring-closure
- C07D213/09—Preparation by ring-closure involving the use of ammonia, amines, amine salts, or nitriles
- C07D213/10—Preparation by ring-closure involving the use of ammonia, amines, amine salts, or nitriles from acetaldehyde or cyclic polymers thereof
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- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/73—Unsubstituted amino or imino radicals
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
- C07D213/80—Acids; Esters in position 3
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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- C07D213/85—Nitriles in position 3
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- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
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- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
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- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2000-289173 | 2000-09-22 | ||
JP2000289173A JP4272338B2 (en) | 2000-09-22 | 2000-09-22 | Pyridine derivatives |
PCT/EP2001/010462 WO2002024693A1 (en) | 2000-09-22 | 2001-09-11 | A process for producing 3,4-dihydro naphthyridinone analogs |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2001291852A1 true AU2001291852A1 (en) | 2002-04-02 |
Family
ID=18772618
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2001289873A Abandoned AU2001289873A1 (en) | 2000-09-22 | 2001-09-10 | Pyridine derivatives with IKB-kinase (IKK-Beta) inhibiting activity |
AU2001291852A Abandoned AU2001291852A1 (en) | 2000-09-22 | 2001-09-11 | A process for producing 3,4-dihydro naphthyridinone analogs |
AU2001289875A Abandoned AU2001289875A1 (en) | 2000-09-22 | 2001-09-11 | A process for producing 2-amino-4,6-disubstituted nicotinic acid ester analogs |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2001289873A Abandoned AU2001289873A1 (en) | 2000-09-22 | 2001-09-10 | Pyridine derivatives with IKB-kinase (IKK-Beta) inhibiting activity |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2001289875A Abandoned AU2001289875A1 (en) | 2000-09-22 | 2001-09-11 | A process for producing 2-amino-4,6-disubstituted nicotinic acid ester analogs |
Country Status (31)
Country | Link |
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US (4) | US6562811B1 (en) |
EP (1) | EP1326856B1 (en) |
JP (1) | JP4272338B2 (en) |
KR (1) | KR20030030030A (en) |
CN (1) | CN1476442A (en) |
AR (1) | AR031613A1 (en) |
AT (1) | ATE381556T1 (en) |
AU (3) | AU2001289873A1 (en) |
BG (1) | BG107632A (en) |
BR (1) | BR0114073A (en) |
CA (1) | CA2422923A1 (en) |
DE (1) | DE60132001T2 (en) |
EC (1) | ECSP034524A (en) |
EE (1) | EE200300113A (en) |
ES (1) | ES2298260T3 (en) |
GT (1) | GT200100189A (en) |
HR (1) | HRP20030306A2 (en) |
HU (1) | HUP0303124A2 (en) |
IL (1) | IL154550A0 (en) |
MA (1) | MA25836A1 (en) |
MX (1) | MXPA03002491A (en) |
NO (1) | NO20031307L (en) |
NZ (1) | NZ524811A (en) |
PE (1) | PE20020508A1 (en) |
PL (1) | PL361811A1 (en) |
RU (1) | RU2003111754A (en) |
SK (1) | SK3452003A3 (en) |
SV (1) | SV2002000637A (en) |
UY (1) | UY26943A1 (en) |
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