AR074395A1 - DERIVATIVES OF INDOL, ITS PREPARATION PROCEDURE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM - Google Patents

DERIVATIVES OF INDOL, ITS PREPARATION PROCEDURE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Info

Publication number
AR074395A1
AR074395A1 ARP090104513A ARP090104513A AR074395A1 AR 074395 A1 AR074395 A1 AR 074395A1 AR P090104513 A ARP090104513 A AR P090104513A AR P090104513 A ARP090104513 A AR P090104513A AR 074395 A1 AR074395 A1 AR 074395A1
Authority
AR
Argentina
Prior art keywords
indol
derivatives
pharmaceutical compositions
compositions containing
preparation procedure
Prior art date
Application number
ARP090104513A
Other languages
Spanish (es)
Inventor
Frank Suzenet
Gerald Guillaumet
Daniel-Henri Caignard
Michael Spedding
Philippe Delagrange
Matthieu Jeanty
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Servier Lab filed Critical Servier Lab
Publication of AR074395A1 publication Critical patent/AR074395A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D209/20—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals substituted additionally by nitrogen atoms, e.g. tryptophane
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Que son afines con los receptores de melatonina. Reivindicación 1: Compuestos de fórmula (1) en la que : R representa un grupo alquilo (C1-6) lineal o ramificado, un grupo cicloalquilo (C3-8), o un grupo cicloalquilo (C3-8) alquilo (C1-6) lineal o ramificado, sus enantiómeros y diastereoisómeros, así como sus sales de adición a una base farmacéuticamente aceptable.That are related to melatonin receptors. Claim 1: Compounds of formula (1) in which: R represents a linear or branched (C1-6) alkyl group, a (C3-8) cycloalkyl group, or a (C1-6) cycloalkyl group ) linear or branched, its enantiomers and diastereoisomers, as well as its addition salts to a pharmaceutically acceptable base.

ARP090104513A 2008-11-25 2009-11-24 DERIVATIVES OF INDOL, ITS PREPARATION PROCEDURE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AR074395A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0806599A FR2938839A1 (en) 2008-11-25 2008-11-25 NOVEL INDOLE DERIVATIVES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.

Publications (1)

Publication Number Publication Date
AR074395A1 true AR074395A1 (en) 2011-01-12

Family

ID=40902727

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP090104513A AR074395A1 (en) 2008-11-25 2009-11-24 DERIVATIVES OF INDOL, ITS PREPARATION PROCEDURE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Country Status (6)

Country Link
CN (1) CN102224138A (en)
AR (1) AR074395A1 (en)
BR (1) BRPI0920898A2 (en)
CA (1) CA2744178A1 (en)
FR (1) FR2938839A1 (en)
WO (1) WO2010061074A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105085366A (en) * 2014-05-07 2015-11-25 北京生命科学研究所 Indole skeleton compound and application thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4393081A (en) * 1981-10-28 1983-07-12 Miles Laboratories, Inc. Methyl 3-acetamido-2-(5-methoxy-indol-3-yl) propanoate and hypotensive use thereof

Also Published As

Publication number Publication date
BRPI0920898A2 (en) 2015-12-29
CN102224138A (en) 2011-10-19
CA2744178A1 (en) 2010-06-03
FR2938839A1 (en) 2010-05-28
WO2010061074A1 (en) 2010-06-03

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