AR113298A2 - METHOD FOR PREPARING A BRIDGED DERIVATIVE OF PIVALATE FROM SPOOLAMINE - Google Patents

METHOD FOR PREPARING A BRIDGED DERIVATIVE OF PIVALATE FROM SPOOLAMINE

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Publication number
AR113298A2
AR113298A2 ARP180101047A ARP180101047A AR113298A2 AR 113298 A2 AR113298 A2 AR 113298A2 AR P180101047 A ARP180101047 A AR P180101047A AR P180101047 A ARP180101047 A AR P180101047A AR 113298 A2 AR113298 A2 AR 113298A2
Authority
AR
Argentina
Prior art keywords
preparing
spoolamine
pivalate
bridged derivative
derivative
Prior art date
Application number
ARP180101047A
Other languages
Spanish (es)
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of AR113298A2 publication Critical patent/AR113298A2/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

Reivindicación 1: Un método para preparar un compuesto de fórmula (1), que comprende hacer reaccionar escopolamina o un derivado de la misma.Claim 1: A method for preparing a compound of formula (1), which comprises reacting scopolamine or a derivative thereof.

ARP180101047A 2015-09-04 2018-04-24 METHOD FOR PREPARING A BRIDGED DERIVATIVE OF PIVALATE FROM SPOOLAMINE AR113298A2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562214727P 2015-09-04 2015-09-04

Publications (1)

Publication Number Publication Date
AR113298A2 true AR113298A2 (en) 2020-04-08

Family

ID=60452274

Family Applications (9)

Application Number Title Priority Date Filing Date
ARP160102711A AR105924A1 (en) 2015-09-04 2016-09-05 THERAPEUTIC COMPOUNDS AND SYNTHESIS
ARP160102710A AR105923A1 (en) 2015-09-04 2016-09-05 THERAPEUTIC COMPOUNDS FOR PAIN AND SYNTHESIS OF THESE
ARP160102708A AR105921A1 (en) 2015-09-04 2016-09-05 THERAPEUTIC COMPOUNDS FOR PAIN AND SYNTHESIS OF THESE
ARP160102707A AR105920A1 (en) 2015-09-04 2016-09-05 THERAPEUTIC COMPOUND FOR THE PAIN AND SYNTHESIS OF THE COMPOUND
ARP160102709A AR105922A1 (en) 2015-09-04 2016-09-05 1 - ((6-METOXINAFTALEN-2-IL) METHYL) -4- (3,3,3-TRIFLUOROPROPANOIL) OCTAHIDRO-1H-2,6-METANOPIRROLO [3,2-B] PIRIDIN-3-IL-USEFUL PIVALATE IN PAIN TREATMENT
ARP180101035A AR111416A2 (en) 2015-09-04 2018-04-23 THERAPEUTIC COMPOUND FOR THE PAIN AND SYNTHESIS OF THE COMPOUND
ARP180101047A AR113298A2 (en) 2015-09-04 2018-04-24 METHOD FOR PREPARING A BRIDGED DERIVATIVE OF PIVALATE FROM SPOOLAMINE
ARP180101061A AR111423A2 (en) 2015-09-04 2018-04-25 THERAPEUTIC COMPOUNDS FOR PAIN AND SYNTHESIS OF THESE
ARP180101062A AR111424A2 (en) 2015-09-04 2018-04-25 PREPARATION METHOD OF 1 - ((6-METOXINAFTALEN-2-IL) METHYL) -4- (3,3,3-TRIFLUROPROPANOL) OCTAHIDRO-1H-2,6-METANOPIRROLO [3,2-B] PIRIDIN-3- IL PIVALATO

Family Applications Before (6)

Application Number Title Priority Date Filing Date
ARP160102711A AR105924A1 (en) 2015-09-04 2016-09-05 THERAPEUTIC COMPOUNDS AND SYNTHESIS
ARP160102710A AR105923A1 (en) 2015-09-04 2016-09-05 THERAPEUTIC COMPOUNDS FOR PAIN AND SYNTHESIS OF THESE
ARP160102708A AR105921A1 (en) 2015-09-04 2016-09-05 THERAPEUTIC COMPOUNDS FOR PAIN AND SYNTHESIS OF THESE
ARP160102707A AR105920A1 (en) 2015-09-04 2016-09-05 THERAPEUTIC COMPOUND FOR THE PAIN AND SYNTHESIS OF THE COMPOUND
ARP160102709A AR105922A1 (en) 2015-09-04 2016-09-05 1 - ((6-METOXINAFTALEN-2-IL) METHYL) -4- (3,3,3-TRIFLUOROPROPANOIL) OCTAHIDRO-1H-2,6-METANOPIRROLO [3,2-B] PIRIDIN-3-IL-USEFUL PIVALATE IN PAIN TREATMENT
ARP180101035A AR111416A2 (en) 2015-09-04 2018-04-23 THERAPEUTIC COMPOUND FOR THE PAIN AND SYNTHESIS OF THE COMPOUND

Family Applications After (2)

Application Number Title Priority Date Filing Date
ARP180101061A AR111423A2 (en) 2015-09-04 2018-04-25 THERAPEUTIC COMPOUNDS FOR PAIN AND SYNTHESIS OF THESE
ARP180101062A AR111424A2 (en) 2015-09-04 2018-04-25 PREPARATION METHOD OF 1 - ((6-METOXINAFTALEN-2-IL) METHYL) -4- (3,3,3-TRIFLUROPROPANOL) OCTAHIDRO-1H-2,6-METANOPIRROLO [3,2-B] PIRIDIN-3- IL PIVALATO

Country Status (1)

Country Link
AR (9) AR105924A1 (en)

Also Published As

Publication number Publication date
AR111423A2 (en) 2019-07-10
AR105924A1 (en) 2017-11-22
AR105921A1 (en) 2017-11-22
AR105920A1 (en) 2017-11-22
AR111416A2 (en) 2019-07-10
AR105922A1 (en) 2017-11-22
AR111424A2 (en) 2019-07-10
AR105923A1 (en) 2017-11-22

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