AP1846A - Pyrazole Derivatives. - Google Patents
Pyrazole Derivatives.Info
- Publication number
- AP1846A AP1846A APAP/P/2002/002469A AP2002002469A AP1846A AP 1846 A AP1846 A AP 1846A AP 2002002469 A AP2002002469 A AP 2002002469A AP 1846 A AP1846 A AP 1846A
- Authority
- AP
- ARIPO
- Prior art keywords
- compounds
- preparation
- reverse transcriptase
- present
- derivatives
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
This invention relates to pyrazole derivatives of formula (I) or pharmaceutically acceptable salts, solvates or derivative thereofs, wherein R1 to R4 are defined in the description, and to processes for the preparation thereof, intermediates used in their preparation of, compositions containing them and the uses of such derivatives. The compounds of the present invention bind to the enzyme reverse transcriptase and are modulators, especially inhibitors thereof. As such the compounds of the present invention are useful in the treatment of a variety of disorders including those in which the inhibition of reverse transcriptase is implicated. Disorders of interest include those caused by Human Immunodificiency Virus (HIV) and genetically related retroviruses, such as acquired immune deficiency syndrome (AIDS).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0108999A GB0108999D0 (en) | 2001-04-10 | 2001-04-10 | Pyrazole derivatives |
GB0127426A GB0127426D0 (en) | 2001-11-15 | 2001-11-15 | Pyrazole derivatives |
Publications (2)
Publication Number | Publication Date |
---|---|
AP2002002469A0 AP2002002469A0 (en) | 2002-06-30 |
AP1846A true AP1846A (en) | 2008-05-09 |
Family
ID=9925828
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
APAP/P/2002/002469A AP1846A (en) | 2001-04-10 | 2002-04-04 | Pyrazole Derivatives. |
Country Status (3)
Country | Link |
---|---|
AP (1) | AP1846A (en) |
GB (1) | GB0127426D0 (en) |
SV (1) | SV2003000979A (en) |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3963742A (en) * | 1974-07-12 | 1976-06-15 | American Cyanamid Company | 1,2-Dialkyl-3,4,5-trisubstituted pyrazolium salts as herbicidal agents |
-
2001
- 2001-11-15 GB GB0127426A patent/GB0127426D0/en not_active Ceased
-
2002
- 2002-04-04 AP APAP/P/2002/002469A patent/AP1846A/en active
- 2002-04-09 SV SV2002000979A patent/SV2003000979A/en unknown
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3963742A (en) * | 1974-07-12 | 1976-06-15 | American Cyanamid Company | 1,2-Dialkyl-3,4,5-trisubstituted pyrazolium salts as herbicidal agents |
Non-Patent Citations (1)
Title |
---|
J. Med. Chem., American Chem. Soc., Washington, US, Vol. 43, 2000, pp 1034-1040 * |
Also Published As
Publication number | Publication date |
---|---|
SV2003000979A (en) | 2003-07-29 |
GB0127426D0 (en) | 2002-01-09 |
AP2002002469A0 (en) | 2002-06-30 |
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