AU2001283539A1 - Tetrahydroisoquinoline-3-carboxylic acid alkoxyguanidines as integrin antagonists - Google Patents
Tetrahydroisoquinoline-3-carboxylic acid alkoxyguanidines as integrin antagonistsInfo
- Publication number
- AU2001283539A1 AU2001283539A1 AU2001283539A AU8353901A AU2001283539A1 AU 2001283539 A1 AU2001283539 A1 AU 2001283539A1 AU 2001283539 A AU2001283539 A AU 2001283539A AU 8353901 A AU8353901 A AU 8353901A AU 2001283539 A1 AU2001283539 A1 AU 2001283539A1
- Authority
- AU
- Australia
- Prior art keywords
- alkoxyguanidines
- tetrahydroisoquinoline
- carboxylic acid
- integrin antagonists
- integrin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US22347800P | 2000-08-07 | 2000-08-07 | |
| US60223478 | 2000-08-07 | ||
| PCT/US2001/041601 WO2002012193A1 (en) | 2000-08-07 | 2001-08-07 | Tetrahydroisoquinoline-3-carboxylic acid alkoxyguanidines as integrin antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2001283539A1 true AU2001283539A1 (en) | 2002-02-18 |
Family
ID=22836666
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001283539A Abandoned AU2001283539A1 (en) | 2000-08-07 | 2001-08-07 | Tetrahydroisoquinoline-3-carboxylic acid alkoxyguanidines as integrin antagonists |
Country Status (3)
| Country | Link |
|---|---|
| US (1) | US20020037897A1 (en) |
| AU (1) | AU2001283539A1 (en) |
| WO (1) | WO2002012193A1 (en) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR0209711A (en) | 2001-05-29 | 2004-11-03 | Kyoto Pharma Ind | Heterocyclic compound and its medicinal use |
| MXPA03010867A (en) | 2001-05-29 | 2004-02-27 | Kyoto Pharma Ind | Novel heterocyclic derivatives and medicinal use thereof. |
| US20070077303A1 (en) * | 2005-09-30 | 2007-04-05 | Azaam Alli | Methods for providing oxidatively stable ophthalmic compositions |
| PT2054045E (en) * | 2006-08-16 | 2011-08-31 | Action Medicines Sl | Use of 2,5-dihydroxybenzene derivatives for the treatment of arthritis and pain |
| JP6425712B2 (en) | 2013-05-14 | 2018-11-21 | ザ ルブリゾル コーポレイションＴｈｅ Ｌｕｂｒｉｚｏｌ Ｃｏｒｐｏｒａｔｉｏｎ | Lubricating composition and method of lubricating a transmission |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5731324A (en) * | 1993-07-22 | 1998-03-24 | Eli Lilly And Company | Glycoprotein IIb/IIIa antagonists |
| DE19548709A1 (en) * | 1995-12-23 | 1997-07-03 | Merck Patent Gmbh | Tyrosine derivatives |
| AU3343097A (en) * | 1996-06-28 | 1998-01-21 | Merck Patent Gmbh | Phenylalamine derivatives as integrin inhibitors |
| CA2309341A1 (en) * | 1997-11-24 | 1999-06-03 | Merck & Co., Inc. | Substituted .beta.-alanine derivatives as cell adhesion inhibitors |
| JP2001524467A (en) * | 1997-11-26 | 2001-12-04 | ３−ディメンショナル ファーマシューティカルズ， インコーポレイテッド | Heteroarylaminoguanidines and alkoxyguanidines and their use as protease inhibitors |
| US6344486B1 (en) * | 1998-04-03 | 2002-02-05 | 3-Dimensional Pharmaceuticals, Inc. | Benzamide and sulfonamide substituted aminoguanidines and alkoxyguanidines as protease inhibitors |
| JP2003501352A (en) * | 1999-05-27 | 2003-01-14 | ３−ディメンショナル ファーマシューティカルズ， インコーポレイテッド | Oxaza heterocycles as protease inhibitors |
-
2001
- 2001-08-06 US US09/921,759 patent/US20020037897A1/en not_active Abandoned
- 2001-08-07 AU AU2001283539A patent/AU2001283539A1/en not_active Abandoned
- 2001-08-07 WO PCT/US2001/041601 patent/WO2002012193A1/en active Application Filing
Also Published As
| Publication number | Publication date |
|---|---|
| US20020037897A1 (en) | 2002-03-28 |
| WO2002012193A1 (en) | 2002-02-14 |
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