AR088943A1 - Acido 2-[(3,5-difluoro-3-metoxi-1,1-bifenil-4-il)amino]nicotinico para el tratamiento de psoriasis - Google Patents

Acido 2-[(3,5-difluoro-3-metoxi-1,1-bifenil-4-il)amino]nicotinico para el tratamiento de psoriasis

Info

Publication number
AR088943A1
AR088943A1 ARP120104381A ARP120104381A AR088943A1 AR 088943 A1 AR088943 A1 AR 088943A1 AR P120104381 A ARP120104381 A AR P120104381A AR P120104381 A ARP120104381 A AR P120104381A AR 088943 A1 AR088943 A1 AR 088943A1
Authority
AR
Argentina
Prior art keywords
difluoro
psoriasis
amino
treatment
nicotinico
Prior art date
Application number
ARP120104381A
Other languages
English (en)
Inventor
Godessart Marina Nuria
Balague Pelaez Cristina
Original Assignee
Almirall Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Almirall Sa filed Critical Almirall Sa
Publication of AR088943A1 publication Critical patent/AR088943A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/455Nicotinic acids, e.g. niacin; Derivatives thereof, e.g. esters, amides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics

Abstract

La presente proporciona ácido 2-[(3,5-difluoro-3-metoxi-1,1-bifenil-4-il)amino]nicotínico, o una sal farmacéuticamente aceptable o N-óxido o solvato o derivado deuterado del mismo, para uso en el tratamiento de psoriasis.
ARP120104381A 2011-11-21 2012-11-21 Acido 2-[(3,5-difluoro-3-metoxi-1,1-bifenil-4-il)amino]nicotinico para el tratamiento de psoriasis AR088943A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP11382356.1A EP2594271A1 (en) 2011-11-21 2011-11-21 2-[(3,5-difluoro-3'-methoxy-1,1'-biphenyl-4-yl)amino]nicotinic acid for the treatment of psoriasis.

Publications (1)

Publication Number Publication Date
AR088943A1 true AR088943A1 (es) 2014-07-16

Family

ID=45349113

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP120104381A AR088943A1 (es) 2011-11-21 2012-11-21 Acido 2-[(3,5-difluoro-3-metoxi-1,1-bifenil-4-il)amino]nicotinico para el tratamiento de psoriasis

Country Status (3)

Country Link
EP (1) EP2594271A1 (es)
AR (1) AR088943A1 (es)
WO (1) WO2013076170A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11311548B2 (en) 2017-03-02 2022-04-26 Aslan Pharmaceuticals Pte. Ltd. Cancer therapy
TW201834649A (zh) * 2017-03-02 2018-10-01 新加坡商亞獅康私人有限公司 癌症療法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2319596B1 (es) 2006-12-22 2010-02-08 Laboratorios Almirall S.A. Nuevos derivados de los acidos amino-nicotinico y amino-isonicotinico.
EP2135610A1 (en) * 2008-06-20 2009-12-23 Laboratorios Almirall, S.A. Combination comprising DHODH inhibitors and methotrexate
EP2228367A1 (en) 2009-03-13 2010-09-15 Almirall, S.A. Addition salts of amines containing hydroxyl and/or carboxylic groups with amino nicotinic acid derivatives as DHODH inhibitors

Also Published As

Publication number Publication date
WO2013076170A1 (en) 2013-05-30
EP2594271A1 (en) 2013-05-22

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal