AU2001256769A1 - Triazole derivatives - Google Patents

Triazole derivatives

Info

Publication number
AU2001256769A1
AU2001256769A1 AU2001256769A AU5676901A AU2001256769A1 AU 2001256769 A1 AU2001256769 A1 AU 2001256769A1 AU 2001256769 A AU2001256769 A AU 2001256769A AU 5676901 A AU5676901 A AU 5676901A AU 2001256769 A1 AU2001256769 A1 AU 2001256769A1
Authority
AU
Australia
Prior art keywords
triazole derivatives
triazole
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001256769A
Inventor
Michael Arlt
Hartmut Greiner
Wataru Hamaguchi
Tetsuya Kimizuka
Atsuyuki Kohara
Kyoichi Maeno
Junji Miyata
Takuma Morita
Itsuro Shimada
Takashi Sugane
Takeshi Suzuki
Takahiko Tobe
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Patent GmbH
Original Assignee
Merck Patent GmbH
Yamanouchi Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent GmbH, Yamanouchi Pharmaceutical Co Ltd filed Critical Merck Patent GmbH
Publication of AU2001256769A1 publication Critical patent/AU2001256769A1/en
Assigned to MERCK PATENT GMBH reassignment MERCK PATENT GMBH Request for Assignment Assignors: MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG, YAMANOUCHI PHARMACEUTICAL CO., LTD.
Abandoned legal-status Critical Current

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    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
    • C—CHEMISTRY; METALLURGY
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    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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