AR042210A1 - PHARMACEUTICAL COMPOSITION CONTAINING ANTIGONISTS OF LEUCOTRIENS B4 (LTB4) AND INHIBITORS OF CYCLLOXYGENASE (COX) - Google Patents

PHARMACEUTICAL COMPOSITION CONTAINING ANTIGONISTS OF LEUCOTRIENS B4 (LTB4) AND INHIBITORS OF CYCLLOXYGENASE (COX)

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Publication number
AR042210A1
AR042210A1 ARP030104350A AR042210A1 AR 042210 A1 AR042210 A1 AR 042210A1 AR P030104350 A ARP030104350 A AR P030104350A AR 042210 A1 AR042210 A1 AR 042210A1
Authority
AR
Argentina
Prior art keywords
pharmaceutically acceptable
solvate
acceptable salt
functional derivative
cyclloxygenase
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Birke Franz Dr
Jennewein Hans Michael Dr
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Priority to ARP030104350 priority Critical patent/AR042210A1/en
Publication of AR042210A1 publication Critical patent/AR042210A1/en

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Abstract

Formulación farmacéutica que comprende un agente antagonista de LTB, que tiene un grupo hidroxi y un grupo benzamidino, o un tautómero, una sal farmacéuticamente aceptable, un solvato, o un derivado fisiológicamente funcional del mismo, en particular un compuesto de fórmula (1), en el que R y A son como se han definido en las reivindicaciones, o un tautómero, una sal farmacéuticamente aceptable, un solvato o un derivado fisiológicamente funcional del mismo (1) y por lo menos un agente inhibidor de ciclooxigenasa-2, un agente inhibidor de cox1/2 combinado, o una sal farmacéuticamente aceptable, un solvato o un derivado fisiológicamente funcional del mismo (2), y un vehículo o excipiente farmacéuticamente aceptable, y opcionalmente uno o más de otros ingredientes terapéuticos. Método para la prevención o el tratamiento de artritis reumatoide, dermatitis atópica y enfermedad cardiaca coronaria entre otras.Pharmaceutical formulation comprising an LTB antagonist agent, which has a hydroxy group and a benzamidino group, or a tautomer, a pharmaceutically acceptable salt, a solvate, or a physiologically functional derivative thereof, in particular a compound of formula (1), wherein R and A are as defined in the claims, or a tautomer, a pharmaceutically acceptable salt, a solvate or a physiologically functional derivative thereof (1) and at least one cyclooxygenase-2 inhibiting agent, an agent combined cox1 / 2 inhibitor, or a pharmaceutically acceptable salt, a solvate or a physiologically functional derivative thereof (2), and a pharmaceutically acceptable carrier or excipient, and optionally one or more other therapeutic ingredients. Method for the prevention or treatment of rheumatoid arthritis, atopic dermatitis and coronary heart disease among others.

ARP030104350 2003-11-26 2003-11-26 PHARMACEUTICAL COMPOSITION CONTAINING ANTIGONISTS OF LEUCOTRIENS B4 (LTB4) AND INHIBITORS OF CYCLLOXYGENASE (COX) AR042210A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ARP030104350 AR042210A1 (en) 2003-11-26 2003-11-26 PHARMACEUTICAL COMPOSITION CONTAINING ANTIGONISTS OF LEUCOTRIENS B4 (LTB4) AND INHIBITORS OF CYCLLOXYGENASE (COX)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ARP030104350 AR042210A1 (en) 2003-11-26 2003-11-26 PHARMACEUTICAL COMPOSITION CONTAINING ANTIGONISTS OF LEUCOTRIENS B4 (LTB4) AND INHIBITORS OF CYCLLOXYGENASE (COX)

Publications (1)

Publication Number Publication Date
AR042210A1 true AR042210A1 (en) 2005-06-15

Family

ID=42777791

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP030104350 AR042210A1 (en) 2003-11-26 2003-11-26 PHARMACEUTICAL COMPOSITION CONTAINING ANTIGONISTS OF LEUCOTRIENS B4 (LTB4) AND INHIBITORS OF CYCLLOXYGENASE (COX)

Country Status (1)

Country Link
AR (1) AR042210A1 (en)

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