AT359063B - METHOD FOR THE PRODUCTION OF NEW ISOTHIAZOLE PYRIDINES AND THEIR ACID ADDITION SALTS - Google Patents

METHOD FOR THE PRODUCTION OF NEW ISOTHIAZOLE PYRIDINES AND THEIR ACID ADDITION SALTS

Info

Publication number
AT359063B
AT359063B AT291977A AT291977A AT359063B AT 359063 B AT359063 B AT 359063B AT 291977 A AT291977 A AT 291977A AT 291977 A AT291977 A AT 291977A AT 359063 B AT359063 B AT 359063B
Authority
AT
Austria
Prior art keywords
pyridines
production
acid addition
addition salts
isothiazole
Prior art date
Application number
AT291977A
Other languages
German (de)
Other versions
ATA291977A (en
Original Assignee
Beecham Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group Ltd filed Critical Beecham Group Ltd
Publication of ATA291977A publication Critical patent/ATA291977A/en
Application granted granted Critical
Publication of AT359063B publication Critical patent/AT359063B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81Amides; Imides
    • C07D213/82Amides; Imides in position 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AT291977A 1976-04-28 1977-04-26 METHOD FOR THE PRODUCTION OF NEW ISOTHIAZOLE PYRIDINES AND THEIR ACID ADDITION SALTS AT359063B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB17165/76A GB1560726A (en) 1976-04-28 1976-04-28 Isothiazolo-pyridines

Publications (2)

Publication Number Publication Date
ATA291977A ATA291977A (en) 1980-03-15
AT359063B true AT359063B (en) 1980-10-27

Family

ID=10090431

Family Applications (1)

Application Number Title Priority Date Filing Date
AT291977A AT359063B (en) 1976-04-28 1977-04-26 METHOD FOR THE PRODUCTION OF NEW ISOTHIAZOLE PYRIDINES AND THEIR ACID ADDITION SALTS

Country Status (18)

Country Link
JP (1) JPS52131597A (en)
AT (1) AT359063B (en)
AU (1) AU2451277A (en)
BE (1) BE853779A (en)
CA (1) CA1073461A (en)
DE (1) DE2718707A1 (en)
DK (1) DK185577A (en)
ES (1) ES457993A1 (en)
FI (1) FI771236A (en)
FR (1) FR2349591A1 (en)
GB (1) GB1560726A (en)
HU (1) HU174416B (en)
IE (1) IE44873B1 (en)
IL (1) IL51812A0 (en)
NL (1) NL7704542A (en)
NZ (1) NZ183755A (en)
SE (1) SE7704800L (en)
ZA (1) ZA771963B (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU84091A1 (en) * 1982-04-16 1984-03-02 Oreal N-CARBAMOYL DERIVATIVES OF ISOTHIAZOLO- (5,4B) PYRIDINE ONE-3, THEIR PREPARATION METHOD AND THEIR USES AS BACTERICIDAL AND FUNGICIDAL AGENTS
LU84491A1 (en) * 1982-11-26 1984-06-13 Oreal ANTI-ACNE COMPOSITION CONTAINING AS AN ACTIVE COMPOUND A DERIVATIVE OF ISOTHIAZOLO- (5,4B) PYRIDINE ONE-3
FR2555450B1 (en) * 1983-11-24 1988-04-01 Oreal ANTI-ACNE COMPOSITION CONTAINING AS AN ACTIVE COMPOUND A DERIVATIVE OF ISOTHIAZOLO- (5,4B) PYRIDINE ONE-3
US5734081A (en) * 1994-08-05 1998-03-31 Warner-Lambert Company Arylthio compounds
US5620997A (en) * 1995-05-31 1997-04-15 Warner-Lambert Company Isothiazolones
US6001863A (en) * 1996-11-26 1999-12-14 Warner-Lambert Company Isothiazolones
JP4853911B2 (en) * 2006-09-26 2012-01-11 独立行政法人産業技術総合研究所 Method for producing isothiazolopyridin-3-one compound
JP4982790B2 (en) * 2006-09-26 2012-07-25 独立行政法人産業技術総合研究所 Method for producing isothiazolopyridin-3-one compound
JP4853910B2 (en) * 2006-09-26 2012-01-11 独立行政法人産業技術総合研究所 Method for producing isothiazolopyridin-3-one compound
FR2968661B1 (en) * 2010-12-14 2016-01-01 Oreal PROCESS FOR DEPIGMENTING KERATINIC MATERIALS USING THIOPYRIDINONE COMPOUNDS
US9938269B2 (en) * 2011-06-30 2018-04-10 Abbvie Inc. Inhibitor compounds of phosphodiesterase type 10A
FR3115207B1 (en) 2020-10-15 2022-10-07 Oreal Use of thiopyridinone compounds to prevent the formation of cutaneous blackheads

Also Published As

Publication number Publication date
GB1560726A (en) 1980-02-06
ZA771963B (en) 1978-03-29
AU2451277A (en) 1978-10-26
DK185577A (en) 1977-10-29
FR2349591B1 (en) 1980-02-01
SE7704800L (en) 1977-10-29
HU174416B (en) 1980-01-28
IE44873B1 (en) 1982-04-21
DE2718707A1 (en) 1977-11-10
IL51812A0 (en) 1977-06-30
BE853779A (en) 1977-10-20
FR2349591A1 (en) 1977-11-25
FI771236A (en) 1977-10-29
IE44873L (en) 1977-10-28
ES457993A1 (en) 1978-07-16
NL7704542A (en) 1977-11-01
NZ183755A (en) 1979-03-28
JPS52131597A (en) 1977-11-04
CA1073461A (en) 1980-03-11
ATA291977A (en) 1980-03-15

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Legal Events

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ELJ Ceased due to non-payment of the annual fee