AR034111A1 -
7-DEAZAPURINE COMPOUNDS N-6 REPLACED FOR ADENOSINE A1 AND A3 RECEIVERS, A METHOD FOR THEIR PREPARATION, A SOLUBLE DRUG, PHARMACEUTICAL COMPOSITION AND USES OF THE SAME FOR THE MANUFACTURE OF MEDICINES AND A METHOD TO INHIBIT THE ACTIVITY OF INHIBITING A1
- Google Patents
7-DEAZAPURINE COMPOUNDS N-6 REPLACED FOR ADENOSINE A1 AND A3 RECEIVERS, A METHOD FOR THEIR PREPARATION, A SOLUBLE DRUG, PHARMACEUTICAL COMPOSITION AND USES OF THE SAME FOR THE MANUFACTURE OF MEDICINES AND A METHOD TO INHIBIT THE ACTIVITY OF INHIBITING A1
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Priority claimed from US09/454,074external-prioritypatent/US6878716B1/en
Application filed by Osi Pharm IncfiledCriticalOsi Pharm Inc
Publication of AR034111A1publicationCriticalpatent/AR034111A1/en
Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Abstract
Un compuesto de 7-deazapurinas N-6 sustituidas, que tiene la estructura 1 donde R3 es un anillo aromático de 5-6 miembros; donde R5 y R6 son independientemente H, o alquilo; un método para su preparación, una prodroga soluble, composición farmacéutica y usos de los mismos para la manufactura de medicamentos y un método para inhibir la actividad de un receptor de adenosina A1.A compound of substituted N-6 7-deazapurines, having structure 1 where R3 is an aromatic ring of 5-6 members; where R5 and R6 are independently H, or alkyl; a method for its preparation, a soluble prodrug, pharmaceutical composition and uses thereof for the manufacture of medicaments and a method for inhibiting the activity of an adenosine A1 receptor.
ARP0001063791999-12-022000-12-01
7-DEAZAPURINE COMPOUNDS N-6 REPLACED FOR ADENOSINE A1 AND A3 RECEIVERS, A METHOD FOR THEIR PREPARATION, A SOLUBLE DRUG, PHARMACEUTICAL COMPOSITION AND USES OF THE SAME FOR THE MANUFACTURE OF MEDICINES AND A METHOD TO INHIBIT THE ACTIVITY OF INHIBITING A1
AR034111A1
(en)
7-DEAZAPURINE COMPOUNDS N-6 REPLACED FOR ADENOSINE A1 AND A3 RECEIVERS, A METHOD FOR THEIR PREPARATION, A SOLUBLE DRUG, PHARMACEUTICAL COMPOSITION AND USES OF THE SAME FOR THE MANUFACTURE OF MEDICINES AND A METHOD TO INHIBIT THE ACTIVITY OF INHIBITING A1
DERIVATIVES OF TRICYCLIC MACROLIDES, A PHARMACEUTICAL COMPOSITION THAT CONTAINS THEM, USE OF THEM TO PREPARE MEDICINES AND PROCEDURE FOR THEIR PREPARATION
DERIVATIVES OF TER.-BUTIL- (7-METHYL-IMIDAZO [1,2, a] PIRIDIN-3-IL) -AMINA, PROCEDURE FOR THEIR PREPARATION, DRUGS THAT CONTAIN THEM, THEIR USE FOR THE PREPARATION OF A MEDICATION FOR THE INHIBITION OF NON-SYNTHEASE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
compound having inhibitory activity against sodium-dependent carrier, pharmaceutical composition comprising the compound, use of the compound in the preparation of a medicine, and process for preparing the compound
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