AR117467A2 - PROCESSES FOR PREPARING ISOQUINOLINONES AND SOLID FORMS OF ISOQUINOLINONES - Google Patents
PROCESSES FOR PREPARING ISOQUINOLINONES AND SOLID FORMS OF ISOQUINOLINONESInfo
- Publication number
- AR117467A2 AR117467A2 ARP190103791A ARP190103791A AR117467A2 AR 117467 A2 AR117467 A2 AR 117467A2 AR P190103791 A ARP190103791 A AR P190103791A AR P190103791 A ARP190103791 A AR P190103791A AR 117467 A2 AR117467 A2 AR 117467A2
- Authority
- AR
- Argentina
- Prior art keywords
- isoquinolinones
- kinase activity
- processes
- preparing
- solid forms
- Prior art date
Links
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Se describen en la presente polimorfos de compuestos químicos que modulan la actividad de quinasa, que incluye la actividad de la PI3 quinasa, y compuestos, composiciones farmacéuticas, y métodos para el tratamiento de enfermedades y afecciones asociadas con la actividad de quinasa, que incluye la actividad de la PI3 quinasa. Además se proporcionan en la presente procedimientos para la preparación de compuestos, polimorfos de los mismos, y composiciones farmacéuticas de los mismos. Reivindicación 1: Un compuesto de fórmula (1), donde el compuesto es el polimorfo que se proporciona en la presente es Forma B, Forma C, Forma D, Forma E, Forma F, Forma G, Forma H, Forma I, Forma J, o una forma amorfa de un compuesto de fórmula (1), o una sal, solvato, o hidrato del mismo; o una mezcla de dos o más de los mismos.Described herein are polymorphs of chemical compounds that modulate kinase activity, including PI3 kinase activity, and compounds, pharmaceutical compositions, and methods for treating diseases and conditions associated with kinase activity, including the PI3 kinase activity. Further provided herein are methods for the preparation of compounds, polymorphs thereof, and pharmaceutical compositions thereof. Claim 1: A compound of formula (1), wherein the compound is the polymorph provided herein is Form B, Form C, Form D, Form E, Form F, Form G, Form H, Form I, Form J , or an amorphous form of a compound of formula (1), or a salt, solvate, or hydrate thereof; or a mixture of two or more of them.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161431304P | 2011-01-10 | 2011-01-10 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR117467A2 true AR117467A2 (en) | 2021-08-11 |
Family
ID=77568205
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP190103791A AR117467A2 (en) | 2011-01-10 | 2019-12-19 | PROCESSES FOR PREPARING ISOQUINOLINONES AND SOLID FORMS OF ISOQUINOLINONES |
Country Status (1)
| Country | Link |
|---|---|
| AR (1) | AR117467A2 (en) |
-
2019
- 2019-12-19 AR ARP190103791A patent/AR117467A2/en unknown
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