SG11202108905UA - Crystalline form of an avibactam derivative - Google Patents

Crystalline form of an avibactam derivative

Info

Publication number
SG11202108905UA
SG11202108905UA SG11202108905UA SG11202108905UA SG11202108905UA SG 11202108905U A SG11202108905U A SG 11202108905UA SG 11202108905U A SG11202108905U A SG 11202108905UA SG 11202108905U A SG11202108905U A SG 11202108905UA SG 11202108905U A SG11202108905U A SG 11202108905UA
Authority
SG
Singapore
Prior art keywords
crystalline form
avibactam derivative
avibactam
derivative
crystalline
Prior art date
Application number
SG11202108905UA
Inventor
Sami Karaborni
Original Assignee
Arixa Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arixa Pharmaceuticals Inc filed Critical Arixa Pharmaceuticals Inc
Publication of SG11202108905UA publication Critical patent/SG11202108905UA/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SG11202108905UA 2019-03-12 2020-03-10 Crystalline form of an avibactam derivative SG11202108905UA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201962817243P 2019-03-12 2019-03-12
PCT/US2020/021795 WO2020185729A1 (en) 2019-03-12 2020-03-10 Crystalline form of an avibactam derivative

Publications (1)

Publication Number Publication Date
SG11202108905UA true SG11202108905UA (en) 2021-09-29

Family

ID=70155371

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11202108905UA SG11202108905UA (en) 2019-03-12 2020-03-10 Crystalline form of an avibactam derivative

Country Status (11)

Country Link
US (1) US11008321B2 (en)
EP (1) EP3938366A1 (en)
JP (1) JP2022524118A (en)
KR (1) KR20210137159A (en)
CN (1) CN113614084A (en)
AU (1) AU2020237440B2 (en)
BR (1) BR112021017874A2 (en)
CA (1) CA3133071A1 (en)
MX (1) MX2021011026A (en)
SG (1) SG11202108905UA (en)
WO (1) WO2020185729A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20210186983A1 (en) * 2019-12-20 2021-06-24 Arixa Pharmaceuticals, Inc. Orally administered combinations of amoxicillin and avibactam derivatives for treating mycobacterial infections

Family Cites Families (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3658849A (en) 1969-02-19 1972-04-25 Reynolds Tobacco Co R Treatment of 2-substituted aldehydes with lead dioxide
DE3045373A1 (en) 1980-12-02 1982-07-01 Henkel KGaA, 4000 Düsseldorf Use of 3-hydroxy-2,2-di:methyl-propionate ester(s) as fragrances - including new propyl ester
US4522811A (en) 1982-07-08 1985-06-11 Syntex (U.S.A.) Inc. Serial injection of muramyldipeptides and liposomes enhances the anti-infective activity of muramyldipeptides
IT1270594B (en) 1994-07-07 1997-05-07 Recordati Chem Pharm CONTROLLED RELEASE PHARMACEUTICAL COMPOSITION OF LIQUID SUSPENSION MOGUISTEIN
FR2812635B1 (en) 2000-08-01 2002-10-11 Aventis Pharma Sa NOVEL HETEROCYCLIC COMPOUNDS, PREPARATION AND USE AS MEDICAMENTS IN PARTICULAR AS ANTI-BACTERIALS
US6627646B2 (en) * 2001-07-17 2003-09-30 Sepracor Inc. Norastemizole polymorphs
UY30244A1 (en) 2006-03-30 2007-11-30 Tanabe Seiyaku Co A PROCESS TO PREPARE DERIVATIVES OF TETRAHYDROQUINOLINE
WO2009033054A1 (en) 2007-09-07 2009-03-12 Xenoport, Inc. Complex pantoic acid ester neopentyl sulfonyl ester cyclization release prodrugs of acamprosate, compositions thereof, and methods of use
US20090082464A1 (en) 2007-09-07 2009-03-26 Bernd Jandeleit Externally masked neopentyl sulfonyl ester cyclization release prodrugs of acamprosate, compositions thereof, and methods of use
WO2009052191A1 (en) 2007-10-15 2009-04-23 Xenoport, Inc. Internally masked neopentyl sulfonyl ester cyclization release prodrugs of acamprosate, compositions thereof, and methods of use
UA101966C2 (en) 2008-01-18 2013-05-27 Мерк Шарп Енд Доме Корп. Beta-lactamase inhibitors
GB0801401D0 (en) 2008-01-25 2008-03-05 Barry Callebaut Ag Composition
WO2009100045A1 (en) 2008-02-04 2009-08-13 Translational Genomics Research Institute Compounds, pharmaceutical compositions and methods of use of hydroxamic acid derivatives
CA2735929C (en) 2008-09-19 2013-12-17 Pfizer Inc. Hydroxamic acid derivatives useful as antibacterial agents
WO2010065709A2 (en) 2008-12-03 2010-06-10 Amin Khan Hydroxamic acid derivatives, preparation and therapeutic uses thereof
US20120053350A1 (en) 2009-04-30 2012-03-01 Ian Mangion Preparation of alkyl esters of n-protected oxo-azacycloalkylcarboxylic acids
CN102638981B (en) 2009-10-14 2015-07-22 默沙东公司 Substituted piperidines that increase p53 activity and the uses thereof
PL2562155T3 (en) 2010-04-20 2019-10-31 Fujifilm Toyama Chemical Co Ltd Hydroxamic acid derivative
WO2011150380A1 (en) 2010-05-28 2011-12-01 Xenoport, Inc. Methods of treatment of fragile x syndrome, down's syndrome, autism and related disorders
WO2012086241A1 (en) 2010-12-22 2012-06-28 Meiji Seikaファルマ株式会社 Optically-active diazabicyclooctane derivative and method for manufacturing same
US8772490B2 (en) 2010-12-22 2014-07-08 Meiji Seika Pharma Co., Ltd. Optically active diazabicyclooctane derivatives and process for preparing the same
HUE027447T2 (en) 2011-05-30 2016-09-28 Sumitomo Chemical Co Cyclohexanone compounds and herbicides comprising the same
US8796257B2 (en) 2011-12-02 2014-08-05 Naeja Pharmaceutical Inc. Bicyclic compounds and their use as antibacterial agents and β-lactamase inhibitors
AU2015316401A1 (en) 2014-09-12 2017-04-06 Fujifilm Toyama Chemical Co., Ltd. Novel pharmaceutical composition containing hydroxamic acid derivative or salt thereof
KR20170047390A (en) 2014-09-12 2017-05-04 토야마 케미칼 컴퍼니 리미티드 Method for using novel hydroxamic acid derivative and antibacterial substance in combination
WO2016116788A1 (en) 2015-01-24 2016-07-28 Wockhardt Limited Nitrogen containing bicyclic compounds and their use in treatment of bacterial infections
JP2018515481A (en) 2015-09-16 2018-06-14 シュアンチュー ファーマ カンパニー,リミティド β-lactamase inhibitors and uses thereof
US20170165371A1 (en) 2017-02-22 2017-06-15 Joel Steven Goldberg Novel synthesis of potential ester prodrugs
US10085999B1 (en) 2017-05-10 2018-10-02 Arixa Pharmaceuticals, Inc. Beta-lactamase inhibitors and uses thereof
JP6991345B2 (en) 2017-10-02 2022-01-12 アリクサ ファーマシューティカルズ、インコーポレイテッド Aztreonam derivatives and their use

Also Published As

Publication number Publication date
KR20210137159A (en) 2021-11-17
AU2020237440B2 (en) 2022-10-20
JP2022524118A (en) 2022-04-27
BR112021017874A2 (en) 2021-12-07
US11008321B2 (en) 2021-05-18
US20200291022A1 (en) 2020-09-17
AU2020237440A1 (en) 2021-09-09
CA3133071A1 (en) 2020-09-17
CN113614084A (en) 2021-11-05
MX2021011026A (en) 2021-10-13
WO2020185729A1 (en) 2020-09-17
EP3938366A1 (en) 2022-01-19

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