AR049472A1 - DERIVATIVES OF 1,2,4 OXADIAZOL ANTAGONISTS OF THE METABOTROPIC GLUTAMATE RECEIVER. PHARMACEUTICAL COMPOSITIONS. - Google Patents
DERIVATIVES OF 1,2,4 OXADIAZOL ANTAGONISTS OF THE METABOTROPIC GLUTAMATE RECEIVER. PHARMACEUTICAL COMPOSITIONS.Info
- Publication number
- AR049472A1 AR049472A1 ARP050100611A AR049472A1 AR 049472 A1 AR049472 A1 AR 049472A1 AR P050100611 A ARP050100611 A AR P050100611A AR 049472 A1 AR049472 A1 AR 049472A1
- Authority
- AR
- Argentina
- Prior art keywords
- antagonists
- pharmaceutical compositions
- derivatives
- oxadiazol
- metabotropic glutamate
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Los compuestos pertenecen a la categoría de derivados heterocíclicos de oxadiazoles utilizados como antagonistas del receptor mGluRS por su accion sobre el sistema nervioso. Composiciones farmacéuticas que los contienen. Reivindicacion 1:Un compuesto, o una de sus sales aceptables para uso farmacéutico, caracterizado porque se selecciona del grupo formado por los compuestos desde el 943 al 1006.The compounds belong to the category of heterocyclic derivatives of oxadiazoles used as antagonists of the mGluRS receptor by their action on the nervous system. Pharmaceutical compositions that contain them. Claim 1: A compound, or one of its salts acceptable for pharmaceutical use, characterized in that it is selected from the group consisting of the compounds from 943 to 1006.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US77986804A | 2004-02-18 | 2004-02-18 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR049472A1 true AR049472A1 (en) | 2006-08-09 |
Family
ID=36940522
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP050100611 AR049472A1 (en) | 2004-02-18 | 2005-02-18 | DERIVATIVES OF 1,2,4 OXADIAZOL ANTAGONISTS OF THE METABOTROPIC GLUTAMATE RECEIVER. PHARMACEUTICAL COMPOSITIONS. |
Country Status (2)
| Country | Link |
|---|---|
| AR (1) | AR049472A1 (en) |
| MY (1) | MY148488A (en) |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9303024B2 (en) | 2011-10-11 | 2016-04-05 | Dana-Farber Cancer Institute, Inc. | Pyrazol-3-ones that activate pro-apoptotic BAX |
| US9663529B2 (en) | 2013-07-02 | 2017-05-30 | Bristol-Myers Squibb Company | Tricyclic pyrido-carboxamide derivatives as rock inhibitors |
| US9914740B2 (en) | 2013-07-02 | 2018-03-13 | Bristol-Myers Squibb Company | Tricyclic pyrido-carboxamide derivatives as rock inhibitors |
| WO2023010192A1 (en) * | 2021-08-02 | 2023-02-09 | Eurofarma Laboratórios S.A. | N-acylhydrazone compounds capable of inhibiting nav1.7 and/or nav1.8, processes for the preparation thereof, compositions, uses, methods for treatment using same, and kits |
-
2005
- 2005-02-17 MY MYPI20050606 patent/MY148488A/en unknown
- 2005-02-18 AR ARP050100611 patent/AR049472A1/en unknown
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9303024B2 (en) | 2011-10-11 | 2016-04-05 | Dana-Farber Cancer Institute, Inc. | Pyrazol-3-ones that activate pro-apoptotic BAX |
| US10000478B2 (en) | 2011-10-11 | 2018-06-19 | Dana-Farber Cancer Institute, Inc. | Pyrazol-3-ones that activate pro-apoptotic BAX |
| US10844053B2 (en) | 2011-10-11 | 2020-11-24 | Dana-Farber Cancer Institute, Inc. | Pyrazol-3-ones that activate pro-apoptotic BAX |
| US9663529B2 (en) | 2013-07-02 | 2017-05-30 | Bristol-Myers Squibb Company | Tricyclic pyrido-carboxamide derivatives as rock inhibitors |
| US9914740B2 (en) | 2013-07-02 | 2018-03-13 | Bristol-Myers Squibb Company | Tricyclic pyrido-carboxamide derivatives as rock inhibitors |
| WO2023010192A1 (en) * | 2021-08-02 | 2023-02-09 | Eurofarma Laboratórios S.A. | N-acylhydrazone compounds capable of inhibiting nav1.7 and/or nav1.8, processes for the preparation thereof, compositions, uses, methods for treatment using same, and kits |
Also Published As
| Publication number | Publication date |
|---|---|
| MY148488A (en) | 2013-04-30 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| UY31127A1 (en) | METABOTROPIC RECEIVER OXYADAZOL LIGANDS FOR GLUTAMATE AND ITS USE AS POTENTIALS - 841 | |
| ECSP109856A (en) | DERIVATIVES OF OXADIAZOL AND ITS USE AS POTENTIALS OF METABOTROPIC RECEIVERS OF GLUTAMATE - 842 | |
| DOP2010000375A (en) | DERIVATIVES OF ISOXAZOL AND ITS USE AS POTENTIATORS OF METABOTROPIC GLUTAMATE RECEPTORS | |
| CO6231028A2 (en) | COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF PROTEIN QUINASA | |
| UY31940A (en) | SUBSTITUTED DERIVATIVES OF 4,5- (SUBSTITUTED-PIRIDIN-3-IL) -1-METHYL-1H-INDOL, ITS PHARMACEUTICALLY ACCEPTABLE SALTS, POLYMORPHOS, ROTÁMEROS, PRO-DRUGS, ANANTIOMERS, HYDRATES, SOLVATOS OF THE SAME AND COMPOSITIONS | |
| UY28764A1 (en) | POLYHETHEROCYCLIC COMPOUNDS AND THEIR USE AS ANTAGONISTS OF THE METABOTROPIC GLUTAMATE RECEIVER | |
| UY29267A1 (en) | PIPERIDINE DERIVATIVES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS | |
| UY28763A1 (en) | TETRAZOL COMPOUNDS AND THEIR USE AS ANTAGONISTS OF THE METABOTROPIC GLUTAMATE RECEIVER | |
| PE20181094A1 (en) | CONDENSED HETEROCYCLIC DERIVATIVES REPLACED BY 2- (HET) ARILO AS PESTICIDES | |
| UY29176A1 (en) | SUBSTITUTED DERIVATIVES OF PURINA, PURINONA AND DEAZAPURINA, COMPOSITIONS THAT CONTAIN THEM, METHODS FOR THEIR PREPARATION AND ITS USES. | |
| UY28775A1 (en) | TETRAHYDROCHINOLINONES AND ITS USE AS ANTAGONISTS OF METABOTROPIC GLUTAMATE RECEPTORS | |
| UY29177A1 (en) | SUBSTITUTED DERIVATIVES OF PURINA, PURINONA AND DEAZAPURINA, COMPOSITIONS THAT CONTAIN METHODS FOR THEIR PREPARATION AND ITS USES | |
| UY28766A1 (en) | ADDITIONAL HETEROPOLYCLIC COMPOUNDS AND THEIR USE AS ANTAGONISTS OF THE METABOTROPIC GLUTAMATE RECEIVER | |
| AR063602A1 (en) | DERIVATIVES OF SPIROINDOLINONE, PHARMACEUTICAL FORMULATIONS THAT CONTAIN THEM AND THEIR USE IN THE OBTAINING OF A MEDICINAL PRODUCT FOR THE TREATMENT OF ONCOLOGICAL DISORDERS. | |
| UY28765A1 (en) | ACETILINIC PIPERAZINE COMPOUNDS AND THEIR USE AS ANTAGONISTS OF THE METABOTROPIC GLUTAMATE RECEPTOR | |
| GT200500175A (en) | CETP INHIBITORS | |
| CL2004000655A1 (en) | COMPOUNDS DERIVED FROM PIPERIDIN-2-ONA 1,6-DISUSTITUTED, ITS SALTS, PHARMACEUTICAL COMPOSITION, AGONISTS OF THE EP4 RECEIVER; USE OF COMPOUNDS TO TREAT OCULAR HYPERTENSION, GLAUCOMA. | |
| CR11518A (en) | CARBAMOIL COMPOUNDS AS DGAT1 190 INHIBITORS | |
| AR078278A1 (en) | ANTAGONISTS OF TIAZOL AND OXAZOL HEPCIDINE, PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM AND USE OF THE SAME FOR THE TREATMENT OF ANEMIAS AND ILLNESSES ASSOCIATED WITH IRON DEFICIENCIES. | |
| UY31863A (en) | DRUG COMBINATIONS UNDERSTANDING A DGAT INHIBITOR AND A PPAR AGONIST | |
| AR049276A1 (en) | OPIOOD CARBOXAMID COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
| UY29798A1 (en) | CARBOXAMIDE DERIVATIVES AS ANTAGONISTS OF THE MUSCARINIC RECEIVER | |
| DOP2010000226A (en) | TRICICLIC COMPOUNDS THAT HAVE ANTAGONIST ACTIVITY OF CORTICOTROPINE RELEASE FACTOR AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME | |
| AR056860A1 (en) | TRIAZOL DERIVATIVES INHIBITORS OF QUINASA TGF-BETA1 RECEPTORS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND USES FOR TUMOR TREATMENT | |
| ECSP10010105A (en) | CGRP ANTAGONISTS |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |