AP1846A - Pyrazole Derivatives. - Google Patents

Pyrazole Derivatives.

Info

Publication number
AP1846A
AP1846A APAP/P/2002/002469A AP2002002469A AP1846A AP 1846 A AP1846 A AP 1846A AP 2002002469 A AP2002002469 A AP 2002002469A AP 1846 A AP1846 A AP 1846A
Authority
AP
ARIPO
Prior art keywords
compounds
preparation
reverse transcriptase
present
derivatives
Prior art date
Application number
APAP/P/2002/002469A
Other versions
AP2002002469A0 (en
Inventor
Lyn Howard Jones
Charles Eric Mowbray
David Anthony Price
Matthew Duncan Selby
Paul Anthony Stupple
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0108999A external-priority patent/GB0108999D0/en
Application filed by Pfizer filed Critical Pfizer
Publication of AP2002002469A0 publication Critical patent/AP2002002469A0/en
Application granted granted Critical
Publication of AP1846A publication Critical patent/AP1846A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

This invention relates to pyrazole derivatives of formula (I) or pharmaceutically acceptable salts, solvates or derivative thereofs, wherein R1 to R4 are defined in the description, and to processes for the preparation thereof, intermediates used in their preparation of, compositions containing them and the uses of such derivatives. The compounds of the present invention bind to the enzyme reverse transcriptase and are modulators, especially inhibitors thereof. As such the compounds of the present invention are useful in the treatment of a variety of disorders including those in which the inhibition of reverse transcriptase is implicated. Disorders of interest include those caused by Human Immunodificiency Virus (HIV) and genetically related retroviruses, such as acquired immune deficiency syndrome (AIDS).
APAP/P/2002/002469A 2001-04-10 2002-04-04 Pyrazole Derivatives. AP1846A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB0108999A GB0108999D0 (en) 2001-04-10 2001-04-10 Pyrazole derivatives
GB0127426A GB0127426D0 (en) 2001-11-15 2001-11-15 Pyrazole derivatives

Publications (2)

Publication Number Publication Date
AP2002002469A0 AP2002002469A0 (en) 2002-06-30
AP1846A true AP1846A (en) 2008-05-09

Family

ID=9925828

Family Applications (1)

Application Number Title Priority Date Filing Date
APAP/P/2002/002469A AP1846A (en) 2001-04-10 2002-04-04 Pyrazole Derivatives.

Country Status (3)

Country Link
AP (1) AP1846A (en)
GB (1) GB0127426D0 (en)
SV (1) SV2003000979A (en)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3963742A (en) * 1974-07-12 1976-06-15 American Cyanamid Company 1,2-Dialkyl-3,4,5-trisubstituted pyrazolium salts as herbicidal agents

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3963742A (en) * 1974-07-12 1976-06-15 American Cyanamid Company 1,2-Dialkyl-3,4,5-trisubstituted pyrazolium salts as herbicidal agents

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
J. Med. Chem., American Chem. Soc., Washington, US, Vol. 43, 2000, pp 1034-1040 *

Also Published As

Publication number Publication date
SV2003000979A (en) 2003-07-29
GB0127426D0 (en) 2002-01-09
AP2002002469A0 (en) 2002-06-30

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