AR018824A1 - Antagonistas del receptor de bradiquinina no peptidica para uso en el control de la presion intraocular y en el tratamiento del glaucoma - Google Patents
Antagonistas del receptor de bradiquinina no peptidica para uso en el control de la presion intraocular y en el tratamiento del glaucomaInfo
- Publication number
- AR018824A1 AR018824A1 ARP990101485A ARP990101485A AR018824A1 AR 018824 A1 AR018824 A1 AR 018824A1 AR P990101485 A ARP990101485 A AR P990101485A AR P990101485 A ARP990101485 A AR P990101485A AR 018824 A1 AR018824 A1 AR 018824A1
- Authority
- AR
- Argentina
- Prior art keywords
- glaucoma
- treatment
- control
- bradiquinine
- peptidic
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/472—Non-condensed isoquinolines, e.g. papaverine
- A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Uso de una composicion que comprende un antagonista de bradiquinina no peptídica para la fabricacion de un medicamento para el ojo para el control depresion intraocular y/o para el tratamiento del glaucoma que comprende una composicion que incluye una cantidad terapéuticamente efectiva de unantagonista de bradiquina no peptídica en un vehículo farmacéuticamente aceptable. Las composiciones comprenden antagonistas no peptídicas debradiquinina.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8073098P | 1998-04-03 | 1998-04-03 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR018824A1 true AR018824A1 (es) | 2001-12-12 |
Family
ID=22159253
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP990101485A AR018824A1 (es) | 1998-04-03 | 1999-03-31 | Antagonistas del receptor de bradiquinina no peptidica para uso en el control de la presion intraocular y en el tratamiento del glaucoma |
Country Status (4)
Country | Link |
---|---|
US (1) | US6500831B1 (es) |
AR (1) | AR018824A1 (es) |
AU (1) | AU2985399A (es) |
WO (1) | WO1999051235A1 (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2481855A1 (en) * | 2002-04-10 | 2003-10-23 | Ortho-Mcneil Pharmaceutical, Inc. | Novel heteroaryl alkylamide derivatives useful as bradykinin receptor modulators |
US7807629B1 (en) | 2007-06-05 | 2010-10-05 | Alcon Research, Ltd. | Use of bradykinin and related B2R agonists to treat ocular hypertension and glaucoma |
TW201210584A (en) | 2010-08-18 | 2012-03-16 | Alcon Res Ltd | Bradykinin receptor agonists and uses thereof to treat ocular hypertension and glaucoma |
CN103622961B (zh) * | 2013-09-06 | 2016-03-02 | 武汉光谷百桥国际生物科技有限公司 | 一种非肽类缓激肽b2受体激动剂在促进毛发生长方面的应用 |
WO2016170382A1 (en) | 2015-04-23 | 2016-10-27 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Pharmaceutical compositions comprising a bradykinin 2 receptor antagonist for prevention or treatment of impaired skin wound healing |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0529499A1 (de) * | 1991-08-22 | 1993-03-03 | Hoechst Aktiengesellschaft | Pharmazeutische Zusammensetzungen enthaltend Bradykinin-Antagonisten zur lokalen Anwendung an Nase und Auge |
-
1999
- 1999-03-04 WO PCT/US1999/004865 patent/WO1999051235A1/en active Application Filing
- 1999-03-04 AU AU29853/99A patent/AU2985399A/en not_active Abandoned
- 1999-03-04 US US09/647,571 patent/US6500831B1/en not_active Expired - Fee Related
- 1999-03-31 AR ARP990101485A patent/AR018824A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
AU2985399A (en) | 1999-10-25 |
US6500831B1 (en) | 2002-12-31 |
WO1999051235A1 (en) | 1999-10-14 |
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