ECSP003372A - OXAMIC ACIDS AND DERIVATIVES AS LEGANDS OF THYROID RECEPTORS - Google Patents
OXAMIC ACIDS AND DERIVATIVES AS LEGANDS OF THYROID RECEPTORSInfo
- Publication number
- ECSP003372A ECSP003372A ECSP003372A ECSP003372A EC SP003372 A ECSP003372 A EC SP003372A EC SP003372 A ECSP003372 A EC SP003372A EC SP003372 A ECSP003372 A EC SP003372A
- Authority
- EC
- Ecuador
- Prior art keywords
- prodrugs
- isomers
- compounds
- legands
- derivatives
- Prior art date
Links
Abstract
La presente invención proporciona nuevos compuestos de la fórmula (gráfico), y profármacos de los mismos, isómeros geométricos y ópticos de los mismos y sales farmacéuticamente aceptables de tales compuestos, profármacos e isómeros, en los que R1-R8 y W son como se describen en este documento. También se proporcionan composiciones farmacéuticas que contienen tales compuestos,, profármacos, isómeros o sales farmacéuticamente aceptables de los mismos, y procedimientos, composiciones farmacéuticas y estuches para el tratamiento de la obesidad, hiperlipidemia, glaucoma, arritmia cardiaca, transtornos cutáneos, enfermedad de tiroides, hipotiroidismo y trastornos y enfermedades relacionadas tales como diabetes mellitus, arterosclerosis, hipertensión, enfermedad cardiaca coronaria, hipercolesterolemia, depresión y osteoporosis.The present invention provides new compounds of the formula (graph), and prodrugs thereof, geometric and optical isomers thereof and pharmaceutically acceptable salts of such compounds, prodrugs and isomers, wherein R1-R8 and W are as described. in this document. Also provided are pharmaceutical compositions containing such compounds, prodrugs, isomers or pharmaceutically acceptable salts thereof, and methods, pharmaceutical compositions and kits for the treatment of obesity, hyperlipidemia, glaucoma, cardiac arrhythmia, skin disorders, thyroid disease, hypothyroidism and related disorders and diseases such as diabetes mellitus, atherosclerosis, hypertension, coronary heart disease, hypercholesterolemia, depression and osteoporosis.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003372 ECSP003372A (en) | 2000-02-29 | 2000-02-29 | OXAMIC ACIDS AND DERIVATIVES AS LEGANDS OF THYROID RECEPTORS |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003372 ECSP003372A (en) | 2000-02-29 | 2000-02-29 | OXAMIC ACIDS AND DERIVATIVES AS LEGANDS OF THYROID RECEPTORS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003372A true ECSP003372A (en) | 2001-09-24 |
Family
ID=42041003
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003372 ECSP003372A (en) | 2000-02-29 | 2000-02-29 | OXAMIC ACIDS AND DERIVATIVES AS LEGANDS OF THYROID RECEPTORS |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003372A (en) |
-
2000
- 2000-02-29 EC ECSP003372 patent/ECSP003372A/en unknown
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