SG11201406550QA - Dosage regimen for a pi-3 kinase inhibitor - Google Patents

Dosage regimen for a pi-3 kinase inhibitor

Info

Publication number
SG11201406550QA
SG11201406550QA SG11201406550QA SG11201406550QA SG11201406550QA SG 11201406550Q A SG11201406550Q A SG 11201406550QA SG 11201406550Q A SG11201406550Q A SG 11201406550QA SG 11201406550Q A SG11201406550Q A SG 11201406550QA SG 11201406550Q A SG11201406550Q A SG 11201406550QA
Authority
SG
Singapore
Prior art keywords
kinase inhibitor
dosage regimen
regimen
dosage
kinase
Prior art date
Application number
SG11201406550QA
Inventor
Samit Hirawat
Cristian Massacesi
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48626588&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG11201406550Q(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of SG11201406550QA publication Critical patent/SG11201406550QA/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SG11201406550QA 2012-05-16 2013-05-14 Dosage regimen for a pi-3 kinase inhibitor SG11201406550QA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261647654P 2012-05-16 2012-05-16
PCT/US2013/040877 WO2013173283A1 (en) 2012-05-16 2013-05-14 Dosage regimen for a pi-3 kinase inhibitor

Publications (1)

Publication Number Publication Date
SG11201406550QA true SG11201406550QA (en) 2014-11-27

Family

ID=48626588

Family Applications (2)

Application Number Title Priority Date Filing Date
SG11201406550QA SG11201406550QA (en) 2012-05-16 2013-05-14 Dosage regimen for a pi-3 kinase inhibitor
SG10201608469RA SG10201608469RA (en) 2012-05-16 2013-05-14 Dosage regimen for a pi-3 kinase inhibitor

Family Applications After (1)

Application Number Title Priority Date Filing Date
SG10201608469RA SG10201608469RA (en) 2012-05-16 2013-05-14 Dosage regimen for a pi-3 kinase inhibitor

Country Status (19)

Country Link
US (2) US10213432B2 (en)
EP (1) EP2849756A1 (en)
JP (2) JP6381523B2 (en)
KR (1) KR20150009540A (en)
CN (1) CN104349779A (en)
AU (1) AU2013263043B2 (en)
BR (1) BR112014028420A2 (en)
CA (1) CA2872526A1 (en)
CL (1) CL2014003101A1 (en)
HK (1) HK1202435A1 (en)
IL (1) IL235567B (en)
MX (1) MX360892B (en)
NZ (1) NZ700924A (en)
PH (1) PH12014502547A1 (en)
RU (1) RU2630975C2 (en)
SG (2) SG11201406550QA (en)
TN (1) TN2014000433A1 (en)
WO (1) WO2013173283A1 (en)
ZA (1) ZA201407406B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX342326B (en) 2011-09-27 2016-09-26 Novartis Ag 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant idh.
UY34632A (en) 2012-02-24 2013-05-31 Novartis Ag OXAZOLIDIN- 2- ONA COMPOUNDS AND USES OF THE SAME
US9296733B2 (en) 2012-11-12 2016-03-29 Novartis Ag Oxazolidin-2-one-pyrimidine derivative and use thereof for the treatment of conditions, diseases and disorders dependent upon PI3 kinases
BR112015023412A8 (en) 2013-03-14 2018-01-23 Novartis Ag 3-pyrimidin-4-yl-oxazolidin-2-ones as mutant idh inhibitors, their pharmaceutical composition and their use.
BR112016011811A2 (en) 2013-12-06 2017-08-08 Novartis Ag USE OF AN ALPHA-ISOFORM SELECTIVE PHOSPHATIDYLINOSITOL 3-KINASE INHIBITOR, THERAPEUTIC REGIME AND PACKAGE
WO2016109426A1 (en) * 2014-12-29 2016-07-07 Verastem, Inc. Oral dosing regimen of a dual mtor and pi3 inhibitor
WO2017009751A1 (en) 2015-07-15 2017-01-19 Pfizer Inc. Pyrimidine derivatives
KR20180073674A (en) * 2015-11-02 2018-07-02 노파르티스 아게 Therapy for phosphatidylinositol 3-kinase inhibitors
WO2018009895A1 (en) * 2016-07-08 2018-01-11 Autotelic Llc Methods for trabedersen dosing by auc

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Also Published As

Publication number Publication date
JP2018108998A (en) 2018-07-12
SG10201608469RA (en) 2016-11-29
JP2015517523A (en) 2015-06-22
CL2014003101A1 (en) 2015-02-27
CA2872526A1 (en) 2013-11-21
US10213432B2 (en) 2019-02-26
PH12014502547A1 (en) 2015-01-21
IL235567B (en) 2019-08-29
RU2630975C2 (en) 2017-09-15
NZ700924A (en) 2016-02-26
JP6381523B2 (en) 2018-08-29
ZA201407406B (en) 2015-11-25
EP2849756A1 (en) 2015-03-25
US20150141426A1 (en) 2015-05-21
RU2014150860A (en) 2016-07-10
HK1202435A1 (en) 2015-10-02
US20190134052A1 (en) 2019-05-09
AU2013263043A1 (en) 2014-10-30
CN104349779A (en) 2015-02-11
TN2014000433A1 (en) 2016-03-30
AU2013263043B2 (en) 2016-06-16
MX360892B (en) 2018-11-20
WO2013173283A1 (en) 2013-11-21
IL235567A0 (en) 2015-01-29
BR112014028420A2 (en) 2017-09-19
MX2014013904A (en) 2015-01-16
KR20150009540A (en) 2015-01-26

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