AR124698A1 - TRICYCLIC DERIVATIVES USEFUL AS INHIBITORS OF PARP7 - Google Patents

TRICYCLIC DERIVATIVES USEFUL AS INHIBITORS OF PARP7

Info

Publication number
AR124698A1
AR124698A1 ARP220100147A ARP220100147A AR124698A1 AR 124698 A1 AR124698 A1 AR 124698A1 AR P220100147 A ARP220100147 A AR P220100147A AR P220100147 A ARP220100147 A AR P220100147A AR 124698 A1 AR124698 A1 AR 124698A1
Authority
AR
Argentina
Prior art keywords
parp7
inhibitors
derivatives useful
tricyclic derivatives
compound
Prior art date
Application number
ARP220100147A
Other languages
Spanish (es)
Inventor
Haijun Li
Mingming Chen
Di Kang
Qinglong Li
Lei Zhang
Man Yan
Wei Long
Yanping Wang
Hao Zhang
Cunbo Ma
Amin Li
Original Assignee
Jacobio Pharmaceuticals Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Jacobio Pharmaceuticals Co Ltd filed Critical Jacobio Pharmaceuticals Co Ltd
Publication of AR124698A1 publication Critical patent/AR124698A1/en

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  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La invención se relaciona con un compuesto de formula (1) que inhibe la actividad de PARP7, un estereoisómero del mismo, un derivado deuterado del mismo, o una sal farmacéuticamente aceptable del mismo, un intermediario para preparar el compuesto, un proceso para preparar el compuesto, una composición que lo comprende, y los métodos de uso del mismo.The invention relates to a compound of formula (1) that inhibits the activity of PARP7, a stereoisomer thereof, a deuterated derivative thereof, or a pharmaceutically acceptable salt thereof, an intermediate for preparing the compound, a process for preparing the compound, a composition comprising it, and methods of use thereof.

ARP220100147A 2021-02-09 2022-01-26 TRICYCLIC DERIVATIVES USEFUL AS INHIBITORS OF PARP7 AR124698A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CN2021076144 2021-02-09

Publications (1)

Publication Number Publication Date
AR124698A1 true AR124698A1 (en) 2023-04-26

Family

ID=86380110

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP220100147A AR124698A1 (en) 2021-02-09 2022-01-26 TRICYCLIC DERIVATIVES USEFUL AS INHIBITORS OF PARP7

Country Status (1)

Country Link
AR (1) AR124698A1 (en)

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