ATE363485T1 - BENZOTHIENO(3,2-C)PYRIDINES AS ALPHA2 ANTAGONISTS - Google Patents
BENZOTHIENO(3,2-C)PYRIDINES AS ALPHA2 ANTAGONISTSInfo
- Publication number
- ATE363485T1 ATE363485T1 AT99947469T AT99947469T ATE363485T1 AT E363485 T1 ATE363485 T1 AT E363485T1 AT 99947469 T AT99947469 T AT 99947469T AT 99947469 T AT99947469 T AT 99947469T AT E363485 T1 ATE363485 T1 AT E363485T1
- Authority
- AT
- Austria
- Prior art keywords
- benzothieno
- pyridines
- alpha2 antagonists
- alpha2
- antagonists
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Emergency Medicine (AREA)
- Psychology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP98203363 | 1998-10-06 |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE363485T1 true ATE363485T1 (en) | 2007-06-15 |
Family
ID=8234188
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT99947469T ATE363485T1 (en) | 1998-10-06 | 1999-10-01 | BENZOTHIENO(3,2-C)PYRIDINES AS ALPHA2 ANTAGONISTS |
Country Status (28)
Country | Link |
---|---|
US (2) | US6426350B1 (en) |
EP (1) | EP1117667B1 (en) |
JP (1) | JP4580555B2 (en) |
KR (1) | KR20010071828A (en) |
CN (1) | CN1158287C (en) |
AR (1) | AR023678A1 (en) |
AT (1) | ATE363485T1 (en) |
AU (1) | AU760226B2 (en) |
BG (1) | BG64625B1 (en) |
BR (1) | BR9913110A (en) |
CA (1) | CA2346084C (en) |
CZ (1) | CZ20011103A3 (en) |
DE (1) | DE69936219T2 (en) |
EE (1) | EE04835B1 (en) |
ES (1) | ES2288025T3 (en) |
HK (1) | HK1039113A1 (en) |
HU (1) | HUP0103612A3 (en) |
ID (1) | ID28280A (en) |
IL (2) | IL142442A0 (en) |
NO (1) | NO20011309L (en) |
NZ (1) | NZ509911A (en) |
PL (1) | PL347184A1 (en) |
RU (1) | RU2222542C2 (en) |
SK (1) | SK4312001A3 (en) |
TR (1) | TR200100954T2 (en) |
TW (1) | TWI251595B (en) |
UA (1) | UA70334C2 (en) |
WO (1) | WO2000020422A1 (en) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE494000T1 (en) * | 2002-03-08 | 2011-01-15 | Max Planck Gesellschaft | USE OF EGFR TRANSACTIVATION INHIBITORS FOR HUMAN CANCER |
CA2480266C (en) * | 2002-04-03 | 2011-07-12 | Orion Corporation | Use of an alpha2-adrenoreceptor antagonist for cns-related diseases |
EP1757605A4 (en) | 2004-04-12 | 2007-12-19 | Taisho Pharmaceutical Co Ltd | Cyclic amine compound |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3752820A (en) * | 1972-03-20 | 1973-08-14 | Colgate Palmolive Co | Substituted-1,2,3,4-tetrahydrobenzothieno(3,2-c)pyridine derivatives |
FR2570701B1 (en) * | 1984-09-27 | 1987-05-22 | Synthelabo | FURO (3,2-C) PYRIDINES DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
US4686226A (en) * | 1985-09-03 | 1987-08-11 | Merck & Co., Inc. | Substituted benzo[b]furo- and benzo[b]thieno quinolizines |
EP0339959A3 (en) * | 1988-04-27 | 1991-03-20 | Glaxo Group Limited | Lactam derivatives |
US5100891A (en) * | 1991-01-18 | 1992-03-31 | Hoechst-Roussel Pharmaceuticals Inc. | Substituted 1,2,3,4-tetrahydrocyclopent[b]indoles, 1,2,3,3a,4,8a-hexahydrocyclopent[B]indoles and related compounds |
ATE247114T1 (en) * | 1994-09-12 | 2003-08-15 | Lilly Co Eli | SEROTONERGIC MODULATORS |
JP3274579B2 (en) * | 1995-01-12 | 2002-04-15 | 住友製薬株式会社 | Agent for treating psychiatric symptoms associated with cerebrovascular disorders |
UA52681C2 (en) * | 1997-04-08 | 2003-01-15 | Янссен Фармацевтика Н.В. | Derivatives of 1,2,3,4-tetrahydro-benzofuro [3,2,-c] pyridine |
-
1999
- 1999-01-10 UA UA2001031998A patent/UA70334C2/en unknown
- 1999-10-01 NZ NZ509911A patent/NZ509911A/en unknown
- 1999-10-01 CZ CZ20011103A patent/CZ20011103A3/en unknown
- 1999-10-01 EE EEP200100206A patent/EE04835B1/en not_active IP Right Cessation
- 1999-10-01 CN CNB998116777A patent/CN1158287C/en not_active Expired - Fee Related
- 1999-10-01 PL PL99347184A patent/PL347184A1/en not_active Application Discontinuation
- 1999-10-01 DE DE69936219T patent/DE69936219T2/en not_active Expired - Lifetime
- 1999-10-01 EP EP99947469A patent/EP1117667B1/en not_active Expired - Lifetime
- 1999-10-01 KR KR1020017000400A patent/KR20010071828A/en active Search and Examination
- 1999-10-01 ES ES99947469T patent/ES2288025T3/en not_active Expired - Lifetime
- 1999-10-01 SK SK431-2001A patent/SK4312001A3/en unknown
- 1999-10-01 RU RU2001111753/04A patent/RU2222542C2/en not_active IP Right Cessation
- 1999-10-01 ID IDW20010781A patent/ID28280A/en unknown
- 1999-10-01 JP JP2000574534A patent/JP4580555B2/en not_active Expired - Fee Related
- 1999-10-01 TW TW088116899A patent/TWI251595B/en not_active IP Right Cessation
- 1999-10-01 BR BR9913110-2A patent/BR9913110A/en not_active Application Discontinuation
- 1999-10-01 CA CA2346084A patent/CA2346084C/en not_active Expired - Fee Related
- 1999-10-01 IL IL14244299A patent/IL142442A0/en active IP Right Grant
- 1999-10-01 US US09/806,432 patent/US6426350B1/en not_active Expired - Lifetime
- 1999-10-01 HU HU0103612A patent/HUP0103612A3/en unknown
- 1999-10-01 AU AU60899/99A patent/AU760226B2/en not_active Ceased
- 1999-10-01 TR TR2001/00954T patent/TR200100954T2/en unknown
- 1999-10-01 AT AT99947469T patent/ATE363485T1/en not_active IP Right Cessation
- 1999-10-01 WO PCT/EP1999/007418 patent/WO2000020422A1/en active IP Right Grant
- 1999-10-05 AR ARP990105039A patent/AR023678A1/en active IP Right Grant
-
2001
- 2001-03-12 BG BG105331A patent/BG64625B1/en unknown
- 2001-03-15 NO NO20011309A patent/NO20011309L/en not_active Application Discontinuation
- 2001-04-04 IL IL142442A patent/IL142442A/en not_active IP Right Cessation
- 2001-12-15 HK HK01108819A patent/HK1039113A1/en not_active IP Right Cessation
-
2002
- 2002-04-16 US US10/123,338 patent/US6774129B2/en not_active Expired - Lifetime
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |