AR090809A1 - BICYCLE COMPOUND - Google Patents

BICYCLE COMPOUND

Info

Publication number
AR090809A1
AR090809A1 ARP130101351A ARP130101351A AR090809A1 AR 090809 A1 AR090809 A1 AR 090809A1 AR P130101351 A ARP130101351 A AR P130101351A AR P130101351 A ARP130101351 A AR P130101351A AR 090809 A1 AR090809 A1 AR 090809A1
Authority
AR
Argentina
Prior art keywords
optionally substituted
ring
hydrogen atom
group
substituent
Prior art date
Application number
ARP130101351A
Other languages
Spanish (es)
Inventor
Matsunaga Nobuyuki
Fujimori Ikuo
Toyofuku Kyoko
Yamashita Tohru
Fujimoto Takuya
Mizojiri Ryo
Yonemori Kazuko
hirose Hideki
Ikeda Zenichi
Yasuma Tsuneo
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/JP2012/077357 external-priority patent/WO2013061962A1/en
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of AR090809A1 publication Critical patent/AR090809A1/en

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Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Reivindicación 1: Un compuesto representado por la fórmula (1) caracterizado porque R¹ es un grupo representado por la fórmula: -COR² donde R² es un átomo de hidrógeno o un sustituyente, o un grupo anular aromático de 5 ó 6 miembros opcionalmente sustituido; R³ es un grupo alquilo C₁₋₆ opcionalmente sustituido con átomos de halógeno, o un grupo cicloalquilo C₃₋₆ opcionalmente sustituido; R⁴ᵃ y R⁴ᵇ son de modo independiente un átomo de hidrógeno o un sustituyente; X es O, CO, CR⁵ᵃR⁵ᵇ (donde R⁵ᵃ y R⁵ᵇ son de modo independiente un átomo de hidrógeno o un sustituyente), NR⁵ᶜ (donde R⁵ᶜ es un átomo de hidrógeno o un grupo alquilo C₁₋₆ opcionalmente sustituido, S, SO, o S(O)₂); anillo A es un anillo aromático de 5 ó 6 miembros también opcionalmente sustituido; anillo P es un heterociclo aromático de 5 miembros también opcionalmente sustituido; anillo Q es un anillo de 5 a 7 miembros también opcionalmente sustituido; y R⁶ es un grupo alquilo C₁₋₆ opcionalmente sustituido o un grupo cicloalquilo C₃₋₆ opcionalmente sustituido; o una de sus sales.Claim 1: A compound represented by the formula (1) characterized in that R¹ is a group represented by the formula: -COR² where R² is a hydrogen atom or a substituent, or an optionally substituted 5 or 6-membered aromatic ring group; R³ is an optionally substituted C₁₋₆ alkyl group with halogen atoms, or an optionally substituted C₃₋₆ cycloalkyl group; R⁴ᵃ and R⁴ᵇ are independently a hydrogen atom or a substituent; X is O, CO, CR⁵ᵃR⁵ᵇ (where R⁵ᵃ and R⁵ᵇ are independently a hydrogen atom or a substituent), NR⁵ᶜ (where R⁵ᶜ is a hydrogen atom or an optionally substituted C₁₋₆ alkyl group, S, SO, or S (O) ₂); Ring A is an optionally substituted 5 or 6-membered aromatic ring; P ring is a 5-membered aromatic heterocycle also optionally substituted; ring Q is a 5 to 7 member ring also optionally substituted; and R⁶ is an optionally substituted C₁₋₆ alkyl group or an optionally substituted C₃₋₆ cycloalkyl group; or one of its salts.

ARP130101351A 2012-05-29 2013-04-23 BICYCLE COMPOUND AR090809A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2012122471 2012-05-29
PCT/JP2012/077357 WO2013061962A1 (en) 2011-10-24 2012-10-23 Bicyclic compound

Publications (1)

Publication Number Publication Date
AR090809A1 true AR090809A1 (en) 2014-12-10

Family

ID=49959126

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP130101351A AR090809A1 (en) 2012-05-29 2013-04-23 BICYCLE COMPOUND

Country Status (3)

Country Link
AR (1) AR090809A1 (en)
TW (1) TW201350491A (en)
UY (1) UY34760A (en)

Also Published As

Publication number Publication date
UY34760A (en) 2013-12-31
TW201350491A (en) 2013-12-16

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