ATE111469T1 - Pyrimido-benzothiazine mit lipoxygenase-hemmung. - Google Patents

Pyrimido-benzothiazine mit lipoxygenase-hemmung.

Info

Publication number
ATE111469T1
ATE111469T1 AT92901466T AT92901466T ATE111469T1 AT E111469 T1 ATE111469 T1 AT E111469T1 AT 92901466 T AT92901466 T AT 92901466T AT 92901466 T AT92901466 T AT 92901466T AT E111469 T1 ATE111469 T1 AT E111469T1
Authority
AT
Austria
Prior art keywords
pyrimido
benzothiazines
compounds
lipoxygenase inhibition
relates
Prior art date
Application number
AT92901466T
Other languages
English (en)
Inventor
Kaoru Shimada
Yuji Shishido
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of ATE111469T1 publication Critical patent/ATE111469T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT92901466T 1991-01-07 1991-12-16 Pyrimido-benzothiazine mit lipoxygenase-hemmung. ATE111469T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP3000159A JPH0739422B2 (ja) 1991-01-07 1991-01-07 新規ピリミド−ベンゾチアジン類および組成物

Publications (1)

Publication Number Publication Date
ATE111469T1 true ATE111469T1 (de) 1994-09-15

Family

ID=11466261

Family Applications (1)

Application Number Title Priority Date Filing Date
AT92901466T ATE111469T1 (de) 1991-01-07 1991-12-16 Pyrimido-benzothiazine mit lipoxygenase-hemmung.

Country Status (11)

Country Link
EP (1) EP0566592B1 (de)
JP (1) JPH0739422B2 (de)
AT (1) ATE111469T1 (de)
CA (1) CA2099558A1 (de)
DE (1) DE69104067T2 (de)
DK (1) DK0566592T3 (de)
ES (1) ES2059209T3 (de)
FI (1) FI933102A0 (de)
IE (1) IE64069B1 (de)
PT (1) PT99979A (de)
WO (1) WO1992012161A1 (de)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1175581A (en) * 1966-11-08 1969-12-23 Pfizer & Co C Pyrimidobenzothiazines and related Compounds
US4845083A (en) * 1983-10-05 1989-07-04 Merck Frosst Canada, Inc. Method of inhibiting mammalian leukotriene biosynthesis

Also Published As

Publication number Publication date
JPH04230690A (ja) 1992-08-19
EP0566592A1 (de) 1993-10-27
FI933102A (fi) 1993-07-06
CA2099558A1 (en) 1992-07-08
DE69104067T2 (de) 1995-02-02
IE920028A1 (en) 1992-07-15
DE69104067D1 (de) 1994-10-20
IE64069B1 (en) 1995-07-12
WO1992012161A1 (en) 1992-07-23
PT99979A (pt) 1993-01-29
ES2059209T3 (es) 1994-11-01
JPH0739422B2 (ja) 1995-05-01
FI933102A0 (fi) 1993-07-06
EP0566592B1 (de) 1994-09-14
DK0566592T3 (da) 1994-10-17

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee