AU2001283841A1 - N-phenyl-4-(4-pyridyl)-2-pyrimidineamine derivatives - Google Patents
N-phenyl-4-(4-pyridyl)-2-pyrimidineamine derivativesInfo
- Publication number
- AU2001283841A1 AU2001283841A1 AU2001283841A AU2001283841A AU2001283841A1 AU 2001283841 A1 AU2001283841 A1 AU 2001283841A1 AU 2001283841 A AU2001283841 A AU 2001283841A AU 2001283841 A AU2001283841 A AU 2001283841A AU 2001283841 A1 AU2001283841 A1 AU 2001283841A1
- Authority
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- Australia
- Prior art keywords
- alkyl
- optionally substituted
- amino
- hydroxy
- alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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Claims (15)
1. A process for protecting a plant against attack or infestation by a phytopathogenic organism, comprising applying at least one compound of the formula I,
wherein n is 0 or 1 ,
PM is halogen, alkoxy, haloalkyl, haloalkoxy or alkyl, R2 is hydrogen, halogen, alkyl, haloalkyl, alkoxy or haloalkoxy, each of R3, R4 and R5 is, independently of the others, hydrogen, lower alkyl or halogen, and R6 is a) hydrazino, that is unsubstituted or one- to threefold substituted by optionally substituted alkyl and/or optionally substituted acyl, b) cyclohexylamino, tetrahydro-4H-pyranyl-4-amino, pyrrolidine-3-amino, 2- or 3-tetrahydro- furylamino, all optionally substitutedby amino. hydroxy, alkoxy, alkyl or alkoxyalkyl, c) piperazinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, alkoxy, alkyl or alkoxyalkyl, d) morpholinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, alkoxy, alkyl or alkoxyalkyl, e) oxazolidinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, hydroxy- lower alkyl, alkoxy, alkyl or alkoxyalkyl, f) thiazolidinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, hydroxy- lower alkyl, alkoxy, alkyl or alkoxyalkyl, g) imidazolidinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, hydroxy- lower alkyl, alkoxy, alkyl or alkoxyalkyl, h) amino or mono- or di-(lower alkyl)amino wherein the lower alkyl moieties are unsubstituted or substituted by one or more substitutents independently selected from the 106
group con- sisting of unsubstituted amino, N-mono- or N,N-di-(lower alkyl)-amino, (lower alkoxy)-lower alk-oxy, lower alkoxycarbonylamino, hydroxy-lower alkoxycarbonylamino, lower alkoxy-lower alkoxycarbonylamino, morpholinyl, hydroxy-lower alkylamino, cyano, halogen, oxo bound to a carbon that is not directly bound to a heteroatom, hydroximino, alkoximino, optionally substituted hydrazono, lower alkenyl, lower alkynyl, guanidyl, lower alkanoylamino, hydroxy-lower alkanoylamino, lower alkoxy-lower alkanoylamino, halo-lower alkanoylamino, lower alkylaminocarbonylamino, hydroxy-lower alkylaminocarbonylamino, lower alkoxy-lower alkylaminocarbonylamino, amidino, di-lower-alkylamino-cyclohexyl, carboxy, lower alkoxycarbonyl, hydroxy-lower alkoxycarbonyl, lower alkoxy-lower alkoxycarbonyl, lower alkylcarbonyldioxy (= lower alkoxycarbonyloxy), hydroxy-lower alkoxycarbonyloxy, lower alkoxy-lower alkoxycarbonyloxy, lower alkanoyloxy, halo-lower alkanoyloxy, hydroxy-lower alkanoyloxy, lower alkoxy-lower alkanoyloxy, carbamoyl, N-mono- or N,N-di- lower alkylcarbamoyl, N-(hydroxy-lower alkyl)carbamoyl, N-lower alkyl-N-hydroxy-lower alkyl-carbamoyl, N,N-di-(hydroxy-lower alkyl)-carbamoyl, N-hydroxy-carbamoyl, hydroxy, lower alkoxy, lower alkenyloxy, lower alkinyloxy, lower haloalkoxy, lower alkylthio, lower alkylsulfinyl, lower alkylsulfonyl, lower alkoxysilyl, 4-tetrahydro-4H-pyranyl, 3-pyrrolidinyl, 2- or 3-tetrahydrofuryl, 2- or 3-dihydrofuryl, piperazinyl, lower alkanoyl-piperazinyl including formylpiperazinyl, optionally substituted heteroaryl and optionally substituted heteroaryloxy i) optionally substituted alkanoylamino, optionally substituted alkenoylamino, optionally substituted alkynoylamino, optionally substituted mono- or di-alkylaminocarbonylamino, optionally substituted alkoxycarbonylamino, optionally substituted mono- or di-alkylamino- sulfonylamino, optionally substituted mono- or di-alkylaminosulfoxylamino, j) N-(optionally substituted alkyl)-N-(optionally substituted lower alkanoyl)-amino, k) N-(optionally substituted alkyl)-N-(optionally substituted alkoxycarbonyl)-amino, I) N-(optionally substituted alkyl)-N-(N',N'-mono- or di-[optionally substituted alkyl]- aminocarbonyl)-amino, or m) N=C(R7,R8) wherein R7 is hydrogen, alkyl, amino, mono- or di-alkylamino and R8 is amino, mono- or dialkylamino or wherein R7 and R8, together with the binding carbon atom, form a saturated five- to seven-membered ring with 0, 1 or 2 ring nitrogen atoms that is optionally substituted by one or more substituents; or a salt thereof; to one or more loci selected from the group consisting of a plant, a part of a plant, seeds and the site of a plant. 107
2. A process according to claim I, wherein the phytopathogenic organism is a fungal organism.
3. A process according to claim 1 , wherein the fungal organism is one or more selected from the group of classes consisting of Ascomycetes, Basidiomycetes, Oomycetes and Fungi imperfecti.
4. A process according to claim 1 wherein the phytopathogenic organism is a bacterium.
5. A process according to claim 1 wherein the phytopathogenic organism is a virus.
6. A process according to claim 1 wherein the phytopathogenic organism is a nematode.
7. A process according to any one of claims 1 to 6 wherein a compound of formula I is applied wherein n is 0 or 1 ,
Ri is halogen, haloalkyl or haloalkoxy,
R2 is hydrogen or alkyl, each of R3, R4 and R5 is, independently of the others, hydrogen, lower alkyl or halogen, and
R6 is as defined in claim 1.
8. A process according to any one of claims 1 to 6 wherein a compound of formula I is applied wherein n is 0 or 1 ,
Ri is halogen, haloalkyl or haloalkoxy,
R2 is hydrogen or alkyl, each of R3, R4 and R5 is hydrogen, and
R6 is as defined in claim 1.
9. A process according to any one of claims 1 to 6 wherein a compound of formula I is applied wherein 108
n is 0
R-i is chloro, trifluoromethyl, trifluoromethoxy or 1 ,1 ,2,2-tetrafluoroethoxy
R2.R3, R and R5 are hydrogen, and
R6 is
(a) hydrazino, that is unsubstituted or one- to threefold substituted by optionally substituted alkyl and/or optionally substituted acyl, (e) amino or mono- or di-(lower alkyl)amino wherein the lower alkyl moieties are unsubstituted or substituted by one or more substitutents independently selected from the group con- sisting of unsubstituted amino, N-mono- or N,N-di-(lower alkyl)-amino, (lower alkoxy)- lower alk-oxy, lower alkoxycarbonylamino, hydroxy-lower alkoxycarbonylamino, lower alkoxy-lower alkoxycarbonylamino, morpholinyl, hydroxy-lower alkylamino, cyano, halogen, oxo bound to a carbon that is not directly bound to a heteroatom, hydroximino, alkoximino, optionally substituted hydrazono, lower alkenyl, lower alkynyl, guanidyl, lower alkanoylamino, hydroxy-lower alkanoylamino, lower alkoxy-lower alkanoylamino, halo-lower alkanoylamino, lower alkylaminocarbonylamino, hydroxy-lower alkylaminocarbonylamino, lower alkoxy-lower alkylaminocarbonylamino, amidino, di-lower-alkylamino-cyclohexyl, carboxy, lower alkoxycarbonyl, hydroxy-lower alkoxycarbonyl, lower alkoxy-lower alkoxycarbonyl, lower alkylcarbonyldioxy (= lower alkoxycarbonyloxy), hydroxy-lower alkoxycarbonyloxy, lower alkoxy-lower alkoxycarbonyloxy, lower alkanoyloxy, halo-lower alkanoyloxy, hydroxy-lower alkanoyloxy, lower alkoxy-lower alkanoyloxy, carbamoyl, N-mono- or N,N-di- lower alkylcarbamoyl, N-(hydroxy-lower alkyl)carbamoyl, N-lower alkyl-N-hydroxy-lower alkyl-carbamoyl, N,N-di-(hydroxy-lower alkyl)-carbamoyl, N-hydroxy-carbamoyl, hydroxy, lower alkoxy, lower alkenyloxy, lower alkinyloxy, lower haloalkoxy, lower alkylthio, lower alkylsulfinyl, lower alkylsulfonyl, lower alkoxysilyl, 4-tetrahydro-4H-pyranyl, 3-pyrrolidinyl, 2- or 3-tetrahydrofuryl, 2- or 3-dihydrofuryl, piperazinyl, lower alkanoyl-piperazinyl including formylpiperazinyl, optionally substituted heteroaryl and optionally substituted heteroaryloxy f) optionally substituted alkanoylamino, optionally substituted alkenoylamino, optionally substituted alkynoylamino, optionally substituted mono- or di-alkylaminocarbonylamino, optionally substituted alkoxycarbonylamino, optionally substituted mono- or di-alkylamino- sulfonylamino, optionally substituted mono- or di-alkylaminosulfoxylamino, g) N-(optionally substituted alkyl)-N-(optionally substituted lower alkanoyl)-amino, h) N-(optionally substituted alkyl)-N-(optionally substituted alkoxycarbonyl)-amino, i) N-(optionally substituted alkyl)-N-(N',N'-mono- or di-[optionally substituted alkyl]- aminocarbonyl)-amino, or 109
j) N=C(R7,R8) wherein R7 is hydrogen, alkyl, amino, mono- or di-alkylamino and R8 is amino, mono- or dialkylamino or wherein R7 and R8, together with the binding carbon atom, form a saturated five- to seven-membered ring with 0, 1 or 2 ring nitrogen atoms that is optionally substituted by one or more substituents; or a salt thereof.
10. A compound of the formula I, wherein n is1 ,
Ri is halogen, alkoxy, haloalkyl, haloalkoxy or alkyl,
R2 is hydrogen, halogen, alkyl, haloalkyl, alkoxy or haloalkoxy, each of R3, R4 and R5 is, independently of the others, hydrogen, lower alkyl or halogen, and
R6 is a) hydrazino, that is unsubstituted or one- to threefold substituted by optionally substituted alkyl and/or optionally substituted acyl, b) cyclohexylamino, tetrahydro-4H-pyranyl-4-amino, pyrrolidine-3-amino, 2- or 3-tetrahydro- furylamino, all optionally substitutedby amino, hydroxy, alkoxy, alkyl or alkoxyalkyl, c) piperazinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, alkoxy, alkyl or alkoxyalkyl, d) morpholinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, alkoxy, alkyl or alkoxyalkyl, e) oxazolidinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, hydroxy- lower alkyl, alkoxy, alkyl or alkoxyalkyl, f) thiazolidinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, hydroxy- lower alkyl, alkoxy, alkyl or alkoxyalkyl, g) imidazolidinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, hydroxy- lower alkyl, alkoxy, alkyl or alkoxyalkyl, h) amino or mono- or di-(lower alkyl)amino wherein the lower alkyl moieties are unsubstituted or substituted by one or more substitutents independently selected from the group con- sisting of unsubstituted amino, N-mono- or N,N-di-(lower alkyl)-amino, (lower alkoxy)-lower alk-oxy, lower alkoxycarbonylamino, hydroxy-lower alkoxycarbonylamino, lower alkoxy-lower alkoxycarbonylamino, morpholinyl, hydroxy-lower alkylamino, cyano, halogen, oxo bound to a carbon that is not directly bound to a heteroatom, hydroximino, alkoximino, optionally substituted hydrazono, lower alkenyl, lower alkynyl, guanidyl, lower alkanoylamino, hydroxy-lower alkanoylamino, lower alkoxy-lower alkanoylamino, halo-lower 110
alkanoylamino, lower alkylaminocarbonylamino, hydroxy-lower alkylaminocarbonylamino, lower alkoxy-lower alkylaminocarbonylamino, amidino, di-lower-alkylamino-cyclohexyl, carboxy, lower alkoxycarbonyl, hydroxy-lower alkoxycarbonyl, lower alkoxy-lower alkoxycarbonyl, lower alkylcarbonyldioxy (= lower alkoxycarbonyloxy), hydroxy-lower alkoxycarbonyloxy, lower alkoxy-lower alkoxycarbonyloxy, lower alkanoyloxy, halo-lower alkanoyloxy, hydroxy-lower alkanoyloxy, lower alkoxy-lower alkanoyloxy, carbamoyl, N-mono- or N,N-di- lower alkylcarbamoyl, N-(hydroxy-lower alkyl)carbamoyl, N-lower alkyl-N-hydroxy-lower alkyl-carbamoyl, N,N-di-(hydroxy-lower alkyl)-carbamoyl, N-hydroxy-carbamoyl, hydroxy, lower alkoxy, lower alkenyloxy, lower alkinyloxy, lower haloalkoxy, lower alkylthio, lower alkylsulfinyl, lower alkylsulfonyl, lower alkoxysilyl, 4-tetrahydro-4H-pyranyl, 3-pyrrolidinyl, 2- or 3-tetrahydrofuryl, 2- or 3-dihydrofuryl, piperazinyl, lower alkanoyl-piperazinyl including formylpiperazinyl, optionally substituted heteroaryl and optionally substituted heteroaryloxy i) optionally substituted alkanoylamino, optionally substituted alkenoylamino, optionally substituted alkynoylamino, optionally substituted mono- or di-alkylaminocarbonylamino, optionally substituted alkoxycarbonylamino, optionally substituted mono- or di-alkylamino- sulfonylamino, optionally substituted mono- or di-alkylaminosulfoxylamino, j) N-(optionally substituted alkyl)-N-(optionally substituted lower alkanoyl)-amino, k) N-(optionally substituted alkyl)-N-(optionally substituted alkoxycarbonyl)-amino, I) N-(optionally substituted alkyl)-N-(N',N'-mono- or di-[optionally substituted alkyl]- aminocarbonyl)-amino, or m) N=C(R7,R8) wherein R7 is hydrogen, alkyl, amino, mono- or di-alkylamino and R8 is amino, mono- or dialkylamino or wherein R7 and R8, together with the binding carbon atom, form a saturated five- to seven-membered ring with 0, 1 or 2 ring nitrogen atoms that is optionally substituted by one or more substituents; or a salt thereof.
11. A compound of the formula I wherein n is 0,
Rt is halogen, alkoxy, haloalkyl, haloalkoxy or alkyl,
R2 is hydrogen, halogen, alkyl, haloalkyl, alkoxy or haloalkoxy, each of R3, R4 and Rs is, independently of the others, hydrogen, lower alkyl or halogen, and
R6 is a) hydrazino, that is mono to threefold substituted by optionally substituted alkyl and/or 1 1 1
optionally substituted acyl, b) tetrahydro-4H-pyranyl-4-amino, pyrrolidine-3-amino, 2- or 3-tetrahydrofurylamino, all optionally substituted by amino, hydroxy, alkoxy, alkyl or alkoxyalkyl c) piperazinyl that is substituted by amino, hydroxy, alkoxy, alkyl, alkoxyalkyl, d) morpholinyl that is substitutedby amino, hydroxy, alkoxy, alkyl, e) oxazolidinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, hydroxy- lower alkyl, alkoxy, alkyl or alkoxyalkyl, f) thiazolidinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, hydroxy- lower alkyl, alkoxy, alkyl or alkoxyalkyl, g) imidazolidinyl that is optionally substituted by amino, amino-lower alkyl, hydroxy, hydroxy- lower alkyl, alkoxy, alkyl or alkoxyalkyl, h) mono- or di-(lower alkyl)amino wherein the lower alkyl moieties are substituted by one or more substitutents independently selected from the group consisting of (lower alkoxy)- lower alkoxy, lower halogenalkoxy, lower alkoxycarbonylamino, halogen, oxo, hydroximi- no, alkoximino, optionally substituted hydrazono, lower alkenyl, lower alkynyl, lower alkylcarbonyldioxy, lower alkanoyloxy, lower alkylcarbamoyl, alkenyloxy, alkynyloxy, lower alkylthio, lower alkylsulfinyl, lower alkylsulfonyl, lower alkoxysilyl, 4-tetrahydro-4H-pyranyl, 3-pyrrolidine, 2- or 3-tetra- hydrofuryl, 2- or 3-dihydrofuryl, substituted heteroaryl and optionally substituted heteroaryloxy, i) optionally substituted alkenoylamino, optionally substituted alkynoylamino, optionally substituted mono- or di-alkylaminocarbonylamino, optionally substituted alkoxycarbonylamino, optionally substituted mono- or di-alkylaminosulfonylamino, optionally substituted mono- or di-alkylaminosulfoxylamino, j) N=C(R7,R8) wherein R7 is hydrogen, alkyl, amino, mono- or di-alkylamino and R8 is amino, mono- or di-alkylamino or wherein R7 and Re, together with the binding carbon atom, form a saturated five- to seven-membered ring with 0, 1 or 2 ring nitrogen atoms that is optionally substituted by one or more substituents; or a salt thereof;
12. A compound of the formula I according to claim 11 selected from the group of N-(3-chloro-phenyl)-4-(ethylamino-4-pyridyl)-2-pyrimidine-amine,
N-(3-chloro-phenyl)-4-[2-{1-(2-methoxy-1-methyl)-ethylamino}-4-pyridyl]-2-pyrimidine-amine, N-(3-chloro-phenyl)-4-[2-(N", N'-dimethyl-acetamidino)-4-pyridyl]-2-pyrimidine-amine, 112
13. The use of a compound of the formula I, or a salt thereof, mentioned in any one of claim 1 to 11 for protection of a plant against attack by a phytopathogenic organism or the treatment of a plant infested by a phytopathogenic organism, said use comprising the administration of a compound of the formula I or a salt thereof, or a composition comprising said compound or salt and a carrier material acceptable for agricultural purposes, to any one or more selected from the group consisting of a plant, a part of a plant, seeds and the locus of a plant.
14. A method of protecting a plant against attack by a phytopathogenic organism and/or the treatment of a plant infested by a phytopathogenic organism, said method comprising administering a compound of the formula I mentioned in any one of claims 1 to 11 or a salt thereof, or a composition comprising said compound or salt and a carrier material acceptable for agricultural purposes, to any one or more selected from the group consisting of a plant, a part of a plant, seeds and the locus of a plant, preferably if in need of such treatment.
15. A composition for protecting a plant against attack by a phytopathogenic organisms and/or the treatment of a plant infested by a phytopathogenic organism, said composition comprising a compound of the formula I as mentioned in any one of claims 1 to 11 or a salt thereof and a carrier material acceptable for agricultural purposes.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0014022.8A GB0014022D0 (en) | 2000-06-08 | 2000-06-08 | Organic compounds |
| GB0014022.8 | 2000-06-08 | ||
| PCT/EP2001/006389 WO2001093682A1 (en) | 2000-06-08 | 2001-06-06 | N-phenyl-4-(4-pyridyl)-2-pyrimidineamine derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2001283841A1 true AU2001283841A1 (en) | 2002-03-07 |
| AU2001283841B2 AU2001283841B2 (en) | 2005-05-05 |
Family
ID=9893268
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001283841A Ceased AU2001283841B2 (en) | 2000-06-08 | 2001-06-06 | N-phenyl-4-(4-pyridyl)-2-pyrimidineamine derivatives |
| AU8384101A Pending AU8384101A (en) | 2000-06-08 | 2001-06-06 | N-phenyl-4-(4-pyridyl)-2-pyrimidineamine derivatives |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU8384101A Pending AU8384101A (en) | 2000-06-08 | 2001-06-06 | N-phenyl-4-(4-pyridyl)-2-pyrimidineamine derivatives |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US7109197B2 (en) |
| EP (1) | EP1292190B1 (en) |
| JP (1) | JP4991080B2 (en) |
| KR (1) | KR20030007867A (en) |
| CN (1) | CN1446048A (en) |
| AT (1) | ATE302549T1 (en) |
| AU (2) | AU2001283841B2 (en) |
| BR (1) | BR0111492A (en) |
| CA (1) | CA2409877A1 (en) |
| DE (1) | DE60112933T2 (en) |
| ES (1) | ES2245992T3 (en) |
| GB (1) | GB0014022D0 (en) |
| IL (1) | IL152899A0 (en) |
| MX (1) | MXPA02011919A (en) |
| PL (1) | PL360434A1 (en) |
| WO (1) | WO2001093682A1 (en) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0100102D0 (en) | 2001-01-03 | 2001-02-14 | Syngenta Participations Ag | Organic compounds |
| GB0129391D0 (en) * | 2001-12-07 | 2002-01-30 | Syngenta Participations Ag | Microbiocidal n-phenyl-n-[4-(4-pyridyl)-2-pyrimidin-2-yl]-amine derivatives |
| PL373484A1 (en) | 2001-12-10 | 2005-09-05 | Amgen Inc. | Vanilloid receptor ligands and their use in treatments |
| GB0129476D0 (en) * | 2001-12-10 | 2002-01-30 | Syngenta Participations Ag | Organic compounds |
| MXPA04011472A (en) * | 2002-05-22 | 2005-02-14 | Amgen Inc | Amino-pyridine, -pyridine and pyridazine derivatives for use as vanilloid receptor ligands for the treatment of pain. |
| PL375447A1 (en) * | 2002-08-14 | 2005-11-28 | Vertex Pharmaceuticals Incorporated | Protein kinase inhibitors and uses thereof |
| WO2004078682A2 (en) * | 2003-03-05 | 2004-09-16 | Irm Llc | Cyclic compounds and compositions as protein kinase inhibitors |
| GB0307269D0 (en) * | 2003-03-28 | 2003-05-07 | Syngenta Ltd | Fungicidal compositions |
| GB0307268D0 (en) * | 2003-03-28 | 2003-05-07 | Syngenta Ltd | Organic compounds |
| US20050130968A1 (en) * | 2003-10-03 | 2005-06-16 | Irvine Nicholas M. | Fungicidal 4-(2-aminopyridin-4-yl)-N-phenyl-1,3,5-triazin-2-amine derivatives |
| GB0428514D0 (en) * | 2004-12-31 | 2005-02-09 | Prosidion Ltd | Compounds |
| AR063946A1 (en) * | 2006-09-11 | 2009-03-04 | Cgi Pharmaceuticals Inc | CERTAIN REPLACED PIRIMIDINS, THE USE OF THE SAME FOR THE TREATMENT OF DISEASES MEDIATED BY THE INHIBITION OF THE ACTIVITY OF BTK AND PHARMACEUTICAL COMPOSITIONS THAT UNDERSTAND THEM. |
| CL2008001460A1 (en) * | 2007-05-16 | 2008-11-21 | Bayer Cropscience Sa | Compounds derived from phenyl-pyrimidin-amino; intermediary compounds; fungicidal composition comprising said compounds; and method to control phytopathogenic fungi from agricultural crops. |
| CN101902912A (en) * | 2007-11-06 | 2010-12-01 | 纳幕尔杜邦公司 | Fungicidal amines |
| TW200940537A (en) * | 2008-02-26 | 2009-10-01 | Astrazeneca Ab | Heterocyclic urea derivatives and methods of use thereof |
| CA2738787A1 (en) * | 2008-11-13 | 2010-05-20 | Bayer Cropscience Ag | Substituted (pyridyl)-azinylamine derivatives as fungicides |
| WO2010055114A1 (en) * | 2008-11-14 | 2010-05-20 | Bayer Cropscience Sa | Substituted (pyridyl)-azinylamine derivatives as plant protection agents |
| EP2264010A1 (en) * | 2009-06-03 | 2010-12-22 | Bayer CropScience AG | Hetarylamidines |
| ES2570784T3 (en) | 2010-12-22 | 2016-05-20 | Purdue Pharma Lp | Substituted pyridines as sodium channel blockers |
| WO2012101065A2 (en) * | 2011-01-28 | 2012-08-02 | Novartis Ag | Pyrimidine biaryl amine compounds and their uses |
| WO2012101066A1 (en) * | 2011-01-28 | 2012-08-02 | Novartis Ag | Pyridine biaryl amine compounds and their uses |
| CN103183669B (en) * | 2011-12-27 | 2015-11-18 | 湖南化工研究院 | Thiazole methylamine yl pyridines compounds and preparation method thereof |
| US20160009732A1 (en) * | 2013-03-14 | 2016-01-14 | Concert Pharmaceuticals, Inc. | Deuterated pacritinib |
| US9339029B2 (en) * | 2014-09-04 | 2016-05-17 | Preceres Inc. | Hydrazinyl lipidoids and uses thereof |
| JP6734267B2 (en) | 2014-09-26 | 2020-08-05 | ザ ケマーズ カンパニー エフシー リミテッド ライアビリティ カンパニー | Isocyanate-derived organosilane |
| CN104387377B (en) * | 2014-10-14 | 2017-03-29 | 湖南海利常德农药化工有限公司 | A kind of preparation method of thiazole methylamine yl pyridines class compound |
| WO2017110861A1 (en) * | 2015-12-25 | 2017-06-29 | 住友化学株式会社 | Plant disease control agent containing oxadiazole compound |
| EA202191890A1 (en) | 2019-01-18 | 2022-02-03 | Астразенека Аб | PCSK9 INHIBITORS AND METHODS FOR THEIR USE |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE151404C (en) | ||||
| DD151404A1 (en) * | 1980-06-13 | 1981-10-21 | Friedrich Franke | FUNGICIDAL AGENTS |
| JPH0629263B2 (en) * | 1985-10-30 | 1994-04-20 | クミアイ化学工業株式会社 | Pyrimidine derivatives and agricultural and horticultural fungicides |
| CA1288433C (en) * | 1986-12-03 | 1991-09-03 | Tsuguhiro Katoh | Pyridinylpyrimidine derivatives, method for production thereof and a fungicide containing them as the active ingredient |
| JP2517992B2 (en) * | 1986-12-03 | 1996-07-24 | 住友化学工業株式会社 | Pyridylpyrimidine derivative and plant disease controlling agent containing the same |
| EP0388838B1 (en) * | 1989-03-22 | 1996-01-10 | Ciba-Geigy Ag | Parasiticide |
| DE4034762A1 (en) | 1990-11-02 | 1992-05-07 | Hoechst Ag | Pyridyl pyrimidine derivs. - are fungicides for plant protection and for protecting and preserving industrial materials |
| DE69429078T2 (en) * | 1993-10-01 | 2002-07-11 | Novartis Ag | PHARMACOLOGICALLY EFFECTIVE PYRIDE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF |
| JP3588116B2 (en) * | 1993-10-01 | 2004-11-10 | ノバルティス アクチェンゲゼルシャフト | Pharmacologically active pyrimidineamine derivatives and process for their production |
| CA2148931A1 (en) * | 1993-10-01 | 1995-04-13 | Jurg Zimmermann | Pyrimidineamine derivatives and processes for the preparation thereof |
| WO1997049697A1 (en) * | 1996-06-21 | 1997-12-31 | Zeneca Limited | Pyridylaminopyrimidines as fungicides |
-
2000
- 2000-06-08 GB GBGB0014022.8A patent/GB0014022D0/en not_active Ceased
-
2001
- 2001-06-06 CN CN01813806A patent/CN1446048A/en active Pending
- 2001-06-06 KR KR1020027016526A patent/KR20030007867A/en not_active Application Discontinuation
- 2001-06-06 WO PCT/EP2001/006389 patent/WO2001093682A1/en active IP Right Grant
- 2001-06-06 IL IL15289901A patent/IL152899A0/en unknown
- 2001-06-06 CA CA002409877A patent/CA2409877A1/en not_active Abandoned
- 2001-06-06 AU AU2001283841A patent/AU2001283841B2/en not_active Ceased
- 2001-06-06 JP JP2002501259A patent/JP4991080B2/en not_active Expired - Fee Related
- 2001-06-06 AU AU8384101A patent/AU8384101A/en active Pending
- 2001-06-06 DE DE60112933T patent/DE60112933T2/en not_active Expired - Lifetime
- 2001-06-06 AT AT01962712T patent/ATE302549T1/en not_active IP Right Cessation
- 2001-06-06 PL PL36043401A patent/PL360434A1/en not_active Application Discontinuation
- 2001-06-06 MX MXPA02011919A patent/MXPA02011919A/en unknown
- 2001-06-06 BR BR0111492-1A patent/BR0111492A/en not_active IP Right Cessation
- 2001-06-06 ES ES01962712T patent/ES2245992T3/en not_active Expired - Lifetime
- 2001-06-06 EP EP01962712A patent/EP1292190B1/en not_active Expired - Lifetime
- 2001-06-06 US US10/297,737 patent/US7109197B2/en not_active Expired - Fee Related
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