ATE446965T1 - METHOD FOR PRODUCING FLUTICASONE PROPIONATES, IN PARTICULAR POLYMORPHO 1 - Google Patents

METHOD FOR PRODUCING FLUTICASONE PROPIONATES, IN PARTICULAR POLYMORPHO 1

Info

Publication number
ATE446965T1
ATE446965T1 AT03704541T AT03704541T ATE446965T1 AT E446965 T1 ATE446965 T1 AT E446965T1 AT 03704541 T AT03704541 T AT 03704541T AT 03704541 T AT03704541 T AT 03704541T AT E446965 T1 ATE446965 T1 AT E446965T1
Authority
AT
Austria
Prior art keywords
polymorpho
producing
propionates
fluticasone propionates
producing fluticasone
Prior art date
Application number
AT03704541T
Other languages
German (de)
Inventor
Steven John Coote
Rosalyn Kay Nice
Mark David Wipperman
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of ATE446965T1 publication Critical patent/ATE446965T1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
AT03704541T 2002-02-04 2003-02-03 METHOD FOR PRODUCING FLUTICASONE PROPIONATES, IN PARTICULAR POLYMORPHO 1 ATE446965T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0202564.1A GB0202564D0 (en) 2002-02-04 2002-02-04 Process
PCT/EP2003/001115 WO2003066653A2 (en) 2002-02-04 2003-02-03 Process for the production of fluticasone propionate, in particular of polymorphic form 1

Publications (1)

Publication Number Publication Date
ATE446965T1 true ATE446965T1 (en) 2009-11-15

Family

ID=9930366

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03704541T ATE446965T1 (en) 2002-02-04 2003-02-03 METHOD FOR PRODUCING FLUTICASONE PROPIONATES, IN PARTICULAR POLYMORPHO 1

Country Status (22)

Country Link
US (1) US20050222107A1 (en)
EP (1) EP1474436B1 (en)
JP (1) JP2005517019A (en)
KR (1) KR20040086331A (en)
CN (1) CN100338087C (en)
AR (1) AR038390A1 (en)
AT (1) ATE446965T1 (en)
AU (1) AU2003206836B2 (en)
BR (1) BR0307243A (en)
CA (1) CA2473896A1 (en)
CO (1) CO5611115A2 (en)
DE (1) DE60329824D1 (en)
GB (1) GB0202564D0 (en)
IS (1) IS7373A (en)
MX (1) MXPA04007530A (en)
NO (1) NO327138B1 (en)
NZ (1) NZ534320A (en)
PL (1) PL372214A1 (en)
RU (1) RU2333218C2 (en)
TW (1) TW200410982A (en)
WO (1) WO2003066653A2 (en)
ZA (1) ZA200405826B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL153462A0 (en) * 2002-12-16 2003-07-06 Chemagis Ltd Thiocarboxylic acid organic salts and processes utilizing the same
AU2013202843B2 (en) * 2006-06-14 2015-11-12 Generics [Uk] Limited Process for the preparation of S-fluoromethyl-6,9-difluoro-11-hydroxy-16-methyl-17-propionyloxy-3-oxo-androsta-1, 4-diene-17-carbothioate and intermediates
CA2835790C (en) * 2006-06-14 2017-05-16 Generics [Uk] Limited Novel process and intermediates
US8841442B2 (en) * 2010-09-01 2014-09-23 Cadila Healthcare Limited Process for preparing fluticasone propionate/furoate
AU2012282936B2 (en) * 2011-07-08 2016-11-10 Pfizer Limited Process for the preparation of fluticasone propionate form 1
US8765725B2 (en) 2012-05-08 2014-07-01 Aciex Therapeutics, Inc. Preparations of hydrophobic therapeutic agents, methods of manufacture and use thereof
CN104350063B (en) 2012-05-08 2018-01-05 尼科斯眼药公司 Preparation, its preparation method and the application of hydrophobic therapeutic agent
DE102012221219B4 (en) * 2012-11-20 2014-05-28 Jesalis Pharma Gmbh Process for increasing the particle size of crystalline drug microparticles
US9815865B2 (en) 2013-01-07 2017-11-14 Nicox Ophthalmics, Inc. Preparations of hydrophobic therapeutic agents, methods of manufacture and use thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2455976A1 (en) * 1974-11-27 1976-08-12 Merck Patent Gmbh PROSTIC ACID DERIVATIVES
PH24267A (en) * 1980-02-15 1990-05-29 Glaxo Group Ltd Androstane carbothioates and pharmaceutical compositions containing the same
US5783677A (en) * 1993-09-24 1998-07-21 Procter & Gamble Pharmaceuticals, Inc. Deoxy and oxygen-substituted sugar-containing 14-aminosteroid compounds
US5488188A (en) * 1994-09-29 1996-01-30 Merrell Dow Pharmaceuticals Inc. Process for the preparation of (E)-1-amino-2-(fluoromethylene)-4-(p-fluorophenyl)butane, novel processes for preparing an intermediate thereof, and novel intermediates thereof
GB9622173D0 (en) * 1996-10-24 1996-12-18 Glaxo Group Ltd Particulate Products
GB9925934D0 (en) * 1999-11-03 1999-12-29 Glaxo Group Ltd Novel apparatus and process
AR032361A1 (en) * 2000-08-05 2003-11-05 Glaxo Group Ltd DERIVATIVES OF ANDROSTAN AND SALTS AND SOLVATOS OF THE SAME, ITS USE FOR THE MANUFACTURE OF MEDICINES, PHARMACEUTICAL COMPOSITIONS THAT INCLUDE SUCH COMPOUNDS, PROCESS FOR THE PREPARATION OF SUCH COMPOUNDS, AND USEFUL INTERMEDIARIES IN THE PREPARATION OF SUCH COMPOUNDS

Also Published As

Publication number Publication date
CN1642969A (en) 2005-07-20
ZA200405826B (en) 2005-08-11
DE60329824D1 (en) 2009-12-10
WO2003066653A3 (en) 2003-12-24
EP1474436A2 (en) 2004-11-10
KR20040086331A (en) 2004-10-08
RU2333218C2 (en) 2008-09-10
CA2473896A1 (en) 2003-08-14
RU2004122928A (en) 2005-05-27
IS7373A (en) 2004-07-26
MXPA04007530A (en) 2004-11-10
NZ534320A (en) 2007-07-27
TW200410982A (en) 2004-07-01
AR038390A1 (en) 2005-01-12
NO327138B1 (en) 2009-05-04
WO2003066653A2 (en) 2003-08-14
US20050222107A1 (en) 2005-10-06
PL372214A1 (en) 2005-07-11
GB0202564D0 (en) 2002-03-20
NO20043664L (en) 2004-09-01
CO5611115A2 (en) 2006-02-28
BR0307243A (en) 2004-12-14
AU2003206836B2 (en) 2009-01-08
CN100338087C (en) 2007-09-19
AU2003206836A1 (en) 2003-09-02
JP2005517019A (en) 2005-06-09
EP1474436B1 (en) 2009-10-28

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