AR053148A1 - COMBINATIONS UNDERSTANDING ALFA-2- DELTA LIGANDS - Google Patents
COMBINATIONS UNDERSTANDING ALFA-2- DELTA LIGANDSInfo
- Publication number
- AR053148A1 AR053148A1 ARP060100746A AR053148A1 AR 053148 A1 AR053148 A1 AR 053148A1 AR P060100746 A ARP060100746 A AR P060100746A AR 053148 A1 AR053148 A1 AR 053148A1
- Authority
- AR
- Argentina
- Prior art keywords
- quinazolin
- spiro
- dihydro
- cyclohexane
- chloro
- Prior art date
Links
Abstract
La presente se refiere a una combinacion de un inhibidor de PDE7 y un ligando alfa-2-delta, y a sales farmacéuticamente aceptables de los mismos, a composiciones farmacéuticas de los mismos y a su uso en tratamiento del dolor, particularmente dolor inflamatorio, neuropático, visceral y nociceptivo. Reivindicacion 2: Una combinacion de acuerdo con la reivindicacion 1, en la que el inhibidor de PDE7 se selecciona entre: 5'-carboxipropoxi-8'-cloro-espiro[ciclohexano-1-4'-(3',4'- dihidro)quinazolin]-2'(1'H)-ona; ácido cis-3-[(8'-cloro-2'-oxo-2',3'-dihidro-1'H-espiro[ciclohexano-1,4'-quinazolin]-5'-il)oxi]ciclobutanocarboxílico, y ácido trans-3-[(8'-cloro-2'-oxo-2',3'-dihidro-1'H-espiro[ciclohexano-1,4'-quinazolin]-5'- il)oxi]ciclobutanocarboxílico; o una sal o solvato farmacéuticamente aceptable del mismo.This refers to a combination of a PDE7 inhibitor and an alpha-2-delta ligand, and pharmaceutically acceptable salts thereof, to pharmaceutical compositions thereof and their use in the treatment of pain, particularly inflammatory, neuropathic, visceral pain. and nociceptive. Claim 2: A combination according to claim 1, wherein the PDE7 inhibitor is selected from: 5'-carboxypropoxy-8'-chloro-spiro [cyclohexane-1-4 '- (3', 4'-dihydro ) quinazolin] -2 '(1'H) -one; cis-3 - [(8'-chloro-2'-oxo-2 ', 3'-dihydro-1'H-spiro [cyclohexane-1,4'-quinazolin] -5'-yl) oxy] cyclobutanecarboxylic acid, and trans-3 - [(8'-chloro-2'-oxo-2 ', 3'-dihydro-1'H-spiro [cyclohexane-1,4'-quinazolin] -5'-yl) oxy] cyclobutanecarboxylic acid ; or a pharmaceutically acceptable salt or solvate thereof.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0504209A GB0504209D0 (en) | 2005-03-01 | 2005-03-01 | New use of PDE7 inhibitors |
US74185405P | 2005-12-02 | 2005-12-02 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR053148A1 true AR053148A1 (en) | 2007-04-25 |
Family
ID=37047905
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP060100746 AR053148A1 (en) | 2005-03-01 | 2006-02-28 | COMBINATIONS UNDERSTANDING ALFA-2- DELTA LIGANDS |
Country Status (3)
Country | Link |
---|---|
JP (1) | JP2006241158A (en) |
AR (1) | AR053148A1 (en) |
TW (1) | TW200642687A (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AP2007004161A0 (en) * | 2005-04-28 | 2007-10-31 | Pfizer Ltd | Amino acid derivatives |
-
2006
- 2006-02-27 TW TW095106683A patent/TW200642687A/en unknown
- 2006-02-28 JP JP2006052759A patent/JP2006241158A/en active Pending
- 2006-02-28 AR ARP060100746 patent/AR053148A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
JP2006241158A (en) | 2006-09-14 |
TW200642687A (en) | 2006-12-16 |
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