ATE528312T1 - METHOD FOR SYNTHESIS OF MACROLIDS - Google Patents
METHOD FOR SYNTHESIS OF MACROLIDSInfo
- Publication number
- ATE528312T1 ATE528312T1 AT07787934T AT07787934T ATE528312T1 AT E528312 T1 ATE528312 T1 AT E528312T1 AT 07787934 T AT07787934 T AT 07787934T AT 07787934 T AT07787934 T AT 07787934T AT E528312 T1 ATE528312 T1 AT E528312T1
- Authority
- AT
- Austria
- Prior art keywords
- macrolides
- making
- macrolids
- synthesis
- methods
- Prior art date
Links
Abstract
This invention relates to a method for making macrolides, and, in particular, to a method for making optionally substituted 20, 23-dipiperidinyl-5-O-mycaminosyl-tylonolide and derivatives thereof, as well as uses of macrolides to make medicaments, methods of treatment using macrolides, and methods for making intermediates that, inter alia, may be used to make macrolides.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US83406706P | 2006-07-28 | 2006-07-28 | |
EP06118159 | 2006-07-31 | ||
PCT/EP2007/057710 WO2008012343A2 (en) | 2006-07-28 | 2007-07-26 | Macrolide synthesis process |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE528312T1 true ATE528312T1 (en) | 2011-10-15 |
Family
ID=37547702
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT07787934T ATE528312T1 (en) | 2006-07-28 | 2007-07-26 | METHOD FOR SYNTHESIS OF MACROLIDS |
Country Status (8)
Country | Link |
---|---|
CN (1) | CN102875622B (en) |
AT (1) | ATE528312T1 (en) |
BR (1) | BRPI0715642C8 (en) |
ES (1) | ES2374950T3 (en) |
NZ (1) | NZ574193A (en) |
RU (1) | RU2450014C2 (en) |
SI (1) | SI2089408T1 (en) |
TW (1) | TWI397534B (en) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN104497082B (en) * | 2015-01-13 | 2017-12-12 | 中国兽医药品监察所 | A kind of synthetic method of tylonolide |
CN113121625B (en) * | 2019-12-31 | 2023-05-23 | 湖北龙翔药业科技股份有限公司 | Preparation method of tylosin |
CN116478217A (en) * | 2023-04-24 | 2023-07-25 | 济南久隆医药科技有限公司 | Continuous synthesis method of tylosin |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE667952A (en) * | 1964-08-05 | |||
JPS5896096A (en) * | 1981-11-30 | 1983-06-07 | Microbial Chem Res Found | 19-decarbonyl-4'-deoxymycaminosyl tylonolide derivative |
IL71032A0 (en) * | 1983-02-28 | 1984-05-31 | Lilly Co Eli | C-20 and c-23-modified macrolide derivatives |
US4629786A (en) * | 1983-02-28 | 1986-12-16 | Eli Lilly And Company | C-20- and C-23 modified macrolide derivatives |
US4921947A (en) * | 1986-03-31 | 1990-05-01 | Eli Lilly And Company | Process for preparing macrolide derivatives |
ES2213597T3 (en) * | 1999-08-30 | 2004-09-01 | Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai | MACROLID ANTIBIOTICS AND TREATMENT OF PASTEURELOSIS. |
US6506885B1 (en) * | 2001-09-27 | 2003-01-14 | The United States Of America As Represented By The Secretary Of Agriculture | Monoclonal antibodies to the drug tilmicosin and a method for detecting the same |
CN101506220B (en) * | 2006-07-28 | 2012-10-17 | 英特威国际有限公司 | Macrolide synthesis process |
-
2007
- 2007-07-26 AT AT07787934T patent/ATE528312T1/en not_active IP Right Cessation
- 2007-07-26 CN CN201210382136.4A patent/CN102875622B/en active Active
- 2007-07-26 ES ES07787934T patent/ES2374950T3/en active Active
- 2007-07-26 NZ NZ574193A patent/NZ574193A/en unknown
- 2007-07-26 TW TW96127367A patent/TWI397534B/en active
- 2007-07-26 BR BRPI0715642A patent/BRPI0715642C8/en active IP Right Grant
- 2007-07-26 SI SI200730813T patent/SI2089408T1/en unknown
- 2007-07-26 RU RU2009107167/04A patent/RU2450014C2/en active
Also Published As
Publication number | Publication date |
---|---|
BRPI0715642A2 (en) | 2013-07-09 |
CN102875622B (en) | 2016-12-07 |
BRPI0715642B8 (en) | 2020-06-30 |
RU2450014C2 (en) | 2012-05-10 |
NZ574193A (en) | 2011-09-30 |
TW200831524A (en) | 2008-08-01 |
ES2374950T3 (en) | 2012-02-23 |
SI2089408T1 (en) | 2012-02-29 |
BRPI0715642C8 (en) | 2020-07-28 |
CN102875622A (en) | 2013-01-16 |
RU2009107167A (en) | 2010-09-10 |
TWI397534B (en) | 2013-06-01 |
BRPI0715642B1 (en) | 2020-06-09 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |