AR028811A1 -
COMPOUNDS DERIVED FROM N-UREIDOALQUIL-PIPERIDINES, PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM AND THEIR USE IN THE MANUFACTURE OF MEDICINES
- Google Patents
COMPOUNDS DERIVED FROM N-UREIDOALQUIL-PIPERIDINES, PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM AND THEIR USE IN THE MANUFACTURE OF MEDICINES
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Application filed by Bristol Myers Squibb Pharma CofiledCriticalBristol Myers Squibb Pharma Co
Priority to ARP000100094ApriorityCriticalpatent/AR028811A1/en
Publication of AR028811A1publicationCriticalpatent/AR028811A1/en
Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Abstract
Describe Compuestos derivados de N-ureídoalquil-piperidinas, moduladores de CCR3 de formula (1) cuyos sustituyentes se enuncian en la memoria descriptiva, o las sales de los mismos aceptables para el uso farmacéutico. Se describen asimismo las compos iciones farmacéuticas que los comprenden y su uso en la fabricacion de medicamentos para tratar afecciones inflamatorias como el asma y otras enfermedades alérgicas.Describes compounds derived from N-ureidoalkyl piperidines, modulators of CCR3 of formula (1) whose substituents are set forth in the specification, or salts thereof acceptable for pharmaceutical use. The pharmaceutical compositions that comprise them and their use in the manufacture of medicaments for treating inflammatory conditions such as asthma and other allergic diseases are also described.
ARP000100094A2000-01-102000-01-10
COMPOUNDS DERIVED FROM N-UREIDOALQUIL-PIPERIDINES, PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM AND THEIR USE IN THE MANUFACTURE OF MEDICINES
AR028811A1
(en)
PIRAZOLOPIRIDINES, PYRROLOPYRIDIDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCEDURES FOR ITS ADMINISTRATION AS AN ANTAGONIST OF THE CORTICO-TROPINE RELEASE FACTOR
IMIDAZOPIRIMIDINE DERIVATIVES AND TRIAZOLOPIRIMIDINE DERIVATIVES, A PROCEDURE FOR THEIR PREPARATION, MEDICINES, A PHARMACEUTICAL COMPOSITION, AND THE USE OF SUCH DERIVATIVES FOR THE PREPARATION OF MEDICINES
SMALL MOLECULES, THE INTERMEDIARIES FOR THEIR SYNTHESIS, THE PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM AND THEIR USE TO PREPARE A MEDICINAL PRODUCT INTENDED FOR TREATMENT OR PROPHYLAXIS OF INFLAMMATORY DISEASES OR MEDIATIONED BY IMMUNE CELLS
DERIVATIVES OF 5-PHENYL-4-METHYL-TIAZOL-2-IL-AMINA AS INHIBITORS OF KINASA ENZYMES PHOSFATIDILINOSITOL 3 (PI3) FOR THE TREATMENT OF INFLAMMATORY DISEASES OF THE RESPIRATORY ROUTES
DERIVATIVES OF ARILPIPERAZINIL-CICLOHEXIL INDOL, PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM AND THE USE OF THE SAME FOR THE MANUFACTURE OF MEDICINES FOR THE TREATMENT OF DEPRESSION
3A, 4,5,6,7,7A-HEXAHIDRO-3H-BENZOIMIDAZOL AND DERIVAODS OF 3A, 4,5,6,, 7,7A-HEXAHIDRO-3-INDOL, ENANTIOMERS, DIASTEREOISOMERS, PHARMACEUTICALLY ACCEPTED SALTS, MIXTURES, COMPOSITIONS , PREPARATIONS AND APPLICATIONS OF THE SAME
COMPOUND DERIVED FROM A REPLACED POLYCLICAL PIRIDONE, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND THE USE OF SUCH COMPOUND AND SUCH COMPOSITION IN THE MANUFACTURE OF USEFUL DRUGS FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL