AR004071A1 - A PROCEDURE FOR SYNTHESIZING COMPOUNDS BY ELECTROCHEMICAL OXIDATION - Google Patents

A PROCEDURE FOR SYNTHESIZING COMPOUNDS BY ELECTROCHEMICAL OXIDATION

Info

Publication number
AR004071A1
AR004071A1 ARP960104853A ARP960104853A AR004071A1 AR 004071 A1 AR004071 A1 AR 004071A1 AR P960104853 A ARP960104853 A AR P960104853A AR P960104853 A ARP960104853 A AR P960104853A AR 004071 A1 AR004071 A1 AR 004071A1
Authority
AR
Argentina
Prior art keywords
procedure
electrochemical oxidation
synthesizing compounds
compounds
synthesis
Prior art date
Application number
ARP960104853A
Other languages
Spanish (es)
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9603756.9A external-priority patent/GB9603756D0/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of AR004071A1 publication Critical patent/AR004071A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/24—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/04—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Un procedimiento para la síntesis de los compuestos (I) en donde X es halógeno, que consiste de, como mínimo en la oxidación electroquímica delreactivo alil acetonida con una sal haluro en un sistema acuoso, dichos compuestos sonútiles como intermediarios para la síntesis de inhibidores derenina o proteasa de VIH u otras proteasas.A procedure for the synthesis of compounds (I) where X is halogen, which consists of, at least, the electrochemical oxidation of the allyl acetonide reagent with a halide salt in an aqueous system, said compounds are useful as intermediates for the synthesis of renin inhibitors or HIV protease or other proteases.

ARP960104853A 1995-10-30 1996-10-22 A PROCEDURE FOR SYNTHESIZING COMPOUNDS BY ELECTROCHEMICAL OXIDATION AR004071A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US812595P 1995-10-30 1995-10-30
GBGB9603756.9A GB9603756D0 (en) 1996-02-22 1996-02-22 Electrochemical oxidation

Publications (1)

Publication Number Publication Date
AR004071A1 true AR004071A1 (en) 1998-09-30

Family

ID=26308784

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP960104853A AR004071A1 (en) 1995-10-30 1996-10-22 A PROCEDURE FOR SYNTHESIZING COMPOUNDS BY ELECTROCHEMICAL OXIDATION

Country Status (4)

Country Link
AR (1) AR004071A1 (en)
AU (1) AU7475896A (en)
TW (1) TW415948B (en)
WO (1) WO1997016450A1 (en)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6048595B2 (en) * 1978-10-03 1985-10-28 株式会社クラレ Method for producing halohydrin and/or epoxy
JPS6048982A (en) * 1983-08-29 1985-03-16 Takasago Corp Production of isosafrole halohydrin and/or isosafrole epoxide
TW380137B (en) * 1994-03-04 2000-01-21 Merck & Co Inc Process for making an epoxide

Also Published As

Publication number Publication date
AU7475896A (en) 1997-05-22
WO1997016450A1 (en) 1997-05-09
TW415948B (en) 2000-12-21

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