AR042210A1 - PHARMACEUTICAL COMPOSITION CONTAINING ANTIGONISTS OF LEUCOTRIENS B4 (LTB4) AND INHIBITORS OF CYCLLOXYGENASE (COX) - Google Patents
PHARMACEUTICAL COMPOSITION CONTAINING ANTIGONISTS OF LEUCOTRIENS B4 (LTB4) AND INHIBITORS OF CYCLLOXYGENASE (COX)Info
- Publication number
- AR042210A1 AR042210A1 ARP030104350A AR042210A1 AR 042210 A1 AR042210 A1 AR 042210A1 AR P030104350 A ARP030104350 A AR P030104350A AR 042210 A1 AR042210 A1 AR 042210A1
- Authority
- AR
- Argentina
- Prior art keywords
- pharmaceutically acceptable
- solvate
- acceptable salt
- functional derivative
- cyclloxygenase
- Prior art date
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Formulación farmacéutica que comprende un agente antagonista de LTB, que tiene un grupo hidroxi y un grupo benzamidino, o un tautómero, una sal farmacéuticamente aceptable, un solvato, o un derivado fisiológicamente funcional del mismo, en particular un compuesto de fórmula (1), en el que R y A son como se han definido en las reivindicaciones, o un tautómero, una sal farmacéuticamente aceptable, un solvato o un derivado fisiológicamente funcional del mismo (1) y por lo menos un agente inhibidor de ciclooxigenasa-2, un agente inhibidor de cox1/2 combinado, o una sal farmacéuticamente aceptable, un solvato o un derivado fisiológicamente funcional del mismo (2), y un vehículo o excipiente farmacéuticamente aceptable, y opcionalmente uno o más de otros ingredientes terapéuticos. Método para la prevención o el tratamiento de artritis reumatoide, dermatitis atópica y enfermedad cardiaca coronaria entre otras.Pharmaceutical formulation comprising an LTB antagonist agent, which has a hydroxy group and a benzamidino group, or a tautomer, a pharmaceutically acceptable salt, a solvate, or a physiologically functional derivative thereof, in particular a compound of formula (1), wherein R and A are as defined in the claims, or a tautomer, a pharmaceutically acceptable salt, a solvate or a physiologically functional derivative thereof (1) and at least one cyclooxygenase-2 inhibiting agent, an agent combined cox1 / 2 inhibitor, or a pharmaceutically acceptable salt, a solvate or a physiologically functional derivative thereof (2), and a pharmaceutically acceptable carrier or excipient, and optionally one or more other therapeutic ingredients. Method for the prevention or treatment of rheumatoid arthritis, atopic dermatitis and coronary heart disease among others.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ARP030104350 AR042210A1 (en) | 2003-11-26 | 2003-11-26 | PHARMACEUTICAL COMPOSITION CONTAINING ANTIGONISTS OF LEUCOTRIENS B4 (LTB4) AND INHIBITORS OF CYCLLOXYGENASE (COX) |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ARP030104350 AR042210A1 (en) | 2003-11-26 | 2003-11-26 | PHARMACEUTICAL COMPOSITION CONTAINING ANTIGONISTS OF LEUCOTRIENS B4 (LTB4) AND INHIBITORS OF CYCLLOXYGENASE (COX) |
Publications (1)
Publication Number | Publication Date |
---|---|
AR042210A1 true AR042210A1 (en) | 2005-06-15 |
Family
ID=42777791
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP030104350 AR042210A1 (en) | 2003-11-26 | 2003-11-26 | PHARMACEUTICAL COMPOSITION CONTAINING ANTIGONISTS OF LEUCOTRIENS B4 (LTB4) AND INHIBITORS OF CYCLLOXYGENASE (COX) |
Country Status (1)
Country | Link |
---|---|
AR (1) | AR042210A1 (en) |
-
2003
- 2003-11-26 AR ARP030104350 patent/AR042210A1/en unknown
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