AR002248A1 - OXAZOLIL- AND THIAZOLYLIMIDAZO-BENZO- AND THENODIACEPINES, PROCEDURE FOR ITS PREPARATION AND USE AS ANSIOLYTIC AND / OR ANTICONVULSIVE AND / OR ORELAJANTS OF MUSCULATURE AND / OR SEDANTE-HIPNOTICOS. - Google Patents

OXAZOLIL- AND THIAZOLYLIMIDAZO-BENZO- AND THENODIACEPINES, PROCEDURE FOR ITS PREPARATION AND USE AS ANSIOLYTIC AND / OR ANTICONVULSIVE AND / OR ORELAJANTS OF MUSCULATURE AND / OR SEDANTE-HIPNOTICOS.

Info

Publication number
AR002248A1
AR002248A1 ARP950100111A AR10011195A AR002248A1 AR 002248 A1 AR002248 A1 AR 002248A1 AR P950100111 A ARP950100111 A AR P950100111A AR 10011195 A AR10011195 A AR 10011195A AR 002248 A1 AR002248 A1 AR 002248A1
Authority
AR
Argentina
Prior art keywords
thiazolylimidazo
benzo
thenodiacepines
sedante
orelajants
Prior art date
Application number
ARP950100111A
Other languages
Spanish (es)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of AR002248A1 publication Critical patent/AR002248A1/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

El invento se refiere a oxazolil- y tiazolilimidazo-benzo tienodiacepinas básicamente sustituidas de la fórmula general (I). Estos compuestos puedenutilizarse como medicamentos ansiolíticos y/o anticonvulsivos y/o relajantes de la musculatura y/o sedante-hipnóticos. El invento se refiere además a un métodode preparación de los compuestos.The invention relates to substantially substituted oxazolyl- and thiazolylimidazo-benzo thienodiazepines of the general formula (I). These compounds can be used as anxiolytic and / or anticonvulsant and / or muscle relaxant and / or sedative-hypnotic drugs. The invention further relates to a method of preparing the compounds.

ARP950100111A 1994-11-11 1995-11-09 OXAZOLIL- AND THIAZOLYLIMIDAZO-BENZO- AND THENODIACEPINES, PROCEDURE FOR ITS PREPARATION AND USE AS ANSIOLYTIC AND / OR ANTICONVULSIVE AND / OR ORELAJANTS OF MUSCULATURE AND / OR SEDANTE-HIPNOTICOS. AR002248A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH338694 1994-11-11

Publications (1)

Publication Number Publication Date
AR002248A1 true AR002248A1 (en) 1998-03-11

Family

ID=4254847

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP950100111A AR002248A1 (en) 1994-11-11 1995-11-09 OXAZOLIL- AND THIAZOLYLIMIDAZO-BENZO- AND THENODIACEPINES, PROCEDURE FOR ITS PREPARATION AND USE AS ANSIOLYTIC AND / OR ANTICONVULSIVE AND / OR ORELAJANTS OF MUSCULATURE AND / OR SEDANTE-HIPNOTICOS.

Country Status (5)

Country Link
AR (1) AR002248A1 (en)
CO (1) CO4520231A1 (en)
PE (1) PE49496A1 (en)
TR (1) TR199501390A2 (en)
ZA (1) ZA959327B (en)

Also Published As

Publication number Publication date
PE49496A1 (en) 1996-12-16
TR199501390A2 (en) 1996-07-21
ZA959327B (en) 1997-01-31
CO4520231A1 (en) 1997-10-15

Similar Documents

Publication Publication Date Title
MX9304819A (en) NEW XANTINA DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION.
MX9204111A (en) SUBSTITUTED TRIAZOLES AND PROCEDURE FOR THEIR OBTAINING.
UY26495A1 (en) "THIAZOLYLAMIDE DERIVATIVES"
GT199900056A (en) NEW DIHYDROPYRIMIDINES
TR200001603T2 (en) New compounds
UY27079A1 (en) PROCEDURE FOR THE PREPARATION OF AN ANTICHOLINERGIC
DK0640592T3 (en) N-acylated tricyclic azaheter rings useful as vasopressin antagonists
AR003401A1 (en) PROCEDURE FOR THE PEPARATION OF SILDENAFIL AND INTERMEDIATE COMPOUNDS FOR SUCH PROCEDURE
AR001081A1 (en) A process to prepare certain aza cyclohexapeptides and compounds prepared by said process
ES2153106T3 (en) AMINOPHENILURACILOS SUBSTITUTED AS HERBICIDES AND INSECTICIDES.
ES2178055T3 (en) SUBSTITUTED AMINIC DERIVATIVES, THEIR PREPARATION PROCEDURE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
ECSP034531A (en) SUBSTITUTED DERIVATIVES OF C-CICLOHEXILMETILAMINA
MX9304399A (en) NOVEL PROCESS TO PREPARE [[2-BROMOETHYL) -AMINO] METHYL] -2-NITRO-1H-IMIDAZOL-1-ETHANOL CHIRAL AND RELATED COMPOUNDS.
AR028743A1 (en) DERIVATIVES OF N-TRIAZOLILMETIL-PIPERAZINA WITH ANTAGONIST ACTION OF NEUROQUININE RECEPTORS
IS4367A (en) CCK or gastrin attenuating 5-heterocyclic-1,5-benzodiazepines
AR001813A1 (en) Chromone derivatives procedure for preparing them and the pharmaceutical compositions containing them
AR005619A1 (en) PROCEDURE FOR PREPARING DICETONIC COMPOUNDS
ES2185196T3 (en) A PROCEDURE FOR THE PREPARATION OF TETRAAZAMACROCICLOS.
AR002248A1 (en) OXAZOLIL- AND THIAZOLYLIMIDAZO-BENZO- AND THENODIACEPINES, PROCEDURE FOR ITS PREPARATION AND USE AS ANSIOLYTIC AND / OR ANTICONVULSIVE AND / OR ORELAJANTS OF MUSCULATURE AND / OR SEDANTE-HIPNOTICOS.
ES2166026T3 (en) DERIVATIVES OF 1,2,3-BENZOTIADIAZOL AND ITS USE AS MICROBICIDES.
ES2123827T3 (en) DERIVATIVES OF THE POLYAMIDIC ACID WITH ANTIGASTRINE ACTIVITY, A METHOD FOR ITS PREPARATION AND ITS PHARMACEUTICAL USE.
ITTO910353A0 (en) NEW TRICYCLIC COMPOUNDS, PROCEDURE FOR THEIR PREPARATION
UY26507A1 (en) SUBSTITUTED 1-NAFTOL AND 2-NAFTOL MANNICH BASES, PROCEDURE FOR THE PREPARATION, MEDICINES CONTAINING THESE COMPOUNDS, AS WELL AS THE USE OF THESE COMPOUNDS FOR THE PREPARATION OF MEDICINES
EE03873B1 (en) Process for the preparation of alkyloxfuranone amine derivatives, compounds obtained by this process and their use
MX9300335A (en) NEW N-ARYLINDOLES AND THEIR USE AS HERBICIDES.