AR075046A1 - DERIVATIVES OF TRIAZOLOPIRIMIDINE OR ITS SALT, PROCESS TO PRODUCE THEM AND PESTICIDE THAT CONTAINS THEM - Google Patents

DERIVATIVES OF TRIAZOLOPIRIMIDINE OR ITS SALT, PROCESS TO PRODUCE THEM AND PESTICIDE THAT CONTAINS THEM

Info

Publication number
AR075046A1
AR075046A1 ARP100100140A ARP100100140A AR075046A1 AR 075046 A1 AR075046 A1 AR 075046A1 AR P100100140 A ARP100100140 A AR P100100140A AR P100100140 A ARP100100140 A AR P100100140A AR 075046 A1 AR075046 A1 AR 075046A1
Authority
AR
Argentina
Prior art keywords
alkyl
substituted
het
case
haloalkyl
Prior art date
Application number
ARP100100140A
Other languages
Spanish (es)
Original Assignee
Ishihara Sangyo Kaisha
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ishihara Sangyo Kaisha filed Critical Ishihara Sangyo Kaisha
Publication of AR075046A1 publication Critical patent/AR075046A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06—Antimalarials
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A61P33/12—Schistosomicides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Reivindicacion 1: Un derivado de triazolopirimidina representado por la formula (1) o su sal, donde R1 es alquilo que puede estar sustituido con A, cicloalquilo que puede estar sustituido con A, alquenilo que puede estar sustituido con A, alquinilo que puede estar sustituido con A, halogeno, ciano, arilo, 1,3-dioxolanilo, COR2, S(O)nR3, NR3R4 o CONR3R4; Het es como se muestra en el grupo de formulas Het1 a Het7; A es halogeno, OR2, alquilo o cicloalquilo; R2 es hidrogeno, alquilo, haloalquilo, alcoxi o NR3R4; R3 es hidrogeno o alquil; R4 es hidrogeno, alquilo, haloalquilo, alquilcarbonilo, alcoxicarbonilo, haloalquilcarbonilo o haloalcoxicarbonilo; X es alquilo, alquenilo, alquinilo, arilo, halogeno, haloalquilo, ciano, nitro, NR3R4, S(O)nR3, OR2 o COR2; Y es oxígeno, azufre o NR5; R5 es aIquilo, haloalquilo, cicloalquilo o arilo; n es un numero entero de 0 a 2; w1 es un numero entero de 1 a 3; w2 es un numero entero de 1 a 2; y en un caso donde w1 o w2 es por lo menos 2, una pluralidad de X pueden ser iguales o diferentes, con la condicion de que quedan excluidos (1) un caso donde R1 es metilo, y Het es 5-hidroxi-3-metil-1-fenil-pirazol-4-ilo, (2) un caso donde R1 es fenilo, y Het es 1-etil-pirazol-4-ilo, (3) un caso donde R1 es metilo, y Het es tiofen-2-ilo sustituido con alquilo y (4) un caso donde R1 es trifluormetilo, y Het es tiofen-2-ilo sustituido con alquilo. Reivindicacion 7: Un método para controlar una plaga, que comprende aplicar una cantidad eficaz del derivado de triazolopirimidina o su sal corno se define en la reivindicacion 1.Claim 1: A triazolopyrimidine derivative represented by the formula (1) or its salt, wherein R 1 is alkyl that may be substituted with A, cycloalkyl that may be substituted with A, alkenyl that may be substituted with A, alkynyl that may be substituted with A, halogen, cyano, aryl, 1,3-dioxolanyl, COR2, S (O) nR3, NR3R4 or CONR3R4; Het is as shown in the group of formulas Het1 to Het7; A is halogen, OR2, alkyl or cycloalkyl; R2 is hydrogen, alkyl, haloalkyl, alkoxy or NR3R4; R3 is hydrogen or alkyl; R4 is hydrogen, alkyl, haloalkyl, alkylcarbonyl, alkoxycarbonyl, haloalkylcarbonyl or haloalkoxycarbonyl; X is alkyl, alkenyl, alkynyl, aryl, halogen, haloalkyl, cyano, nitro, NR3R4, S (O) nR3, OR2 or COR2; Y is oxygen, sulfur or NR5; R5 is alkyl, haloalkyl, cycloalkyl or aryl; n is an integer from 0 to 2; w1 is an integer from 1 to 3; w2 is an integer from 1 to 2; and in a case where w1 or w2 is at least 2, a plurality of X may be the same or different, with the proviso that (1) a case where R1 is methyl, and Het is 5-hydroxy-3- are excluded methyl-1-phenyl-pyrazol-4-yl, (2) a case where R1 is phenyl, and Het is 1-ethyl-pyrazol-4-yl, (3) a case where R1 is methyl, and Het is thiophene- 2-yl substituted with alkyl and (4) a case where R1 is trifluoromethyl, and Het is thiophene-2-yl substituted with alkyl. Claim 7: A method of controlling a pest, which comprises applying an effective amount of the triazolopyrimidine derivative or its salt as defined in claim 1.

ARP100100140A 2009-01-29 2010-01-22 DERIVATIVES OF TRIAZOLOPIRIMIDINE OR ITS SALT, PROCESS TO PRODUCE THEM AND PESTICIDE THAT CONTAINS THEM AR075046A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2009017716 2009-01-29

Publications (1)

Publication Number Publication Date
AR075046A1 true AR075046A1 (en) 2011-03-02

Family

ID=41735290

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP100100140A AR075046A1 (en) 2009-01-29 2010-01-22 DERIVATIVES OF TRIAZOLOPIRIMIDINE OR ITS SALT, PROCESS TO PRODUCE THEM AND PESTICIDE THAT CONTAINS THEM

Country Status (4)

Country Link
JP (1) JP2010195771A (en)
AR (1) AR075046A1 (en)
TW (1) TW201029575A (en)
WO (1) WO2010087294A1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112013007604B1 (en) * 2010-10-18 2018-06-05 E.I. Du Pont De Nemours And Company COMPOUND, COMPOSITION, METHOD FOR CONTROLING A PARASITARY NEMATOID AND TREATED SEED
WO2019121352A1 (en) * 2017-12-20 2019-06-27 Basf Se Herbicidal pyrimidine compounds
CN109180684B (en) * 2018-09-28 2020-09-11 郑州大学 Diaryl compound and preparation method thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4444774A (en) 1982-07-29 1984-04-24 American Cyanamid Company 7-Heteroaryl[1,2,4]triazolo[1,5-a]pyrimidines
DE10063115A1 (en) * 2000-12-18 2002-06-27 Bayer Ag triazolopyrimidines
UY28506A1 (en) * 2003-09-12 2005-04-29 Basf Ag 6-HALOGEN- (1,2,4) TRIAZOL (1,5-A) PYRIMIDINS TO COMBAT ANIMAL PESTS.
JP5231829B2 (en) 2007-02-15 2013-07-10 石原産業株式会社 Pyridyl-triazolopyrimidine derivatives or salts thereof, pest control agents containing them, and methods for producing them
JP2009017716A (en) 2007-07-06 2009-01-22 Toyota Motor Corp Voltage protection control apparatus for rotating machine

Also Published As

Publication number Publication date
WO2010087294A1 (en) 2010-08-05
TW201029575A (en) 2010-08-16
JP2010195771A (en) 2010-09-09

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