AR126601A1 - PREPARATION OF THYAZOLYL-PIPERIDINYL COMPOUNDS CONTAINING PHENYLSULPHILIMINES OR SULFOXIMINES AND INTERMEDIATE THEREOF - Google Patents
PREPARATION OF THYAZOLYL-PIPERIDINYL COMPOUNDS CONTAINING PHENYLSULPHILIMINES OR SULFOXIMINES AND INTERMEDIATE THEREOFInfo
- Publication number
- AR126601A1 AR126601A1 ARP220102016A ARP220102016A AR126601A1 AR 126601 A1 AR126601 A1 AR 126601A1 AR P220102016 A ARP220102016 A AR P220102016A AR P220102016 A ARP220102016 A AR P220102016A AR 126601 A1 AR126601 A1 AR 126601A1
- Authority
- AR
- Argentina
- Prior art keywords
- formula
- preparation
- sulfoximines
- compounds containing
- thyazolyl
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 150000003839 salts Chemical class 0.000 abstract 4
- 238000000034 method Methods 0.000 abstract 3
- PPBRXRYQALVLMV-UHFFFAOYSA-N Styrene Chemical compound C=CC1=CC=CC=C1 PPBRXRYQALVLMV-UHFFFAOYSA-N 0.000 abstract 2
- GPLUYPFUSVDDII-UHFFFAOYSA-N N=[S+]C1=CC=CC=C1 Chemical class N=[S+]C1=CC=CC=C1 GPLUYPFUSVDDII-UHFFFAOYSA-N 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 150000002923 oximes Chemical class 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
- 125000005555 sulfoximide group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Abstract
La presente invención divulga un procedimiento para la preparación de compuestos de tiazolil-piperidinil que contienen fenil sulfiliminas o sulfoximinas de fórmula (1) en donde, R¹, R², Rᵃ, Q, n y m son como se define en la descripción e intermedios para la preparación del compuesto de fórmula (1) o sales del mismo. Reivindicación 17: Un procedimiento para preparar un compuesto de fórmula (3) de acuerdo con la reivindicación 16, en donde dicho procedimiento comprende la etapa de: hacer reaccionar un estireno de fórmula (5) o sales del mismo en donde, Q, R² y m son como se han definido anteriormente, con una oxima de fórmula (4) o sales de la misma en presencia de una base y un disolvente adecuados en donde, X es halógeno, para obtener el compuesto de fórmula (3) o sales del mismo.The present invention discloses a process for the preparation of thiazolyl-piperidinyl compounds containing phenyl sulfilimines or sulfoximines of formula (1) wherein, R¹, R², Rᵃ, Q, n and m are as defined in the description and intermediates for the preparation of the compound of formula (1) or salts thereof. Claim 17: A procedure for preparing a compound of formula (3) according to claim 16, wherein said procedure comprises the step of: reacting a styrene of formula (5) or salts thereof wherein, Q, R² and m are as defined above, with an oxime of formula (4) or salts thereof in the presence of a suitable base and solvent wherein, X is halogen, to obtain the compound of formula (3) or salts thereof.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN202111034193 | 2021-07-29 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR126601A1 true AR126601A1 (en) | 2023-10-25 |
Family
ID=83149194
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP220102016A AR126601A1 (en) | 2021-07-29 | 2022-07-28 | PREPARATION OF THYAZOLYL-PIPERIDINYL COMPOUNDS CONTAINING PHENYLSULPHILIMINES OR SULFOXIMINES AND INTERMEDIATE THEREOF |
Country Status (3)
| Country | Link |
|---|---|
| AR (1) | AR126601A1 (en) |
| TW (1) | TW202312878A (en) |
| WO (1) | WO2023007429A1 (en) |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008013622A2 (en) | 2006-07-27 | 2008-01-31 | E. I. Du Pont De Nemours And Company | Fungicidal azocyclic amides |
| US20120122928A1 (en) | 2010-08-11 | 2012-05-17 | Bayer Cropscience Ag | Heteroarylpiperidine and -Piperazine Derivatives as Fungicides |
| WO2016024350A1 (en) | 2014-08-13 | 2016-02-18 | 株式会社エス・ディー・エス バイオテック | Condensed 11-membered ring compounds and agricultural and horticultural fungicide containing same |
| US20160242416A1 (en) * | 2015-02-23 | 2016-08-25 | E I Du Pont De Nemours And Company | Fungicidal isoxazoline carbinols |
| AR120377A1 (en) | 2019-11-11 | 2022-02-09 | Pi Industries Ltd | HETEROAROMATIC DERIVATIVES OF SULFILIMINES OR SULFOXIMINES WITH FUNGICIDAL ACTIVITY |
-
2022
- 2022-07-28 AR ARP220102016A patent/AR126601A1/en unknown
- 2022-07-28 WO PCT/IB2022/057001 patent/WO2023007429A1/en unknown
- 2022-07-29 TW TW111128688A patent/TW202312878A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2023007429A1 (en) | 2023-02-02 |
| TW202312878A (en) | 2023-04-01 |
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