AU6360999A - Process for producing 4-arylpiperidine-3-carbinols and related compounds - Google Patents

Process for producing 4-arylpiperidine-3-carbinols and related compounds

Info

Publication number
AU6360999A
AU6360999A AU63609/99A AU6360999A AU6360999A AU 6360999 A AU6360999 A AU 6360999A AU 63609/99 A AU63609/99 A AU 63609/99A AU 6360999 A AU6360999 A AU 6360999A AU 6360999 A AU6360999 A AU 6360999A
Authority
AU
Australia
Prior art keywords
arylpiperidine
carbinols
producing
related compounds
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU63609/99A
Inventor
Franciscus Bernardus Gemma Benneker
Hans Jan Hoorn
Theodorus Hendricus Antonius Peters
Frantisek Picha
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthon BV
Original Assignee
Synthon BV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthon BV filed Critical Synthon BV
Publication of AU6360999A publication Critical patent/AU6360999A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/74—Oxygen atoms
    • C07D211/76—Oxygen atoms attached in position 2 or 6
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU63609/99A 1998-11-02 1999-11-01 Process for producing 4-arylpiperidine-3-carbinols and related compounds Abandoned AU6360999A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10667398P 1998-11-02 1998-11-02
US60106673 1998-11-02
PCT/IB1999/001762 WO2000026187A1 (en) 1998-11-02 1999-11-01 Process for producing 4-arylpiperidine-3-carbinols and related compounds

Publications (1)

Publication Number Publication Date
AU6360999A true AU6360999A (en) 2000-05-22

Family

ID=22312658

Family Applications (1)

Application Number Title Priority Date Filing Date
AU63609/99A Abandoned AU6360999A (en) 1998-11-02 1999-11-01 Process for producing 4-arylpiperidine-3-carbinols and related compounds

Country Status (5)

Country Link
EP (1) EP1124802A1 (en)
AU (1) AU6360999A (en)
CZ (1) CZ20011465A3 (en)
NO (1) NO20012099L (en)
WO (1) WO2000026187A1 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AP9901698A0 (en) * 1997-05-29 1999-12-31 Smithkline Beecham Corp Novel process.
US20010053862A1 (en) * 1998-12-22 2001-12-20 Bruce Ronsen Process for preparing arylpiperidine carbinol intermediates and derivatives
EP1140832A4 (en) * 1998-12-22 2004-11-03 Pentech Pharmaceuticals Inc Process for preparing arylpiperidine carbinol intermediates and derivatives
CZ20023694A3 (en) * 2000-05-12 2003-05-14 Synthon B. V. Tosylate salts of 4-(p-fluorophenyl)-piperidine-3-methanols
JP2004520333A (en) 2001-01-04 2004-07-08 フエルレル インターナショナル，ソシエダッド アノニマ A method for producing (±) -trans-4-p-fluorophenyl-3-hydroxymethyl-1-methylpiperidine.
CA2464327A1 (en) 2001-10-22 2003-05-30 Synthon B.V. N-formyl derivatives of paroxetine
WO2007089193A1 (en) * 2006-02-02 2007-08-09 Astrazeneca Ab A process for preparing 2-hydroxy-3- [5- (morpholin-4-ylmethyl)pyridin-2-yl] lh-indole-5-carbonitrile as a free base or salts thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI792076A (en) * 1978-07-05 1980-01-06 Ciba Geigy Ag FOERFARANDE FOER FRAMSTAELLNING AV NYA FENYLPIPERIDINDERIVAT
EP0223334B1 (en) * 1985-08-10 1991-07-10 Beecham Group Plc Process for the preparation of aryl-piperidine carbinols
US5258517A (en) * 1992-08-06 1993-11-02 Sepracor, Inc. Method of preparing optically pure precursors of paroxetine
GB9526645D0 (en) * 1995-12-28 1996-02-28 Chiroscience Ltd Stereoselective synthesis
JP3446468B2 (en) * 1996-04-15 2003-09-16 旭硝子株式会社 Method for producing piperidine carbinols
AP9901698A0 (en) * 1997-05-29 1999-12-31 Smithkline Beecham Corp Novel process.

Also Published As

Publication number Publication date
NO20012099L (en) 2001-07-02
NO20012099D0 (en) 2001-04-27
CZ20011465A3 (en) 2001-08-15
EP1124802A1 (en) 2001-08-22
WO2000026187A1 (en) 2000-05-11

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase