AR110371A1 - Formulación de comprimido farmacéutico - Google Patents

Formulación de comprimido farmacéutico

Info

Publication number
AR110371A1
AR110371A1 ARP170103512A ARP170103512A AR110371A1 AR 110371 A1 AR110371 A1 AR 110371A1 AR P170103512 A ARP170103512 A AR P170103512A AR P170103512 A ARP170103512 A AR P170103512A AR 110371 A1 AR110371 A1 AR 110371A1
Authority
AR
Argentina
Prior art keywords
heart failure
formulation
pharmaceutical tablets
hfref
hfpef
Prior art date
Application number
ARP170103512A
Other languages
English (en)
Inventor
Stroyer Anke Dr
Schwer Christine Dr
Pfeffer Michael Dr
Lobback Carmen Dr
Ide Katrin Dr
Serno Peter Dr
Original Assignee
Bayer Pharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Pharma AG filed Critical Bayer Pharma AG
Publication of AR110371A1 publication Critical patent/AR110371A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hospice & Palliative Care (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Medicinal Preparation (AREA)

Abstract

Formulación de comprimido farmacéutico que comprende 2-{4-[2-({[2-(4-clorofenil)-1,3-tiazol-4-il]metil}sulfanil)-3,5-diciano-6-(pirrolidin-1-il)piridin-4-il]fenoxi}etil-L-alanil-L-alaninato (neladenoson bialanato) en la forma de una de sus sales, en donde libera el ingrediente activo rápidamente, y a procesos para su producción, al uso de este como un medicamento, y al uso de este para la profilaxis y/o tratamiento de trastornos cardiovasculares, por ejemplo insuficiencia cardíaca crónica agravada, insuficiencia cardíaca con fracción de eyección del ventrículo izquierdo reducida o conservada (HFrEF o HFpEF), angina pectoris y lesión isquémica durante un síndrome coronario agudo.
ARP170103512A 2016-12-16 2017-12-14 Formulación de comprimido farmacéutico AR110371A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP16204750 2016-12-16

Publications (1)

Publication Number Publication Date
AR110371A1 true AR110371A1 (es) 2019-03-20

Family

ID=57614148

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP170103512A AR110371A1 (es) 2016-12-16 2017-12-14 Formulación de comprimido farmacéutico

Country Status (4)

Country Link
AR (1) AR110371A1 (es)
TW (1) TW201836592A (es)
UY (1) UY37525A (es)
WO (1) WO2018108884A1 (es)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7807715B2 (en) 2006-06-09 2010-10-05 Ucb Pharma Gmbh Pharmaceutical compositions comprising fesoterodine
DE102009006602A1 (de) 2009-01-29 2010-08-05 Bayer Schering Pharma Aktiengesellschaft Alkylamino-substituierte Dicyanopyridine und deren Aminosäureester-Prodrugs
BR112017023852A2 (pt) 2015-05-06 2018-07-17 Bayer Pharma Aktiengesellschaft Processo para preparar monocloridrato de l- alaninato de 2-{4-[2-({[2-(4-clorofenil)-1,3-tiazol-4-il] metil}sulfanil)-3,5-diciano-6-(pirrolidin-1-il)piridin-4- il]fenoxi}etil-l-alanila.

Also Published As

Publication number Publication date
UY37525A (es) 2018-06-29
TW201836592A (zh) 2018-10-16
WO2018108884A1 (de) 2018-06-21

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