MXPA05013469A - Derivados de piperazina y metodos de uso. - Google Patents

Derivados de piperazina y metodos de uso.

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Publication number
MXPA05013469A
MXPA05013469A MXPA05013469A MXPA05013469A MXPA05013469A MX PA05013469 A MXPA05013469 A MX PA05013469A MX PA05013469 A MXPA05013469 A MX PA05013469A MX PA05013469 A MXPA05013469 A MX PA05013469A MX PA05013469 A MXPA05013469 A MX PA05013469A
Authority
MX
Mexico
Prior art keywords
methods
diseases
compounds
processes
treatment
Prior art date
Application number
MXPA05013469A
Other languages
English (en)
Inventor
Tanya Peterkin
Original Assignee
Amgen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amgen Inc filed Critical Amgen Inc
Publication of MXPA05013469A publication Critical patent/MXPA05013469A/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
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    • C07D243/08—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 not condensed with other rings
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Cardiology (AREA)
  • Addiction (AREA)
  • Molecular Biology (AREA)
  • Psychiatry (AREA)
  • Vascular Medicine (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Toxicology (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)

Abstract

Se describen los compuestos seleccionados que son efectivos para el tratamiento de dolor y enfermedades, tales como enfermedades mediadas por la inflamacion. La invencion abarca los nuevos compuestos, analogos, profarmacos y derivados farmaceuticamente aceptables de los mismos, las composiciones farmaceuticas y los metodos para la profilaxis y tratamiento de las enfermedades y otros trastornos o condiciones que involucran dolor, inflamaciones y similares. La presente invencion tambien se refiere a los procesos para elaborar tales compuestos, asi como a los intermediarios utiles en tales procesos, asi como los intermediarios utiles en tales procesos.
MXPA05013469A 2003-06-20 2004-06-21 Derivados de piperazina y metodos de uso. MXPA05013469A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US48030303P 2003-06-20 2003-06-20
PCT/US2004/019935 WO2005061467A2 (en) 2003-06-20 2004-06-21 Piperazine derivatives as bradykinin antagonists

Publications (1)

Publication Number Publication Date
MXPA05013469A true MXPA05013469A (es) 2006-03-09

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MXPA05013469A MXPA05013469A (es) 2003-06-20 2004-06-21 Derivados de piperazina y metodos de uso.

Country Status (18)

Country Link
US (2) US7393852B2 (es)
EP (1) EP1656355B1 (es)
JP (1) JP2007516176A (es)
KR (1) KR20060036399A (es)
CN (1) CN1849121A (es)
AT (1) ATE388708T1 (es)
AU (1) AU2004303757B2 (es)
BR (1) BRPI0411673A (es)
CA (1) CA2529314A1 (es)
DE (1) DE602004012418T2 (es)
ES (1) ES2302079T3 (es)
IL (1) IL172419A0 (es)
IS (1) IS8175A (es)
MX (1) MXPA05013469A (es)
NO (1) NO20060278L (es)
RU (1) RU2006101541A (es)
WO (1) WO2005061467A2 (es)
ZA (1) ZA200600579B (es)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7328349B2 (en) 2001-12-14 2008-02-05 Bbn Technologies Corp. Hash-based systems and methods for detecting, preventing, and tracing network worms and viruses
US20040073617A1 (en) 2000-06-19 2004-04-15 Milliken Walter Clark Hash-based systems and methods for detecting and preventing transmission of unwanted e-mail
US7200105B1 (en) * 2001-01-12 2007-04-03 Bbn Technologies Corp. Systems and methods for point of ingress traceback of a network attack
BRPI0411673A (pt) * 2003-06-20 2006-08-08 Amgen Inc composto, sal farmaceuticamente aceitável, composição farmacêutica, e, uso de um composto
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