AR096803A1 - BENCIL-1H-PIRAZOLO [3,4-B] PIRIDINES AND ITS USE - Google Patents
BENCIL-1H-PIRAZOLO [3,4-B] PIRIDINES AND ITS USEInfo
- Publication number
- AR096803A1 AR096803A1 ARP140102484A ARP140102484A AR096803A1 AR 096803 A1 AR096803 A1 AR 096803A1 AR P140102484 A ARP140102484 A AR P140102484A AR P140102484 A ARP140102484 A AR P140102484A AR 096803 A1 AR096803 A1 AR 096803A1
- Authority
- AR
- Argentina
- Prior art keywords
- fluorine
- represents hydrogen
- oxides
- prevention
- salts
- Prior art date
Links
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente solicitud se refiere a bencil-1H-pirazoIo[3,4-b]piridinas, a procedimientos para su preparación, a su uso solas o en combinaciones para el tratamiento y/o la prevención de enfermedades así como a su uso para la preparación de medicamentos para el tratamiento y/o la prevención de enfermedades, en particular para el tratamiento y/o la prevención de enfermedades cardiocirculatorias. Reivindicación 1: Compuesto de la fórmula (1) en la que R¹ representa hidrógeno o flúor, R² representa hidrógeno o flúor, R³ representa hidrógeno, cloro o flúor, R⁴ representa hidrógeno, cloro, flúor o metilo, con la condición que al menos dos de los restos R¹, R², R³ o R⁴ sean diferentes de hidrógeno, R⁵ representa hidrógeno o flúor, R⁶ representa metilo, R⁷ representa metilo, o R⁶ y R⁷ junto con el átomo de carbono al que están unidos, forman un anillo de ciclopropilo, así como sus N-óxidos, sales, solvatos, sales de los N-óxidos y solvatos de los N-óxidos y sales.The present application relates to benzyl-1 H -pyrazo [3,4-b] pyridines, processes for their preparation, their use alone or in combinations for the treatment and / or prevention of diseases as well as their use for preparation of medicaments for the treatment and / or prevention of diseases, in particular for the treatment and / or prevention of cardiocirculatory diseases. Claim 1: Compound of the formula (1) wherein R¹ represents hydrogen or fluorine, R² represents hydrogen or fluorine, R³ represents hydrogen, chlorine or fluorine, R⁴ represents hydrogen, chlorine, fluorine or methyl, with the condition that at least two of the residues R,, R², R³ or R⁴ are different from hydrogen, R⁵ represents hydrogen or fluorine, R⁶ represents methyl, R⁷ represents methyl, or R⁶ and R⁷ together with the carbon atom to which they are attached, form a cyclopropyl ring, as well as its N-oxides, salts, solvates, salts of the N-oxides and solvates of the N-oxides and salts.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP13175889 | 2013-07-10 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR096803A1 true AR096803A1 (en) | 2016-02-03 |
Family
ID=48747469
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP140102484A AR096803A1 (en) | 2013-07-10 | 2014-07-03 | BENCIL-1H-PIRAZOLO [3,4-B] PIRIDINES AND ITS USE |
Country Status (2)
Country | Link |
---|---|
AR (1) | AR096803A1 (en) |
MA (1) | MA38775A1 (en) |
-
2014
- 2014-07-03 AR ARP140102484A patent/AR096803A1/en unknown
- 2014-07-08 MA MA38775A patent/MA38775A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
MA38775A1 (en) | 2017-07-31 |
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