AU2001290311A1 - Thienopyrimidine compounds and their salts and process for preparation of both - Google Patents
Thienopyrimidine compounds and their salts and process for preparation of bothInfo
- Publication number
- AU2001290311A1 AU2001290311A1 AU2001290311A AU9031101A AU2001290311A1 AU 2001290311 A1 AU2001290311 A1 AU 2001290311A1 AU 2001290311 A AU2001290311 A AU 2001290311A AU 9031101 A AU9031101 A AU 9031101A AU 2001290311 A1 AU2001290311 A1 AU 2001290311A1
- Authority
- AU
- Australia
- Prior art keywords
- salts
- preparation
- thienopyrimidine compounds
- thienopyrimidine
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2000-299872 | 2000-09-29 | ||
JP2000299872 | 2000-09-29 | ||
PCT/JP2001/008530 WO2002026745A1 (en) | 2000-09-29 | 2001-09-28 | Thienopyrimidine compounds and their salts and process for preparation of both |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2001290311A1 true AU2001290311A1 (en) | 2002-04-08 |
Family
ID=18781622
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2001290311A Abandoned AU2001290311A1 (en) | 2000-09-29 | 2001-09-28 | Thienopyrimidine compounds and their salts and process for preparation of both |
Country Status (7)
Country | Link |
---|---|
EP (1) | EP1329454A1 (en) |
JP (1) | JPWO2002026745A1 (en) |
KR (1) | KR20030034232A (en) |
CN (1) | CN1458933A (en) |
AU (1) | AU2001290311A1 (en) |
CA (1) | CA2423981A1 (en) |
WO (1) | WO2002026745A1 (en) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2217956B1 (en) | 2003-01-23 | 2006-04-01 | Almirall Prodesfarma, S.A. | NEW DERIVATIVES OF 4-AMINOTIENE (2,3-D) PIRIMIDIN-6-CARBONITRILE. |
TW200621257A (en) * | 2004-10-20 | 2006-07-01 | Astellas Pharma Inc | Pyrimidine derivative fused with nonaromatic ring |
US7674822B2 (en) | 2004-11-24 | 2010-03-09 | Wyeth | PTP1b inhibitors |
KR101288144B1 (en) * | 2005-06-14 | 2013-07-18 | 아스카 세이야쿠 가부시키가이샤 | Thienopyrimidine derivative |
KR101507182B1 (en) * | 2006-12-07 | 2015-03-30 | 제넨테크, 인크. | Phosphoinositide 3-kinase inhibitor compounds and methods of use |
US20100093714A1 (en) * | 2008-10-13 | 2010-04-15 | Devraj Chakravarty | AMIDES OF THIENO[2,3-d]PYRIMIDINE AND THEIR USE AS ADENOSINE A2a RECEPTOR ANTAGONISTS |
SI2540728T1 (en) | 2010-02-17 | 2019-06-28 | Takeda Pharmaceutical Company Limited | Heterocyclic compound |
CN104053661B (en) | 2011-11-23 | 2018-06-19 | 癌症研究技术有限公司 | The thienopyrimidines inhibitor of atypical protein kinase C |
KR20140110066A (en) * | 2012-01-10 | 2014-09-16 | 에프. 호프만-라 로슈 아게 | Thienopyrimidine compounds |
CN103664991B (en) * | 2012-09-19 | 2016-12-28 | 中国科学院福建物质结构研究所 | Thiophene [2,3 d] pyrimidine derivatives, Its Preparation Method And Use |
CA2905751A1 (en) | 2013-03-13 | 2014-10-09 | Forma Therapeutics, Inc. | Novel compounds and compositions for inhibition of fasn |
SG11201804901WA (en) | 2015-12-22 | 2018-07-30 | SHY Therapeutics LLC | Compounds for the treatment of cancer and inflammatory disease |
EA201992780A1 (en) | 2017-06-21 | 2020-06-02 | ШАЙ ТЕРАПЬЮТИКС ЭлЭлСи | COMPOUNDS THAT INTERACT WITH THE RAS SUPERFAMILY FOR TREATMENT OF CANCER, INFLAMMATORY DISEASES, RAS OPATIAS AND FIBROUS DISEASE |
WO2019023651A2 (en) * | 2017-07-28 | 2019-01-31 | Massachusetts Institute Of Technology | Small molecule modulators of the androgen receptor |
TWI767148B (en) | 2018-10-10 | 2022-06-11 | 美商弗瑪治療公司 | Inhibiting fatty acid synthase (fasn) |
EP3873214A4 (en) | 2018-10-29 | 2022-07-13 | Forma Therapeutics, Inc. | Solid forms of (4-(2-fluoro-4-(1-methyl-1 h-benzo[d]imidazol-5-yl)benzoyl) piperazin-1-yl)(1-hydroxycyclopropyl)methanone |
US20230148450A9 (en) * | 2019-03-01 | 2023-05-11 | Revolution Medicines, Inc. | Bicyclic heteroaryl compounds and uses thereof |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5869486A (en) * | 1995-02-24 | 1999-02-09 | Ono Pharmaceutical Co., Ltd. | Fused pyrimidines and pyriazines as pharmaceutical compounds |
DE19632423A1 (en) * | 1996-08-12 | 1998-02-19 | Merck Patent Gmbh | Thienopyrimidines |
DE19644228A1 (en) * | 1996-10-24 | 1998-04-30 | Merck Patent Gmbh | Thienopyrimidines |
DE19752952A1 (en) * | 1997-11-28 | 1999-06-02 | Merck Patent Gmbh | Thienopyrimidines |
-
2001
- 2001-09-28 JP JP2002531129A patent/JPWO2002026745A1/en not_active Withdrawn
- 2001-09-28 WO PCT/JP2001/008530 patent/WO2002026745A1/en not_active Application Discontinuation
- 2001-09-28 AU AU2001290311A patent/AU2001290311A1/en not_active Abandoned
- 2001-09-28 KR KR10-2003-7004523A patent/KR20030034232A/en not_active Application Discontinuation
- 2001-09-28 CA CA002423981A patent/CA2423981A1/en not_active Abandoned
- 2001-09-28 EP EP01970282A patent/EP1329454A1/en not_active Withdrawn
- 2001-09-28 CN CN01815848A patent/CN1458933A/en active Pending
Also Published As
Publication number | Publication date |
---|---|
CA2423981A1 (en) | 2003-03-28 |
EP1329454A1 (en) | 2003-07-23 |
CN1458933A (en) | 2003-11-26 |
JPWO2002026745A1 (en) | 2004-02-05 |
WO2002026745A1 (en) | 2002-04-04 |
KR20030034232A (en) | 2003-05-01 |
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