IT1176770B - DERIVATIVES OF BENZOSSAZOLONE AND BENZOTIAZOLONE PRO CEDIMENTS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOUND THAT CONTAINS THEM - Google Patents

DERIVATIVES OF BENZOSSAZOLONE AND BENZOTIAZOLONE PRO CEDIMENTS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOUND THAT CONTAINS THEM

Info

Publication number
IT1176770B
IT1176770B IT2278584A IT2278584A IT1176770B IT 1176770 B IT1176770 B IT 1176770B IT 2278584 A IT2278584 A IT 2278584A IT 2278584 A IT2278584 A IT 2278584A IT 1176770 B IT1176770 B IT 1176770B
Authority
IT
Italy
Prior art keywords
cediments
benzotiazolone
benzossazolone
pro
derivatives
Prior art date
Application number
IT2278584A
Other languages
Italian (it)
Other versions
IT8422785A0 (en
IT8422785A1 (en
Original Assignee
Fujisawa Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co
Publication of IT8422785A0 publication Critical patent/IT8422785A0/en
Publication of IT8422785A1 publication Critical patent/IT8422785A1/en
Application granted granted Critical
Publication of IT1176770B publication Critical patent/IT1176770B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT2278584A 1983-09-22 1984-09-21 DERIVATIVES OF BENZOSSAZOLONE AND BENZOTIAZOLONE PRO CEDIMENTS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOUND THAT CONTAINS THEM IT1176770B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB838325370A GB8325370D0 (en) 1983-09-22 1983-09-22 Benzoxazoline and benzothiazoline derivatives

Publications (3)

Publication Number Publication Date
IT8422785A0 IT8422785A0 (en) 1984-09-21
IT8422785A1 IT8422785A1 (en) 1986-03-21
IT1176770B true IT1176770B (en) 1987-08-18

Family

ID=10549143

Family Applications (1)

Application Number Title Priority Date Filing Date
IT2278584A IT1176770B (en) 1983-09-22 1984-09-21 DERIVATIVES OF BENZOSSAZOLONE AND BENZOTIAZOLONE PRO CEDIMENTS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOUND THAT CONTAINS THEM

Country Status (4)

Country Link
AU (1) AU3431784A (en)
GB (1) GB8325370D0 (en)
IT (1) IT1176770B (en)
WO (1) WO1985001289A1 (en)

Cited By (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010129596A1 (en) * 2009-05-04 2010-11-11 Agios Pharmaceuticals, Inc. Pmk2 modulators for use in the treatment of cancer
US8742119B2 (en) 2009-04-06 2014-06-03 Agios Pharmaceuticals, Inc. Pyruvate kinase M2 modulators, therapeutic compositions and related methods of use
US8889667B2 (en) 2010-12-29 2014-11-18 Agios Pharmaceuticals, Inc Therapeutic compounds and compositions
US9115086B2 (en) 2009-06-29 2015-08-25 Agios Pharmaceuticals, Inc. Therapeutic compositions and related methods of use
US9181231B2 (en) 2011-05-03 2015-11-10 Agios Pharmaceuticals, Inc Pyruvate kinase activators for use for increasing lifetime of the red blood cells and treating anemia
US9221792B2 (en) 2010-12-17 2015-12-29 Agios Pharmaceuticals, Inc N-(4-(azetidine-1-carbonyl) phenyl)-(hetero-) arylsulfonamide derivatives as pyruvate kinase M2 (PMK2) modulators
US9328077B2 (en) 2010-12-21 2016-05-03 Agios Pharmaceuticals, Inc Bicyclic PKM2 activators
US9365545B2 (en) 2013-03-15 2016-06-14 Agios Pharmaceuticals, Inc Therapeutic compounds and compositions
US9980961B2 (en) 2011-05-03 2018-05-29 Agios Pharmaceuticals, Inc. Pyruvate kinase activators for use in therapy
US10029987B2 (en) 2009-06-29 2018-07-24 Agios Pharmaceuticals, Inc. Therapeutic compounds and compositions
US11234976B2 (en) 2015-06-11 2022-02-01 Agios Pharmaceuticals, Inc. Methods of using pyruvate kinase activators

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK288287A (en) * 1986-06-09 1987-12-10 Pfizer HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL PREPARATIONS FOR TREATMENT OF ALLERGIC OR INFLAMMATORY CONDITIONS
JPH0283376A (en) * 1988-09-19 1990-03-23 Pfizer Pharmaceut Co Ltd Benzoxazolone derivative and antiallergic or anti-inflammatory composition
IL93473A0 (en) * 1989-02-28 1990-11-29 Pfizer Antiinflammatory benzoxazolones
FR2646350B1 (en) * 1989-04-28 1991-06-28 Adir NOVEL BENZOTHIAZOLINON DERIVATIVES, THEIR PREPARATION PROCESS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME
US5166353A (en) * 1989-04-28 1992-11-24 Adir Et Compagnie Benzothiazolinone compounds
JPH0678327B2 (en) * 1989-07-20 1994-10-05 ファイザー製薬株式会社 4,5,6,7, -tetrasubstituted benzoxazolones
JPH06759B2 (en) * 1989-09-22 1994-01-05 ファイザー製薬株式会社 Novel benzimidazole compound
JPH0717589B2 (en) * 1990-01-22 1995-03-01 ファイザー製薬株式会社 Novel 1,3-dicarbonyl compound and composition thereof
US7022480B1 (en) 2001-10-11 2006-04-04 The Regents Of The University Of California Exons of the hSKCa3/KCNN3 gene

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2244506B1 (en) * 1973-06-26 1977-02-25 Inst Nat Sante Rech Med
FR2244507A1 (en) * 1973-06-26 1975-04-18 Inst Nat Sante Rech Med Chalcones and analogues - analgesics having low toxicity
DE2634787C2 (en) * 1976-08-03 1983-01-27 Hoechst Ag, 6000 Frankfurt Process for the preparation of sulfuric acid half-ester compounds and their use
JPS5697268A (en) * 1979-12-28 1981-08-05 Fujisawa Pharmaceut Co Ltd Lower alkanoic acid derivative, salt and preparation thereof and preventing agent and remedy for diabetic complication containing the same as active constituent
FR2491066A1 (en) * 1980-09-29 1982-04-02 Cerm Cent Europ Rech Mauvernay BENZOXAZOLINONES SUBSTITUTED IN 6 BY AN AMINOALCOHOL OR AMINOCETONE CHAIN, THEIR PREPARATION AND THEIR THERAPEUTIC USE

Cited By (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9657004B2 (en) 2009-04-06 2017-05-23 Agios Pharmaceuticals, Inc Pyruvate kinase M2 modulators, therapeutic compositions and related methods of use
US8742119B2 (en) 2009-04-06 2014-06-03 Agios Pharmaceuticals, Inc. Pyruvate kinase M2 modulators, therapeutic compositions and related methods of use
US9938259B2 (en) 2009-04-06 2018-04-10 Agios Pharmaceuticals, Inc. Therapeutic compositions and related methods of use
WO2010129596A1 (en) * 2009-05-04 2010-11-11 Agios Pharmaceuticals, Inc. Pmk2 modulators for use in the treatment of cancer
US10988448B2 (en) 2009-06-29 2021-04-27 Agios Pharmaceuticals, Inc. Therapeutic compounds and compositions
US11866411B2 (en) 2009-06-29 2024-01-09 Agios Pharmaceutical, Inc. Therapeutic compounds and compositions
USRE49582E1 (en) 2009-06-29 2023-07-18 Agios Pharmaceuticals, Inc. Therapeutic compounds and compositions
US9115086B2 (en) 2009-06-29 2015-08-25 Agios Pharmaceuticals, Inc. Therapeutic compositions and related methods of use
US10029987B2 (en) 2009-06-29 2018-07-24 Agios Pharmaceuticals, Inc. Therapeutic compounds and compositions
US9221792B2 (en) 2010-12-17 2015-12-29 Agios Pharmaceuticals, Inc N-(4-(azetidine-1-carbonyl) phenyl)-(hetero-) arylsulfonamide derivatives as pyruvate kinase M2 (PMK2) modulators
US9328077B2 (en) 2010-12-21 2016-05-03 Agios Pharmaceuticals, Inc Bicyclic PKM2 activators
US10087169B2 (en) 2010-12-21 2018-10-02 Agios Pharmaceuticals, Inc. Bicyclic PKM2 activators
US9199968B2 (en) 2010-12-29 2015-12-01 Agios Pharmaceuticals, Inc. Therapeutic compounds and compositions
US8889667B2 (en) 2010-12-29 2014-11-18 Agios Pharmaceuticals, Inc Therapeutic compounds and compositions
US10632114B2 (en) 2011-05-03 2020-04-28 Agios Pharmaceuticals, Inc. Pyruvate kinase activators for use in therapy
US9980961B2 (en) 2011-05-03 2018-05-29 Agios Pharmaceuticals, Inc. Pyruvate kinase activators for use in therapy
US9181231B2 (en) 2011-05-03 2015-11-10 Agios Pharmaceuticals, Inc Pyruvate kinase activators for use for increasing lifetime of the red blood cells and treating anemia
US11793806B2 (en) 2011-05-03 2023-10-24 Agios Pharmaceuticals, Inc. Pyruvate kinase activators for use in therapy
US9365545B2 (en) 2013-03-15 2016-06-14 Agios Pharmaceuticals, Inc Therapeutic compounds and compositions
US11234976B2 (en) 2015-06-11 2022-02-01 Agios Pharmaceuticals, Inc. Methods of using pyruvate kinase activators

Also Published As

Publication number Publication date
WO1985001289A1 (en) 1985-03-28
IT8422785A0 (en) 1984-09-21
IT8422785A1 (en) 1986-03-21
AU3431784A (en) 1985-04-23
GB8325370D0 (en) 1983-10-26

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