ECSP961694A - PROCEDURE FOR PREPARING OLANZAPINE (CASE X - 9992M) - Google Patents

PROCEDURE FOR PREPARING OLANZAPINE (CASE X - 9992M)

Info

Publication number
ECSP961694A
ECSP961694A ECSP961694A ECSP961694A EC SP961694 A ECSP961694 A EC SP961694A EC SP961694 A ECSP961694 A EC SP961694A EC SP961694 A ECSP961694 A EC SP961694A
Authority
EC
Ecuador
Prior art keywords
procedure
case
olanzapine
preparing
methyl
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Terrence Michael Hotten
David Edward Tupper
Charles Arthur Bunnell
Barry Arnold Hendriksen
Samuel Dean Larsen
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP961694 priority Critical patent/ECSP961694A/en
Publication of ECSP961694A publication Critical patent/ECSP961694A/en

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  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

El invento se refiere a un nuevo procedimiento para preparar 2-metil-4-(4-metil-1-piperacinil)-10H-tieno[2,3-b][1,5] benzodiacepina (denominada en lo sucesivo con su nombre genérico "olanzapina") y a nuevos solvatos alcohólicos valiosos en este procedimiento, especilamente una forma de solvato monometanólico cristalino de un compuesto de la siguiente fórmula: (gráfico).The invention relates to a new process for preparing 2-methyl-4- (4-methyl-1-piperazinyl) -10H-thieno [2,3-b] [1,5] benzodiazepine (hereinafter named Generic "Olanzapine") and to new valuable alcoholic solvates in this process, specifically a form of crystalline monomethanolic solvate of a compound of the following formula: (graph).

ECSP961694 1996-03-21 1996-03-21 PROCEDURE FOR PREPARING OLANZAPINE (CASE X - 9992M) ECSP961694A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP961694 ECSP961694A (en) 1996-03-21 1996-03-21 PROCEDURE FOR PREPARING OLANZAPINE (CASE X - 9992M)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP961694 ECSP961694A (en) 1996-03-21 1996-03-21 PROCEDURE FOR PREPARING OLANZAPINE (CASE X - 9992M)

Publications (1)

Publication Number Publication Date
ECSP961694A true ECSP961694A (en) 1997-11-04

Family

ID=42042426

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP961694 ECSP961694A (en) 1996-03-21 1996-03-21 PROCEDURE FOR PREPARING OLANZAPINE (CASE X - 9992M)

Country Status (1)

Country Link
EC (1) ECSP961694A (en)

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