FR2290443A1 - Antibacterial bis-penicillin esters - contg. and alkanedioyloxymethyl alcohol residue - Google Patents
Antibacterial bis-penicillin esters - contg. and alkanedioyloxymethyl alcohol residueInfo
- Publication number
- FR2290443A1 FR2290443A1 FR7436775A FR7436775A FR2290443A1 FR 2290443 A1 FR2290443 A1 FR 2290443A1 FR 7436775 A FR7436775 A FR 7436775A FR 7436775 A FR7436775 A FR 7436775A FR 2290443 A1 FR2290443 A1 FR 2290443A1
- Authority
- FR
- France
- Prior art keywords
- penicillin
- alkanedioyloxymethyl
- contg
- och
- alcohol residue
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Penicillin derivs. of formula (I) are new: (where A and A' (same or different) are direct bonds or divalent gps. selected from 5-methyl-3,4-isoxazolylene, (MIO) CH2,OCH2,OCH(Me), OCH(Et), OCH(Ph), CH(OMe), CH(NH2) and CH(N=CH2); R and R' (same or different) are H or 1 or 2 gps. selected from Cl, OH and Me; B is a 1-6C satd. divalent hydrocarbon radical). Cpds. (I) have long-lasting antibacterial activity comparable to that of alkanoyloxymethyl penicillin esters, but with the added advantage that two penicillin groupings with different activities can be combined in the same cpd.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7436775A FR2290443A1 (en) | 1974-11-06 | 1974-11-06 | Antibacterial bis-penicillin esters - contg. and alkanedioyloxymethyl alcohol residue |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7436775A FR2290443A1 (en) | 1974-11-06 | 1974-11-06 | Antibacterial bis-penicillin esters - contg. and alkanedioyloxymethyl alcohol residue |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2290443A1 true FR2290443A1 (en) | 1976-06-04 |
FR2290443B3 FR2290443B3 (en) | 1977-08-05 |
Family
ID=9144698
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7436775A Granted FR2290443A1 (en) | 1974-11-06 | 1974-11-06 | Antibacterial bis-penicillin esters - contg. and alkanedioyloxymethyl alcohol residue |
Country Status (1)
Country | Link |
---|---|
FR (1) | FR2290443A1 (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0083484A1 (en) * | 1981-12-22 | 1983-07-13 | Pfizer Inc. | 1,1-Alkanediol dicarboxylate linked antibacterial agents |
-
1974
- 1974-11-06 FR FR7436775A patent/FR2290443A1/en active Granted
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0083484A1 (en) * | 1981-12-22 | 1983-07-13 | Pfizer Inc. | 1,1-Alkanediol dicarboxylate linked antibacterial agents |
JPH02270881A (en) * | 1981-12-22 | 1990-11-05 | Pfizer Inc | 1,1-alkanedioldicarboxilate binding antibacterial agent |
Also Published As
Publication number | Publication date |
---|---|
FR2290443B3 (en) | 1977-08-05 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |