AR103632A2 - BENCIMIDAZOL DERIVATIVES - Google Patents
BENCIMIDAZOL DERIVATIVESInfo
- Publication number
- AR103632A2 AR103632A2 ARP160100340A ARP160100340A AR103632A2 AR 103632 A2 AR103632 A2 AR 103632A2 AR P160100340 A ARP160100340 A AR P160100340A AR P160100340 A ARP160100340 A AR P160100340A AR 103632 A2 AR103632 A2 AR 103632A2
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- hydrogen
- membered heterocyclyl
- independently
- nr16r17
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Reivindicación 1: Un compuesto de fórmula (1), en la que: cada R¹ es independientemente halo, alquilo C₁₋₆, alcoxi C₁₋₆, -CF₃, -CN, o -NR¹⁶R¹⁷; R² es hidrógeno o alquilo C₁₋₆; R³B es hidrógeno, alquilo C₁₋₆, -(CH₂)ₜarilo C₆₋₁₂, o -(CH₂)ₜcarbociclilo C₃₋₁₂; R⁴ es hidrógeno o alquilo C₁₋₆; R¹⁰ es -(CH₂)ₜarilo C₆₋₁₂ o -(CH₂)ₜ(heterociclilo de 4 a 14 miembros), en los que cada uno de dichos arilo C₆₋₁₂ y (heterociclilo de 4 a 14 miembros) está opcionalmente sustituido con de 1 a 5 sustituyentes cada uno de los cuales se selecciona independientemente de -alquil C₁₋₆, -CN, halo, -CF₃, -OCF₃, -NR¹⁶R¹⁷, alcoxi C₁₋₆, -NO₂, -(CH₂)ₜarilo C₆₋₁₂, -C(O)alquilo C₁₋₆, -C(O)CF₃, azido, (heterociclilo de 4 a 12 miembros), y -S(alquilo C₁₋₆); cada R¹⁶ y R¹⁷ está independientemente seleccionado de hidrógeno y alquilo C₁₋₆; n es 0, 1, 2, 3, ó 4; y cada t es independientemente 0, 1, ó 2; o una sal farmacéuticamente aceptable del mismo.Claim 1: A compound of formula (1), wherein: each R¹ is independently halo, C alquilo alkyl, C₁₋₆ alkoxy, -CF₃, -CN, or -NR¹⁶R¹⁷; R² is hydrogen or C₁₋₆ alkyl; R³B is hydrogen, C₁₋₆ alkyl, - (CH₂) C₆₋₁₂aryl, or - (CH₂) C₃₋₁₂carbocyclyl; R⁴ is hydrogen or C₁₋₆ alkyl; R¹⁰ is - (CH₂) ₜaryl C₆₋₁₂ or - (CH₂) ₜ (4 to 14-membered heterocyclyl), in which each of said C₆₋₁₂ and (4 to 14-membered heterocyclyl) is optionally substituted with 1 to 5 substituents each of which is independently selected from -C₁₋₆ alkyl, -CN, halo, -CF₃, -OCF₃, -NR¹⁶R¹⁷, C₁₋₆ alkoxy, -NO₂, - (CH₂) Ciloaryl, -C (O) C₁₋₆ alkyl, -C (O) CF₃, azido, (4-12 membered heterocyclyl), and -S (C₁₋₆ alkyl); each R¹⁶ and R¹⁷ is independently selected from hydrogen and C₁₋₆ alkyl; n is 0, 1, 2, 3, or 4; and each t is independently 0, 1, or 2; or a pharmaceutically acceptable salt thereof.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US94728707P | 2007-06-29 | 2007-06-29 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR103632A2 true AR103632A2 (en) | 2017-05-24 |
Family
ID=43038355
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP160100340A AR103632A2 (en) | 2007-06-29 | 2016-02-05 | BENCIMIDAZOL DERIVATIVES |
Country Status (3)
| Country | Link |
|---|---|
| AR (1) | AR103632A2 (en) |
| UA (1) | UA93313C2 (en) |
| ZA (1) | ZA200908626B (en) |
-
2008
- 2008-06-16 UA UAA200912326A patent/UA93313C2/en unknown
-
2009
- 2009-12-04 ZA ZA200908626A patent/ZA200908626B/en unknown
-
2016
- 2016-02-05 AR ARP160100340A patent/AR103632A2/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200908626B (en) | 2010-08-25 |
| UA93313C2 (en) | 2011-01-25 |
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