AR120803A1 -
SOLID FORMS OF 2-[3-[4-AMINO-3-(2-FLUORO-4-PHENOXI-PHENYL)PYRAZOLO[3,4-D]PYRIMIDIN-1-IL]PIPERIDINE-1-CARBONYL]-4-METHYL -4-[4-(OXETAN-3-IL)PIPERAZIN-1-IL]PENT-2-ENENITRILE
- Google Patents
SOLID FORMS OF 2-[3-[4-AMINO-3-(2-FLUORO-4-PHENOXI-PHENYL)PYRAZOLO[3,4-D]PYRIMIDIN-1-IL]PIPERIDINE-1-CARBONYL]-4-METHYL -4-[4-(OXETAN-3-IL)PIPERAZIN-1-IL]PENT-2-ENENITRILE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Principia Biopharma IncfiledCriticalPrincipia Biopharma Inc
Publication of AR120803A1publicationCriticalpatent/AR120803A1/en
Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Abstract
Formas sólidas del compuesto de fórmula (1) se describen. También se describen composiciones farmacéuticas que los comprenden, métodos para tratar desórdenes y condiciones mediadas por actividad de BTK usando los mismos, y métodos para preparar el Compuesto de fórmula (1) y formas cristalinas de este.Solid forms of the compound of formula (1) are described. Pharmaceutical compositions comprising them, methods of treating disorders and conditions mediated by BTK activity using the same, and methods of preparing the Compound of formula (1) and crystalline forms thereof are also described.
ARP200103533A2019-12-202020-12-17
SOLID FORMS OF 2-[3-[4-AMINO-3-(2-FLUORO-4-PHENOXI-PHENYL)PYRAZOLO[3,4-D]PYRIMIDIN-1-IL]PIPERIDINE-1-CARBONYL]-4-METHYL -4-[4-(OXETAN-3-IL)PIPERAZIN-1-IL]PENT-2-ENENITRILE
AR120803A1
(en)
SOLID FORMS OF 2-[3-[4-AMINO-3-(2-FLUORO-4-PHENOXI-PHENYL)PYRAZOLO[3,4-D]PYRIMIDIN-1-IL]PIPERIDINE-1-CARBONYL]-4-METHYL -4-[4-(OXETAN-3-IL)PIPERAZIN-1-IL]PENT-2-ENENITRILE
Crystal forms of 2-[3-[4-amino-3-(2-fluoro-4-phenoxy-phenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-carbonyl]- 4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile