WO1997020823A3 - 2-amino quinazoline derivatives as npy receptor antagonists - Google Patents

2-amino quinazoline derivatives as npy receptor antagonists Download PDF

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Publication number
WO1997020823A3
WO1997020823A3 PCT/EP1996/005067 EP9605067W WO9720823A3 WO 1997020823 A3 WO1997020823 A3 WO 1997020823A3 EP 9605067 W EP9605067 W EP 9605067W WO 9720823 A3 WO9720823 A3 WO 9720823A3
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WO
WIPO (PCT)
Prior art keywords
receptor antagonists
npy receptor
quinazoline derivatives
amino quinazoline
formula
Prior art date
Application number
PCT/EP1996/005067
Other languages
French (fr)
Other versions
WO1997020823A2 (en
Inventor
Heinrich Rueeger
Tibur Schmidlin
Pascal Rigollier
Yasuchika Yamaguchi
Marina Tintelnot-Blomley
Walter Schilling
Leoluca Criscione
Robert Mah
Original Assignee
Ciba Geigy Ag
Heinrich Rueeger
Tibur Schmidlin
Pascal Rigollier
Yasuchika Yamaguchi
Tintelnot Blomley Marina
Walter Schilling
Leoluca Criscione
Robert Mah
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag, Heinrich Rueeger, Tibur Schmidlin, Pascal Rigollier, Yasuchika Yamaguchi, Tintelnot Blomley Marina, Walter Schilling, Leoluca Criscione, Robert Mah filed Critical Ciba Geigy Ag
Priority to AU76929/96A priority Critical patent/AU7692996A/en
Publication of WO1997020823A2 publication Critical patent/WO1997020823A2/en
Publication of WO1997020823A3 publication Critical patent/WO1997020823A3/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4

Abstract

The invention relates to a compound of formula (I) in which the variables are as defined and or a salt or a tautomer thereof; and relates to a method of treatment of disorders or diseases associated with NPY receptor subtype Y5, to pharmaceutical compositions comprising a compound of formula (I) or a pharmaceutically acceptable salt thereof and to the manufacture of the compounds of formula (I) or a salt thereof.
PCT/EP1996/005067 1995-12-01 1996-11-18 2-amino quinazoline derivatives as npy receptor antagonists WO1997020823A2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU76929/96A AU7692996A (en) 1995-12-01 1996-11-18 Receptor antagonists

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US56637895A 1995-12-01 1995-12-01
US08/566,378 1995-12-01

Publications (2)

Publication Number Publication Date
WO1997020823A2 WO1997020823A2 (en) 1997-06-12
WO1997020823A3 true WO1997020823A3 (en) 1997-07-17

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP1996/005067 WO1997020823A2 (en) 1995-12-01 1996-11-18 2-amino quinazoline derivatives as npy receptor antagonists

Country Status (3)

Country Link
AU (1) AU7692996A (en)
WO (1) WO1997020823A2 (en)
ZA (1) ZA9610020B (en)

Cited By (1)

* Cited by examiner, † Cited by third party
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US8299066B2 (en) 2008-04-21 2012-10-30 Shionogi & Co., Ltd. Compounds having NPY Y5 receptor antagonistic activity

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WO1997020823A2 (en) 1997-06-12
ZA9610020B (en) 1997-06-01

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