JOP20210047A1 - عامل وقائي و/أو علاجي للأعراض السلوكية والنفسية المصحوبة بمرض تنكسي عصبي أو الأعراض الإندفاعية المصحوبة بمرض ذهني، يحتوي على بريكسبيرازول أو ملحه - Google Patents

عامل وقائي و/أو علاجي للأعراض السلوكية والنفسية المصحوبة بمرض تنكسي عصبي أو الأعراض الإندفاعية المصحوبة بمرض ذهني، يحتوي على بريكسبيرازول أو ملحه

Info

Publication number
JOP20210047A1
JOP20210047A1 JOP/2021/0047A JOP20210047A JOP20210047A1 JO P20210047 A1 JOP20210047 A1 JO P20210047A1 JO P20210047 A JOP20210047 A JO P20210047A JO P20210047 A1 JOP20210047 A1 JO P20210047A1
Authority
JO
Jordan
Prior art keywords
symptoms associated
behavioral
prophylactic
salt
therapeutic agent
Prior art date
Application number
JOP/2021/0047A
Other languages
English (en)
Inventor
Ishikawa Dai
Sato Shinji
Maeda Kenji
Nakamura Mai
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of JOP20210047A1 publication Critical patent/JOP20210047A1/ar

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Dermatology (AREA)

Abstract

يتعلق هذا الاختراع بعامل وقائي و/أو علاجي للأعراض السلوكية والنفسية المصاحبة لمرض تنكسي عصبي أو الأعراض الاندفاعية المصاحبة للمرض العقلي، والذي يحتوي على المركب 7 - [4 - (4-بنزو [ب] –ثيوفين-4-يل-بيبرازين-1-يل)بوتوكسي]-1 اتش- كينولين-2-ون أو ملحه كمركب فعال او كعنصر فعال.
JOP/2021/0047A 2012-10-25 2012-10-25 عامل وقائي و/أو علاجي للأعراض السلوكية والنفسية المصحوبة بمرض تنكسي عصبي أو الأعراض الإندفاعية المصحوبة بمرض ذهني، يحتوي على بريكسبيرازول أو ملحه JOP20210047A1 (ar)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261718305P 2012-10-25 2012-10-25
US201361782467P 2013-03-14 2013-03-14

Publications (1)

Publication Number Publication Date
JOP20210047A1 true JOP20210047A1 (ar) 2017-06-16

Family

ID=49585556

Family Applications (2)

Application Number Title Priority Date Filing Date
JOP/2021/0047A JOP20210047A1 (ar) 2012-10-25 2012-10-25 عامل وقائي و/أو علاجي للأعراض السلوكية والنفسية المصحوبة بمرض تنكسي عصبي أو الأعراض الإندفاعية المصحوبة بمرض ذهني، يحتوي على بريكسبيرازول أو ملحه
JOP/2013/0313A JOP20130313B1 (ar) 2012-10-25 2013-10-24 عامل وقائي و/أو علاجي للأعراض السلوكية والنفسية المصحوبة بمرض تنكسي عصبي أو الأعراض الإندفاعية المصحوبة بمرض ذهني، يحتوي على بريكسبيرازول أو ملحه

Family Applications After (1)

Application Number Title Priority Date Filing Date
JOP/2013/0313A JOP20130313B1 (ar) 2012-10-25 2013-10-24 عامل وقائي و/أو علاجي للأعراض السلوكية والنفسية المصحوبة بمرض تنكسي عصبي أو الأعراض الإندفاعية المصحوبة بمرض ذهني، يحتوي على بريكسبيرازول أو ملحه

Country Status (22)

Country Link
US (4) US20150272946A1 (ar)
EP (2) EP3848033A1 (ar)
JP (5) JP6329140B2 (ar)
KR (1) KR102245016B1 (ar)
CN (4) CN112402421A (ar)
AR (1) AR093247A1 (ar)
AU (1) AU2013335613B2 (ar)
BR (1) BR112015008759A2 (ar)
CA (1) CA2889196C (ar)
EA (1) EA201590808A1 (ar)
HK (1) HK1212609A1 (ar)
IL (1) IL238402B (ar)
JO (2) JOP20210047A1 (ar)
MX (1) MX371279B (ar)
MY (1) MY180185A (ar)
NZ (1) NZ708321A (ar)
PH (1) PH12015500925B1 (ar)
SG (2) SG11201503152TA (ar)
TW (1) TWI643620B (ar)
UA (1) UA116549C2 (ar)
WO (1) WO2014065437A1 (ar)
ZA (1) ZA201503640B (ar)

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TWI415845B (zh) 2006-10-03 2013-11-21 Arena Pharm Inc 用於治療與５-ｈｔ2ａ血清素受體相關聯病症之作為５-ｈｔ2ａ血清素受體之調節劑的吡唑衍生物
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WO2009123714A2 (en) 2008-04-02 2009-10-08 Arena Pharmaceuticals, Inc. Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor
US9126946B2 (en) 2008-10-28 2015-09-08 Arena Pharmaceuticals, Inc. Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)urea and crystalline forms related thereto
NO2364142T3 (ar) 2008-10-28 2018-06-16
BR112016024510A2 (pt) 2014-04-22 2017-08-15 H Lundbeck As ?medicamento, uso de brexpiprazol ou de um sal farmaceuticamente aceitável do mesmo, métodos para prevenção ou tratamento de um transtorno relacionado com substância e para produção de uma composição farmacêutica, composição farmacêutica, e, kit?
WO2016115144A1 (en) * 2015-01-12 2016-07-21 Reviva Pharmaceuticals Inc. Methods for treating alzheimer's disease
WO2016115150A1 (en) * 2015-01-12 2016-07-21 Reviva Pharmaceuticals Inc. Methods for treating psychosis associated with parkinson's disease
AU2016276966A1 (en) 2015-06-12 2018-01-18 Axovant Sciences Gmbh Diaryl and arylheteroaryl urea derivatives useful for the prophylaxis and treatment of REM sleep behavior disorder
JP2018520187A (ja) * 2015-07-15 2018-07-26 アクソヴァント サイエンシーズ ゲゼルシャフト ミット ベシュレンクテル ハフツングAxovant Sciences GmbH 神経変性疾患と関連する幻覚の予防および処置のために有用な５−ｈｔ２ａセロトニン受容体のモジュレーターとしてのジアリールおよびアリールヘテロアリール尿素誘導体
CN105175401A (zh) * 2015-10-16 2015-12-23 北京康立生医药技术开发有限公司 一种依匹哌唑的制备方法
CN105541819B (zh) * 2016-02-04 2018-09-14 浙江永宁药业股份有限公司 一种依匹唑派的制备方法及其中间体和中间体的制备方法
CN115813888A (zh) 2016-12-20 2023-03-21 罗曼治疗系统股份公司 包含阿塞那平的透皮治疗系统
US11337932B2 (en) 2016-12-20 2022-05-24 Lts Lohmann Therapie-Systeme Ag Transdermal therapeutic system containing asenapine and polysiloxane or polyisobutylene
WO2019002204A1 (en) 2017-06-26 2019-01-03 Lts Lohmann Therapie-Systeme Ag TRANSDERMAL THERAPEUTIC SYSTEM CONTAINING ASENAPINE AND SILICONE-TYPE ACRYLIC HYBRID POLYMER
KR20200110317A (ko) 2017-12-05 2020-09-23 선오비온 파마슈티컬스 인코포레이티드 결정형 및 이의 제조 방법
EP3720434A4 (en) 2017-12-05 2021-09-01 Sunovion Pharmaceuticals Inc. NON-RACEMIC MIXTURES AND THEIR USE
EP3501506B1 (en) 2017-12-19 2019-10-09 Alfred E. Tiefenbacher (GmbH & Co. KG) Pharmaceutical tablet composition comprising brexpiprazole
CN112704672A (zh) 2018-06-20 2021-04-27 罗曼治疗系统股份公司 含有阿塞那平的透皮治疗系统
AU2020286441A1 (en) 2019-06-04 2022-01-06 Sunovion Pharmaceuticals Inc. Modified release formulations and uses thereof
JPWO2021029020A1 (ar) * 2019-08-13 2021-02-18
BR112022026067A2 (pt) * 2020-06-24 2023-01-17 Univ Hokkaido Nat Univ Corp Agentes de proteção de células endoteliais vasculares, da barreira hematoencefálica da medula espinhal e do sistema nervoso central, e, composição farmacêutica para prevenir e/ou tratar uma doença acompanhada de um distúrbio da barreira hematoencefálica da medula espinhal
CN112137994B (zh) * 2020-09-15 2022-10-14 中山大学 小分子化合物在制备抗丝状病毒药物中的应用
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JP4315393B2 (ja) 2005-04-14 2009-08-19 大塚製薬株式会社 複素環化合物
JP4540700B2 (ja) * 2006-10-13 2010-09-08 大塚製薬株式会社 医薬
JP2011136906A (ja) * 2008-04-18 2011-07-14 Otsuka Pharmaceut Co Ltd 複素環化合物
AR085840A1 (es) * 2011-04-05 2013-10-30 Otsuka Pharma Co Ltd Medicamento que contiene un compuesto que es 7-[4-(4-benzo[b]tiofen-4-il-piperazin-1-il)butoxi]-1h-quinolin-2-ona
TWI562991B (en) * 2012-04-23 2016-12-21 Otsuka Pharma Co Ltd Dihydrate of benzothiophene compound or of a salt thereof, and process for producing the same
AR090775A1 (es) * 2012-04-23 2014-12-03 Otsuka Pharma Co Ltd Preparado inyectable
EP2822136B1 (en) * 2013-07-03 2018-08-29 Siemens Aktiengesellschaft Method and arrangement for transferring electrical power for subsea applications

Also Published As

Publication number Publication date
WO2014065437A1 (en) 2014-05-01
EA201590808A1 (ru) 2015-08-31
PH12015500925A1 (en) 2015-06-29
EP3848033A1 (en) 2021-07-14
SG10201702828TA (en) 2017-05-30
JP2021181448A (ja) 2021-11-25
AU2013335613B2 (en) 2018-07-12
CN112402421A (zh) 2021-02-26
BR112015008759A2 (pt) 2017-07-04
JP2023123441A (ja) 2023-09-05
AR093247A1 (es) 2015-05-27
CA2889196A1 (en) 2014-05-01
TW201427665A (zh) 2014-07-16
KR102245016B1 (ko) 2021-04-26
NZ708321A (en) 2019-03-29
KR20150074156A (ko) 2015-07-01
SG11201503152TA (en) 2015-05-28
MX2015005174A (es) 2015-09-04
CN114712360A (zh) 2022-07-08
UA116549C2 (uk) 2018-04-10
CN104755082A (zh) 2015-07-01
US20150272946A1 (en) 2015-10-01
CN108578408A (zh) 2018-09-28
ZA201503640B (en) 2016-08-31
IL238402B (en) 2018-11-29
US20190314367A1 (en) 2019-10-17
IL238402A0 (en) 2015-06-30
US20170258787A1 (en) 2017-09-14
PH12015500925B1 (en) 2015-06-29
TWI643620B (zh) 2018-12-11
JP2020045345A (ja) 2020-03-26
JP2018138555A (ja) 2018-09-06
JP6329140B2 (ja) 2018-05-23
US20220370442A1 (en) 2022-11-24
MX371279B (es) 2020-01-24
CA2889196C (en) 2021-02-16
HK1212609A1 (zh) 2016-06-17
AU2013335613A1 (en) 2015-06-04
JP2015535211A (ja) 2015-12-10
EP2911670A1 (en) 2015-09-02
MY180185A (en) 2020-11-24
JOP20130313B1 (ar) 2021-08-17

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