MX2009013815A - Compuestos de quinazolinona y metodos de uso para los mismos. - Google Patents
Compuestos de quinazolinona y metodos de uso para los mismos.Info
- Publication number
- MX2009013815A MX2009013815A MX2009013815A MX2009013815A MX2009013815A MX 2009013815 A MX2009013815 A MX 2009013815A MX 2009013815 A MX2009013815 A MX 2009013815A MX 2009013815 A MX2009013815 A MX 2009013815A MX 2009013815 A MX2009013815 A MX 2009013815A
- Authority
- MX
- Mexico
- Prior art keywords
- methods
- present
- compounds
- quinazolinone
- quinazolinone compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
- C07D239/90—Oxygen atoms with acyclic radicals attached in position 2 or 3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
Abstract
La presente invención se refiere a compuestos de quinazolinona, y métodos de preparación de estos compuestos; la presente invención también se refiere a composiciones farmacéuticas que comprenden los compuestos de quinazolinona; la presente invención proporciona métodos para tratar un trastorno proliferativo celular, tal como cáncer, al administrar a un sujeto en necesidad del mismo, una cantidad terapéuticamente efectiva de un compuesto de quinazolinona de la presente invención.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US94583807P | 2007-06-22 | 2007-06-22 | |
PCT/US2008/067571 WO2009002808A2 (en) | 2007-06-22 | 2008-06-19 | Quinazolinone compounds and methods of use thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2009013815A true MX2009013815A (es) | 2010-03-01 |
Family
ID=39846620
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2009013815A MX2009013815A (es) | 2007-06-22 | 2008-06-19 | Compuestos de quinazolinona y metodos de uso para los mismos. |
Country Status (13)
Country | Link |
---|---|
US (1) | US8232285B2 (es) |
EP (1) | EP2173724B1 (es) |
JP (1) | JP2010530885A (es) |
KR (1) | KR20100024494A (es) |
CN (1) | CN101801937A (es) |
AU (1) | AU2008268613A1 (es) |
BR (1) | BRPI0813355A2 (es) |
CA (1) | CA2704282A1 (es) |
IL (1) | IL202740A0 (es) |
MX (1) | MX2009013815A (es) |
TW (1) | TW200918069A (es) |
WO (1) | WO2009002808A2 (es) |
ZA (1) | ZA201000183B (es) |
Families Citing this family (15)
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US8268807B2 (en) * | 2010-04-19 | 2012-09-18 | Sri International | Compositions and method for the treatment of multiple myeloma |
US8940742B2 (en) | 2012-04-10 | 2015-01-27 | Infinity Pharmaceuticals, Inc. | Heterocyclic compounds and uses thereof |
WO2015051241A1 (en) | 2013-10-04 | 2015-04-09 | Infinity Pharmaceuticals, Inc. | Heterocyclic compounds and uses thereof |
CA2925944C (en) | 2013-10-04 | 2023-01-10 | Infinity Pharmaceuticals, Inc. | Heterocyclic compounds and uses thereof |
US20150132575A1 (en) * | 2013-11-14 | 2015-05-14 | Honeywell International Inc. | Luminescent fibers, articles including the same, and methods of forming the same |
EP4066834A1 (en) | 2014-03-19 | 2022-10-05 | Infinity Pharmaceuticals, Inc. | Heterocyclic compounds for use in the treatment of pi3k-gamma mediated disorders |
WO2016054491A1 (en) | 2014-10-03 | 2016-04-07 | Infinity Pharmaceuticals, Inc. | Heterocyclic compounds and uses thereof |
CN108349985A (zh) | 2015-09-14 | 2018-07-31 | 无限药品股份有限公司 | 异喹啉酮的固体形式、其制备方法、包含其的组合物及其使用方法 |
US10759806B2 (en) | 2016-03-17 | 2020-09-01 | Infinity Pharmaceuticals, Inc. | Isotopologues of isoquinolinone and quinazolinone compounds and uses thereof as PI3K kinase inhibitors |
US10919914B2 (en) | 2016-06-08 | 2021-02-16 | Infinity Pharmaceuticals, Inc. | Heterocyclic compounds and uses thereof |
TW201813963A (zh) | 2016-09-23 | 2018-04-16 | 美商基利科學股份有限公司 | 磷脂醯肌醇3-激酶抑制劑 |
TW201815787A (zh) | 2016-09-23 | 2018-05-01 | 美商基利科學股份有限公司 | 磷脂醯肌醇3-激酶抑制劑 |
TW201825465A (zh) | 2016-09-23 | 2018-07-16 | 美商基利科學股份有限公司 | 磷脂醯肌醇3-激酶抑制劑 |
WO2019217957A1 (en) * | 2018-05-11 | 2019-11-14 | The United States Of America, As Represented By The Secretary, Department Of Health And Human Services | Quinoline compounds and their preparation and use as antimalarial agents |
CN113354590A (zh) * | 2020-03-05 | 2021-09-07 | 宁波康柏睿格医药科技有限公司 | 拮抗nod1/2受体信号通路的喹唑啉酮类化合物 |
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-
2008
- 2008-06-19 AU AU2008268613A patent/AU2008268613A1/en not_active Abandoned
- 2008-06-19 WO PCT/US2008/067571 patent/WO2009002808A2/en active Application Filing
- 2008-06-19 CA CA2704282A patent/CA2704282A1/en not_active Abandoned
- 2008-06-19 MX MX2009013815A patent/MX2009013815A/es not_active Application Discontinuation
- 2008-06-19 CN CN200880104552A patent/CN101801937A/zh active Pending
- 2008-06-19 KR KR1020107001013A patent/KR20100024494A/ko not_active Application Discontinuation
- 2008-06-19 EP EP08771527A patent/EP2173724B1/en active Active
- 2008-06-19 JP JP2010513424A patent/JP2010530885A/ja not_active Withdrawn
- 2008-06-19 US US12/142,762 patent/US8232285B2/en active Active
- 2008-06-19 BR BRPI0813355-7A2A patent/BRPI0813355A2/pt not_active IP Right Cessation
- 2008-06-20 TW TW097123156A patent/TW200918069A/zh unknown
-
2009
- 2009-12-15 IL IL202740A patent/IL202740A0/en unknown
-
2010
- 2010-01-11 ZA ZA2010/00183A patent/ZA201000183B/en unknown
Also Published As
Publication number | Publication date |
---|---|
IL202740A0 (en) | 2010-06-30 |
EP2173724B1 (en) | 2012-12-05 |
AU2008268613A1 (en) | 2008-12-31 |
US20090130097A1 (en) | 2009-05-21 |
WO2009002808A3 (en) | 2009-07-23 |
CA2704282A1 (en) | 2008-12-31 |
ZA201000183B (en) | 2011-03-30 |
EP2173724A2 (en) | 2010-04-14 |
US8232285B2 (en) | 2012-07-31 |
KR20100024494A (ko) | 2010-03-05 |
TW200918069A (en) | 2009-05-01 |
CN101801937A (zh) | 2010-08-11 |
JP2010530885A (ja) | 2010-09-16 |
BRPI0813355A2 (pt) | 2014-12-30 |
WO2009002808A2 (en) | 2008-12-31 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
HH | Correction or change in general | ||
FA | Abandonment or withdrawal |