AR021540A1 - PROCEDURE FOR OBTAINING DERIVATIVES OF PIRAZOLILBENZOILO, AS WELL AS NEW DERIVATIVES OF PIRAZOLILBENZOILO - Google Patents

PROCEDURE FOR OBTAINING DERIVATIVES OF PIRAZOLILBENZOILO, AS WELL AS NEW DERIVATIVES OF PIRAZOLILBENZOILO

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Publication number
AR021540A1
AR021540A1 ARP990106175A AR021540A1 AR 021540 A1 AR021540 A1 AR 021540A1 AR P990106175 A ARP990106175 A AR P990106175A AR 021540 A1 AR021540 A1 AR 021540A1
Authority
AR
Argentina
Prior art keywords
alkyl
halogen
cyano
nitro
group
Prior art date
Application number
Other languages
Spanish (es)
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of AR021540A1 publication Critical patent/AR021540A1/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5

Abstract

El presente invento se refiere a un procedimiento para la obtencion de derivados de pirazolilbenzoilo de la formula (1) en la que los sustituyentes tienenlos significados siguientes: R1 hidrogeno, alquilo C1-4 o halogenoalquilo C1-4; R2 hidrogeno;al quilo C1-6, alquenilo C2-6, alquinilo C2-6, bencilo, benzoilo,alquilcarbonilo C1-4, hidroxicarbonil-C1-4-alquilo, alcoxicarbonil C1-4-alquilo C1-4, alquilsulfonilo C1-4 o fenilsulfonilo, pudiendo estos grupos estarsustituidos por alquilo C1-4,alcoxi C1-4, alquiltio C1-4, halogeno, hidroxi, amino, nitro o ciano; A, B, D cada uno independientemente del otro, hidrogeno;alquilo C1-6, alquenilo C2-6, alquinilo C2-6, alcoxi C1-4, pudiendo estos grupos estar sustituidos por halogeno, hidroxi,alcoxi C 1-4 o ciano; halogeno,hidroxi, ciano, nitro, un grupo -(Y)n-S(O)mR3 o un grupo -(Y)n-CO-R4; Z hidrogeno; alquilo C1-6, alquenilo C2-6, alquinilo C2-6, alcoxi C1-4, pudiendo estosgrupos estar sustituidos por halogeno, hidroxi, alcoxi C1-4 ociano; hal ogeno, hidroxi, ciano, nitro, un grupo -(Y)n-S(O)mR3 o un grupo -(Y)n-CO-R4; fenilo,que puede estar sustituido por alquilo C1-4, halogenoalquilo C1-4, halogeno, hidroxi, ciano o nitro; un radical heterocíclico saturado o sin saturar de 5o 6miembros, que contiene de uno a tres heteroátomos, seleccionados del grupo oxígeno, azufre o nitrogeno, que eventualmente está sustituido por halogeno, ciano,nitro, un grupo -CO-R4, alquilo C1-4, halogenoalquilo C1-4, cicloalquilo C3-8, alcoxiC1-4, halogenoa lcoxi C1-4, alquiltio C1-4, halogenoalquiltio C1-4,di-C1-4-alquilamino, fenilo eventualmente sustituido por halogeno, ciano, nitro, alquil C1-4 o halogenoalquilo C1-4 o un grupo oxo, que eventualmente puedeestar presente también enla forma tautomera como grupo hidroxi, o que puede formar con un anillo fenilo condensado, eventualmente sustituido por halogeno,ciano, nitro, alquilo C1-4 o halogenoalquilo C1-4, un carbociclo condensado o un segundo heterociclo condensado,eventualmente sustituido p or halogeno, ciano,nitro, alquilo C1-4, di-C1-4-alquilamino, alcoxi C1-4, halogenoalcoxi C1-4 o halogenoalquilo C1-4, un sistema bicíclico; Y O, NR5, n cero o uno, m cero, uno oThe present invention relates to a process for obtaining pyrazolylbenzoyl derivatives of the formula (1) in which the substituents have the following meanings: R 1 hydrogen, C 1-4 alkyl or C 1-4 halogenoalkyl; R2 hydrogen; C1-6 chyl, C2-6 alkenyl, C2-6 alkynyl, benzyl, benzoyl, C1-4 alkylcarbonyl, hydroxycarbonyl-C1-4-alkyl, C1-4 alkoxycarbonyl-C1-4 alkyl, C1-4 alkylsulfonyl or phenylsulfonyl, these groups being substituted by C1-4 alkyl, C1-4 alkoxy, C1-4 alkylthio, halogen, hydroxy, amino, nitro or cyano; A, B, D each independently of the other, hydrogen; C1-6 alkyl, C2-6 alkenyl, C2-6 alkynyl, C1-4 alkoxy, these groups may be substituted by halogen, hydroxy, C 1-4 alkoxy or cyano ; halogen, hydroxy, cyano, nitro, a group - (Y) n-S (O) mR3 or a group - (Y) n-CO-R4; Z hydrogen; C1-6 alkyl, C2-6 alkenyl, C2-6 alkynyl, C1-4 alkoxy, these groups may be substituted by halogen, hydroxy, C1-4 alkoxy; halogen, hydroxy, cyano, nitro, a group - (Y) n-S (O) mR3 or a group - (Y) n-CO-R4; phenyl, which may be substituted by C1-4 alkyl, halogen C1-4 alkyl, halogen, hydroxy, cyano or nitro; a saturated or unsaturated heterocyclic radical of 5-6 members, containing one to three heteroatoms, selected from the oxygen, sulfur or nitrogen group, which is eventually substituted by halogen, cyano, nitro, a -CO-R4 group, C1-4 alkyl , C1-4 halogenoalkyl, C3-8 cycloalkyl, C1-4 alkoxy, C1-4 haloxya, C1-4 alkylthio, C1-4 halogenoalkylthio, di-C1-4-alkylamino, phenyl optionally substituted by halogen, cyano, nitro, alkyl C1-4 or halogen C1-4 alkyl or an oxo group, which may also be present in the tautomeric form as a hydroxy group, or which may form with a condensed phenyl ring, optionally substituted by halogen, cyano, nitro, C1-4 alkyl or halogenoalkyl C1-4, a condensed carbocycle or a second condensed heterocycle, optionally substituted by halogen, cyano, nitro, C1-4 alkyl, di-C1-4-alkylamino, C1-4 alkoxy, C1-4 halogenoalkoxy or C1-4 halogenoalkyl , a bicyclic system; Y O, NR5, n zero or one, m zero, one or

ARP990106175 1998-12-04 1999-12-03 PROCEDURE FOR OBTAINING DERIVATIVES OF PIRAZOLILBENZOILO, AS WELL AS NEW DERIVATIVES OF PIRAZOLILBENZOILO AR021540A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19855850 1998-12-04

Publications (1)

Publication Number Publication Date
AR021540A1 true AR021540A1 (en) 2002-07-24

Family

ID=7889889

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP990106175 AR021540A1 (en) 1998-12-04 1999-12-03 PROCEDURE FOR OBTAINING DERIVATIVES OF PIRAZOLILBENZOILO, AS WELL AS NEW DERIVATIVES OF PIRAZOLILBENZOILO

Country Status (4)

Country Link
AR (1) AR021540A1 (en)
AU (1) AU2094700A (en)
WO (1) WO2000034247A2 (en)
ZA (2) ZA200105476B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3997255B2 (en) 2004-02-13 2007-10-24 ワーナー−ランバート カンパニー リミテッド ライアビリティー カンパニー Androgen receptor modulator
US7507860B2 (en) 2004-04-13 2009-03-24 Pfizer Inc. Androgen modulators
TW200724139A (en) 2005-05-05 2007-07-01 Warner Lambert Co Androgen modulators

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57212162A (en) * 1981-06-23 1982-12-27 Sankyo Co Ltd Pyrazole derivative and herbicide
KR19980702466A (en) * 1995-02-24 1998-07-15 페라 스타르크, 요헨 카르크 Pyrazol-4-yl-benzoyl derivatives and their use as herbicides
WO1997041117A1 (en) * 1996-04-26 1997-11-06 Nippon Soda Co., Ltd. Novel benzene derivatives substituted by heterocycles and herbicides
AU1670797A (en) * 1996-04-26 1997-11-19 Nippon Soda Co., Ltd. Benzene derivatives substituted by heterocycles and herbicides
HUP9902423A3 (en) * 1996-04-26 2001-02-28 Nippon Soda Co Benzene derivatives substituted by heterocycles and herbicides
AU3297397A (en) * 1996-06-06 1998-01-05 E.I. Du Pont De Nemours And Company Herbicidal pyridinyl and pyrazolylphenyl ketones
WO1998021187A1 (en) * 1996-11-13 1998-05-22 Nippon Soda Co., Ltd. Novel heterocycle substituted benzene derivatives and herbicide

Also Published As

Publication number Publication date
WO2000034247A2 (en) 2000-06-15
ZA200105477B (en) 2002-07-18
WO2000034247A3 (en) 2000-11-23
ZA200105476B (en) 2002-07-16
AU2094700A (en) 2000-06-26

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