AU2001234175A1 - Novel cyclic amide derivatives - Google Patents

Novel cyclic amide derivatives

Info

Publication number
AU2001234175A1
AU2001234175A1 AU2001234175A AU2001234175A AU2001234175A1 AU 2001234175 A1 AU2001234175 A1 AU 2001234175A1 AU 2001234175 A AU2001234175 A AU 2001234175A AU 2001234175 A AU2001234175 A AU 2001234175A AU 2001234175 A1 AU2001234175 A1 AU 2001234175A1
Authority
AU
Australia
Prior art keywords
amide derivatives
cyclic amide
novel cyclic
novel
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU2001234175A
Other versions
AU2001234175B2 (en
Inventor
Akira Nakao
Masahiro Okuyama
Mitsuru Ooizumi
Ken-Ichi Saito
Haruko Yamabe
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Mitsubishi Pharma Corp
Original Assignee
Mitsubishi Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsubishi Pharma Corp filed Critical Mitsubishi Pharma Corp
Priority claimed from PCT/JP2001/001413 external-priority patent/WO2001064670A1/en
Publication of AU2001234175A1 publication Critical patent/AU2001234175A1/en
Application granted granted Critical
Publication of AU2001234175B2 publication Critical patent/AU2001234175B2/en
Anticipated expiration legal-status Critical
Expired legal-status Critical Current

Links

AU2001234175A 2000-02-29 2001-02-26 Novel cyclic amide derivatives Expired AU2001234175B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2000054674 2000-02-29
JP2000-54674 2000-02-29
PCT/JP2001/001413 WO2001064670A1 (en) 2000-02-29 2001-02-26 Novel cyclic amide derivatives

Publications (2)

Publication Number Publication Date
AU2001234175A1 true AU2001234175A1 (en) 2001-11-22
AU2001234175B2 AU2001234175B2 (en) 2004-10-07

Family

ID=18575896

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2001234175A Expired AU2001234175B2 (en) 2000-02-29 2001-02-26 Novel cyclic amide derivatives
AU3417501A Pending AU3417501A (en) 2000-02-29 2001-02-26 Novel cyclic amide derivatives

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU3417501A Pending AU3417501A (en) 2000-02-29 2001-02-26 Novel cyclic amide derivatives

Country Status (19)

Country Link
US (1) US7166617B2 (en)
EP (1) EP1260512B1 (en)
JP (1) JP4859324B2 (en)
KR (1) KR100815772B1 (en)
CN (1) CN100384836C (en)
AT (1) ATE366249T1 (en)
AU (2) AU2001234175B2 (en)
CA (1) CA2401711C (en)
CY (1) CY1106858T1 (en)
DE (1) DE60129210T2 (en)
DK (1) DK1260512T3 (en)
ES (1) ES2291293T3 (en)
HU (1) HUP0300203A3 (en)
IL (2) IL151533A0 (en)
NZ (1) NZ521576A (en)
PT (1) PT1260512E (en)
RU (1) RU2257384C2 (en)
TW (1) TWI296625B (en)
WO (1) WO2001064670A1 (en)

Families Citing this family (42)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7550459B2 (en) * 2001-12-28 2009-06-23 Acadia Pharmaceuticals, Inc. Tetrahydroquinoline analogues as muscarinic agonists
EP1461318B9 (en) * 2001-12-28 2005-12-28 Acadia Pharmaceuticals Inc. Tetrahydroquinoline analogues as muscarinic agonists
CA2543419A1 (en) * 2003-10-24 2005-05-06 Leyi Gong Ccr3 receptor antagonists
US20060019969A1 (en) * 2004-07-24 2006-01-26 Laboratorios Dr. Esteve S.A. Use of compounds active on the sigma receptor for the treatment of allodynia
US8329694B2 (en) 2005-06-24 2012-12-11 Toyama Chemical Co., Ltd. Quinoxalinones as antibacterial composition
US7807706B2 (en) * 2005-08-12 2010-10-05 Astrazeneca Ab Metabotropic glutamate-receptor-potentiating isoindolones
JP2009509921A (en) * 2005-08-12 2009-03-12 アストラゼネカ アクチボラグ Substituted isoindolones and their use as metabotropic glutamate receptor potentiators
US7868008B2 (en) * 2005-08-12 2011-01-11 Astrazeneca Ab Substituted isoindolones and their use as metabotropic glutamate receptor potentiators
JP2009512711A (en) 2005-10-21 2009-03-26 ブレインセルス，インコーポレイティド Regulation of neurogenesis by PDE inhibition
AU2006308889A1 (en) 2005-10-31 2007-05-10 Braincells, Inc. GABA receptor mediated modulation of neurogenesis
TW200804281A (en) * 2006-02-16 2008-01-16 Astrazeneca Ab New metabotropic glutamate receptor-potentiating isoindolones
US20100216734A1 (en) 2006-03-08 2010-08-26 Braincells, Inc. Modulation of neurogenesis by nootropic agents
US7678808B2 (en) 2006-05-09 2010-03-16 Braincells, Inc. 5 HT receptor mediated neurogenesis
AU2007249399A1 (en) 2006-05-09 2007-11-22 Braincells, Inc. Neurogenesis by modulating angiotensin
US7998971B2 (en) * 2006-09-08 2011-08-16 Braincells Inc. Combinations containing a 4-acylaminopyridine derivative
US20100184806A1 (en) 2006-09-19 2010-07-22 Braincells, Inc. Modulation of neurogenesis by ppar agents
CN101186612B (en) * 2006-11-15 2012-10-03 天津和美生物技术有限公司 Pyrroline derivative capable of inhibiting cell to release tumor necrotic factor and its preparation and application
US8247563B2 (en) 2006-12-11 2012-08-21 Reviva Pharmaceuticals, Inc. Compositions, synthesis, and methods of using indanone based cholinesterase inhibitors
TWI417100B (en) * 2007-06-07 2013-12-01 Astrazeneca Ab Oxadiazole derivatives and their use as metabotropic glutamate receptor potentiators-842
WO2009010479A2 (en) * 2007-07-13 2009-01-22 Euroscreen S.A. Heterocyclic methylene piperidine derivatives and their use
DE102007047737A1 (en) * 2007-10-05 2009-04-30 Merck Patent Gmbh Piperidine and piperazine derivatives
US7790760B2 (en) * 2008-06-06 2010-09-07 Astrazeneca Ab Metabotropic glutamate receptor isoxazole ligands and their use as potentiators 286
WO2010099217A1 (en) 2009-02-25 2010-09-02 Braincells, Inc. Modulation of neurogenesis using d-cycloserine combinations
EP2353591A1 (en) 2010-02-04 2011-08-10 Laboratorios Del. Dr. Esteve, S.A. Sigma ligands for potentiating the analgesic effect of opioids and opiates in post-operative pain and attenuating the dependency thereof
EP3335731A1 (en) * 2010-07-20 2018-06-20 Minerva Neurosciences, Inc. Use of cyclic amide derivatives to treat sleep disorders
ES2914120T3 (en) * 2010-07-20 2022-06-07 Minerva Neurosciences Inc Methods of Using Cyclic Amide Derivatives to Treat Sigma Receptor Mediated Disorders
US8937900B2 (en) 2010-07-20 2015-01-20 Qualcomm Incorporated Enhancing pilot channel transmission in TD-SCDMA multicarrier systems using secondary carrier frequencies
EP2415471A1 (en) 2010-08-03 2012-02-08 Laboratorios Del. Dr. Esteve, S.A. Use of sigma ligands in opioid-induced hyperalgesia
EP2524694A1 (en) 2011-05-19 2012-11-21 Laboratorios Del. Dr. Esteve, S.A. Use of sigma ligands in diabetes type-2 associated pain
CN103524515B (en) 2012-07-03 2016-07-06 浙江海正药业股份有限公司 Benzodioxole derivatives with inhibiting activity of acetylcholinesterase and its production and use
US10179776B2 (en) * 2014-06-09 2019-01-15 Intra-Cellular Therapies, Inc. Compounds and methods of use to treat schizophrenia
WO2016089766A1 (en) 2014-12-02 2016-06-09 Minerva Neurosciences, Inc. Compositions comprising 2-((1-(2(4-fluorophenyl)-2-oxoethyl)piperidin-4-yl)methyl)isoindolin-1-one for treating schizophrenia
WO2016199878A1 (en) * 2015-06-11 2016-12-15 富山化学工業株式会社 Sigma-receptor binding agent
CN105523939B (en) * 2015-12-30 2017-11-14 李函璞 A kind of preparation method of lenalidomide intermediate
US20190216793A1 (en) * 2016-05-25 2019-07-18 Minerva Neurosciences, Inc. Compositions and methods for treating negative symptoms in non-schizophrenic patients
WO2018237207A1 (en) 2017-06-21 2018-12-27 Minerva Neurosciences, Inc. Gastro-resistant controlled release oral dosage forms
US11083723B2 (en) 2018-08-21 2021-08-10 Minerva Neurosciences, Inc. Use of roluperidone to treat negative symptoms and disorders, increase neuroplasticity, and promote neuroprotection
WO2020264486A1 (en) 2019-06-28 2020-12-30 Teva Czech Industries S.R.O Solid state forms of roluperidone and salts thereof
WO2021236879A1 (en) 2020-05-20 2021-11-25 The Board Of Trustees Of The University Of Illinois Method for treating lysosomal storage diseases with histatin peptides
AU2021325927A1 (en) 2020-08-14 2023-02-23 Minerva Neurosciences, Inc. Condensed azacycles as sigma ligand compounds and uses thereof
CN113651767B (en) * 2021-09-18 2023-06-09 江西中医药大学 Benzisoxazole heterocyclic compound and preparation method and application thereof
US20230255953A1 (en) 2022-02-14 2023-08-17 Minerva Neurosciences, Inc. Use of roluperidone in preventing relapse in schizophrenia patients

Family Cites Families (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3797494A (en) 1969-04-01 1974-03-19 Alza Corp Bandage for the administration of drug by controlled metering through microporous materials
US3742951A (en) 1971-08-09 1973-07-03 Alza Corp Bandage for controlled release of vasodilators
US3996934A (en) 1971-08-09 1976-12-14 Alza Corporation Medical bandage
US3947578A (en) 1972-07-28 1976-03-30 Roussel Uclaf Omega-[4-(3"-indolyl)-piperidino]-alkyl-arylketones as nevroleptics
US3921636A (en) 1973-01-15 1975-11-25 Alza Corp Novel drug delivery device
US4000287A (en) 1974-12-16 1976-12-28 Ciba-Geigy Corporation Isoindolinopiperidines
US4031894A (en) 1975-12-08 1977-06-28 Alza Corporation Bandage for transdermally administering scopolamine to prevent nausea
US4062953A (en) 1976-06-24 1977-12-13 E. R. Squibb & Sons, Inc. Various 2-substituted-1H-benz[de]isoquinoline-1,3(2H)-diones
US4168315A (en) 1977-09-28 1979-09-18 The Upjohn Company Dianisyl thiazole compound, compositions and method of antithrombotic treatment
US4495194A (en) 1982-11-12 1985-01-22 Mead Johnson & Company Antihypertensive isoindole derivatives
US4912117A (en) 1985-07-02 1990-03-27 Merrell Dow Pharmaceuticals Inc. Novel chemical compounds
US4783471A (en) 1985-07-02 1988-11-08 Merrell Dow Pharmaceuticals Inc. N-aralkyl piperidine methanol derivatives and the uses thereof
US5169096A (en) 1985-07-02 1992-12-08 Merrell Dow Pharmaceuticals Inc. N-aralkyl-piperidine-methanol derivatives
US5021428A (en) 1985-07-02 1991-06-04 Merrell Dow Pharmaceuticals Inc. Novel chemical compounds for the prophylactic treatment of migraine
US4762842A (en) 1985-10-01 1988-08-09 Eli Lilly And Company Selective method for blocking 5HT2 receptors
AU593194B2 (en) 1986-09-26 1990-02-01 Sumitomo Pharmaceuticals Company, Limited Imide derivatives ,and their production and use
EP0296477B1 (en) * 1987-06-26 1996-05-15 Hitachi, Ltd. Superconducting wire
US4877798A (en) 1987-11-23 1989-10-31 Merrell Dow Pharmaceuticals Inc. Treatment of fibromyalgia
US5166211A (en) 1987-12-17 1992-11-24 Merrell Dow Pharmaceuticals Inc. Method of using 1,4-disubstituted piperidinyl compounds in the treatment of coronary vasospasons and variant angina
US5093341A (en) 1987-12-17 1992-03-03 Merrell Dow Pharmaceuticals Inc. N-aralkyl piperidine derivatives useful as antithrombolytic agents
EP0325063B1 (en) 1988-01-21 1994-03-09 Merrell Dow Pharmaceuticals Inc. Use of 1,4-disubstituted-piperidinyl compounds in the manufacture of a medicament for the treatment of insomnia
EP0339342A1 (en) 1988-04-23 1989-11-02 Bayer Ag N-substituted N-amino pyrroles
US5182399A (en) 1988-10-13 1993-01-26 Merrell Dow Pharmaceuticals Inc. Process for preparing piperidinyl benzimidazoles
US4908372A (en) 1988-10-13 1990-03-13 Merrell Dow Pharmaceuticals Inc. Antihistaminic piperidinyl benzimidazoles
FR2641278B1 (en) 1989-01-05 1991-03-22 Lipha PIPERIDINES, METHODS OF PREPARATION AND MEDICAMENTS CONTAINING THEM
US5356906A (en) 1989-10-27 1994-10-18 The Du Pont Merck Pharmaceutical Company (N-phthalimidoalkyl) piperidines useful as treatments for psychosis
KR927002347A (en) * 1989-10-27 1992-09-03 레이몬드 지. 아너 (N-phthalimidoalkyl) piperidine
US5106855A (en) 1989-12-20 1992-04-21 Merrell Dow Pharmaceuticals Inc. Method for the treatment of glaucoma
US5292752A (en) 1989-12-21 1994-03-08 Merrell Dow Pharmaceuticals Inc. Antithrombotic compounds
DK0531410T3 (en) 1990-06-01 1995-01-30 Merrell Dow Pharma (+) - alpha- (2,3-Demethoxyphenyl) -1- (2- (4-fluorophenyl) ethyl) -4-piperidinemethanol
ATE145208T1 (en) 1990-07-06 1996-11-15 Yoshitomi Pharmaceutical CONDENSED THIOPHENE COMPOUNDS AND THEIR USE
KR100226954B1 (en) 1990-12-14 1999-10-15 슈테펜엘.네스비트 Piperidinyl benzimidazole derivatives, the pharmaceutical composition containing them and the process of them
US5231099A (en) 1991-04-15 1993-07-27 Du Pont Merck Pharmaceutical Company Use of sigma receptor antagonists to enhance the effects of antipsychotic drugs
DK0626968T3 (en) 1992-02-13 2001-12-31 Merrell Pharma Inc Thiacyclic piperidinyl derivatives
WO1998031800A2 (en) 1997-01-21 1998-07-23 Human Genome Sciences, Inc. Human proteins
DE19905823C1 (en) 1999-02-12 2000-06-08 Deutsches Krebsforsch Collimator for high energy radiation, e.g. for the treatment of tumors, comprises numerous opposing scree sections made of radiation absorbing material
EP1192257A2 (en) 1999-03-18 2002-04-03 Incyte Pharmaceuticals, Inc. Human regulators of intracellular phosphorylation

Similar Documents

Publication Publication Date Title
AU2001234175A1 (en) Novel cyclic amide derivatives
AU2001280187A1 (en) Cyclic amine derivatives
AU2001241128A1 (en) Novel amide compounds
AU2001241142A1 (en) Cyclic compounds
EG22695A (en) Novel phenyl-propargylether derivatives
AU2001280099A1 (en) 4-acylaminopyrazole derivatives
AU2001230584A1 (en) 1h-imidazopyridine derivatives
AU2001230537A1 (en) Pyridoxazine derivatives
AU2001281802A1 (en) 6-phenylpyrrolopyrimidinedione derivatives
AU2001278790A1 (en) 1h-imidazopyridine derivatives
AU2001234313A1 (en) Novel phenylheteroalkylamine derivatives
AU2001254661A1 (en) Aminosulfonylbiphenyl derivatives
AU2001230565A1 (en) Perfluoroisopropylbenzene derivatives
AU2002363600A1 (en) Novel phenyl-propargylether derivatives
AU2001242772A1 (en) 3-substituted-4-pyrimidone derivatives
AU2001280176A1 (en) Novel ester or amide derivatives
AU2001280120A1 (en) Cyclic peptide derivative
AU2001288484A1 (en) Novel metallotexaphyrin derivatives
AU2001246541A1 (en) Novel alpha-sulfin- and alpha-sulfonamino acid amide derivatives
AU2001276716A1 (en) Cyclic amine derivatives and use thereof
AU2001289782A1 (en) Pyrrolotriazolopyrimidinone derivatives
AU2001241084A1 (en) Imidazolylbenzophenone derivatives
SI1260512T1 (en) Novel cyclic amide derivatives
AU2320400A (en) Cyclic amine derivatives and uses thereof
AU2001228836A1 (en) Novel difluoroprostaglandin derivative