NO20054905L - 2-acylamino-4-fenyltiazolderivater, fremgangsmate for deres fremstilling og anvendelse av de samme som i terapeutika - Google Patents

2-acylamino-4-fenyltiazolderivater, fremgangsmate for deres fremstilling og anvendelse av de samme som i terapeutika

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Publication number
NO20054905L
NO20054905L NO20054905A NO20054905A NO20054905L NO 20054905 L NO20054905 L NO 20054905L NO 20054905 A NO20054905 A NO 20054905A NO 20054905 A NO20054905 A NO 20054905A NO 20054905 L NO20054905 L NO 20054905L
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Norway
Prior art keywords
acylamino
preparation
same
therapeutics
methods
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NO20054905A
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English (en)
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NO20054905D0 (no
Inventor
Bernard Labeeuw
Pierre Casellas
Samir Jegham
Pierre Carayon
Daniel Floutard
Pierre Fraisse
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Sanofi Aventis
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Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of NO20054905D0 publication Critical patent/NO20054905D0/no
Publication of NO20054905L publication Critical patent/NO20054905L/no

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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10—Spiro-condensed systems
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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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Abstract

Oppfinnelsen vedrører derivater av 2-acylamino-4-fenyltiazol med den generelle formel (I). Oppfinnelsen vedrører også en fremgangsmåte for fremstilling derav og anvendelse av de samme i terapeutiske midler.
NO20054905A 2003-04-25 2005-10-24 2-acylamino-4-fenyltiazolderivater, fremgangsmate for deres fremstilling og anvendelse av de samme som i terapeutika NO20054905L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0305213A FR2854158B1 (fr) 2003-04-25 2003-04-25 Derives de 2-acylamino-4-phenylethiazole, leur preparation et leur application en therapeutique
PCT/FR2004/000981 WO2004096798A2 (fr) 2003-04-25 2004-04-22 Derives de 2-acylamino-4-phenylthiazole, leur preparation et leur application en therapeutique

Publications (2)

Publication Number Publication Date
NO20054905D0 NO20054905D0 (no) 2005-10-24
NO20054905L true NO20054905L (no) 2006-01-25

Family

ID=33104460

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20054905A NO20054905L (no) 2003-04-25 2005-10-24 2-acylamino-4-fenyltiazolderivater, fremgangsmate for deres fremstilling og anvendelse av de samme som i terapeutika

Country Status (24)

Country Link
US (2) US7504511B2 (no)
EP (1) EP1656373B1 (no)
JP (2) JP4839208B2 (no)
KR (1) KR20060006935A (no)
CN (1) CN1826339A (no)
AR (1) AR044070A1 (no)
AT (1) ATE541843T1 (no)
AU (1) AU2004234101A1 (no)
BR (1) BRPI0409716A (no)
CA (1) CA2521158A1 (no)
CO (1) CO5640106A2 (no)
CR (1) CR8037A (no)
EC (1) ECSP056111A (no)
FR (1) FR2854158B1 (no)
MA (1) MA27769A1 (no)
MX (1) MXPA05011522A (no)
NO (1) NO20054905L (no)
OA (1) OA13049A (no)
RS (1) RS20050769A (no)
RU (1) RU2348630C2 (no)
TN (1) TNSN05254A1 (no)
TW (1) TW200510325A (no)
WO (1) WO2004096798A2 (no)
ZA (1) ZA200508608B (no)

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JO2676B1 (en) * 2004-04-06 2012-06-17 جانسين فارماسوتيكا ان. في Derivatives of second-aza-spiro- (5,4) -dikan and their use as antihistamines
FR2872813B1 (fr) 2004-07-09 2007-01-19 Sanofi Synthelabo Derives de 2-carbamide-4-phenylthiazole, leur preparation et leur application en therapeutique
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RU2348630C2 (ru) 2009-03-10
CR8037A (es) 2008-07-29
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OA13049A (fr) 2006-11-10
FR2854158B1 (fr) 2006-11-17
US7777041B2 (en) 2010-08-17
CO5640106A2 (es) 2006-05-31
US7504511B2 (en) 2009-03-17
ZA200508608B (en) 2007-01-31
ATE541843T1 (de) 2012-02-15
KR20060006935A (ko) 2006-01-20
CA2521158A1 (fr) 2004-11-11
US20060135575A1 (en) 2006-06-22
CN1826339A (zh) 2006-08-30
FR2854158A1 (fr) 2004-10-29
TNSN05254A1 (en) 2007-07-10
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AR044070A1 (es) 2005-08-24
JP2006524669A (ja) 2006-11-02
EP1656373B1 (fr) 2012-01-18
NO20054905D0 (no) 2005-10-24
WO2004096798A2 (fr) 2004-11-11
ECSP056111A (es) 2006-03-01
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TW200510325A (en) 2005-03-16
BRPI0409716A (pt) 2006-05-02
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US20090156574A1 (en) 2009-06-18
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