ZA201601461B - Polymorphic form of pyrrole derivative and intermediate thereof - Google Patents
Polymorphic form of pyrrole derivative and intermediate thereofInfo
- Publication number
- ZA201601461B ZA201601461B ZA2016/01461A ZA201601461A ZA201601461B ZA 201601461 B ZA201601461 B ZA 201601461B ZA 2016/01461 A ZA2016/01461 A ZA 2016/01461A ZA 201601461 A ZA201601461 A ZA 201601461A ZA 201601461 B ZA201601461 B ZA 201601461B
- Authority
- ZA
- South Africa
- Prior art keywords
- polymorphic form
- pyrrole derivative
- pyrrole
- derivative
- polymorphic
- Prior art date
Links
- 150000003233 pyrroles Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/333—Radicals substituted by oxygen or sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/325—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Hematology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/IN2014/000551 WO2015029066A1 (en) | 2013-08-29 | 2014-08-28 | Polymorphic form of pyrrole derivative and intermediate thereof |
| IN2828MU2013 IN2013MU02828A (OSRAM) | 2013-08-29 | 2014-08-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA201601461B true ZA201601461B (en) | 2017-05-31 |
Family
ID=51947417
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA2016/01461A ZA201601461B (en) | 2013-08-29 | 2016-03-03 | Polymorphic form of pyrrole derivative and intermediate thereof |
Country Status (7)
| Country | Link |
|---|---|
| US (3) | US9951009B2 (OSRAM) |
| EP (1) | EP3039011A1 (OSRAM) |
| IN (1) | IN2013MU02828A (OSRAM) |
| MX (1) | MX371021B (OSRAM) |
| PH (1) | PH12016500394A1 (OSRAM) |
| WO (1) | WO2015029066A1 (OSRAM) |
| ZA (1) | ZA201601461B (OSRAM) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2825456C (en) | 2011-01-31 | 2016-01-05 | Cadila Healthcare Limited | Treatment for lipodystrophy |
| CA2900435C (en) | 2013-04-22 | 2017-02-14 | Cadila Healthcare Limited | A novel composition for nonalcoholic fatty liver disease (nafld) |
| PH12015502667B1 (en) | 2013-05-30 | 2023-10-18 | Zydus Lifesciences Ltd | A process for preparation of pyrroles having hypolipidemic hypocholesteremic activities |
| TW201513857A (zh) | 2013-07-05 | 2015-04-16 | Cadila Healthcare Ltd | 協同性組成物 |
| IN2013MU02470A (OSRAM) | 2013-07-25 | 2015-06-26 | Cadila Healthcare Ltd | |
| US10112898B2 (en) | 2013-09-06 | 2018-10-30 | Cadila Healthcare Limited | Process for the preparation of saroglitazar pharmaceutical salts |
| US20180125816A1 (en) * | 2015-05-11 | 2018-05-10 | Cadila Healthcare Limited | Saroglitazar magnesium for the treatment of chylomicronemia syndrome |
| US10385017B2 (en) | 2015-10-14 | 2019-08-20 | Cadila Healthcare Limited | Pyrrole compound, compositions and process for preparation thereof |
| ES2894261T3 (es) | 2016-12-09 | 2022-02-14 | Cadila Healthcare Ltd | Tratamiento de la colangitis biliar primaria |
| MX2020008066A (es) * | 2018-01-30 | 2020-09-25 | Kainos Medicine Inc | Formas de sal de compuesto organico. |
| WO2020183379A1 (en) * | 2019-03-11 | 2020-09-17 | Cadila Healthcare Limited | Novel salts, crystalline forms and premix of hypolipidemic agent |
| US12201611B2 (en) * | 2020-07-24 | 2025-01-21 | Zydus Lifesciences Limited | Composition comprising high purity pyrrole derivative and method for preparation thereof |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6713494B1 (en) * | 1996-08-28 | 2004-03-30 | Eli Lilly And Company | Amorphous benzothiophenes, methods of preparation and methods of use |
| TR200001903T2 (tr) * | 1998-01-07 | 2000-11-21 | Meiji Seika Kaisha, Ltd. | Kristalografik açıdan kararlı, şekilsiz sefalosporin bileşimleri ve bunların üretilmesine ilişkin işlem. |
| SI20425A (sl) * | 1999-12-10 | 2001-06-30 | LEK tovarna farmacevtskih in kemi�nih izdelkov d.d. | Priprava amorfnega atorvastatina |
| US6514995B1 (en) | 2000-09-25 | 2003-02-04 | Advanced Research And Technology Institute, Inc. | Enediyne compounds and methods related thereto |
| US6627760B1 (en) * | 2001-06-25 | 2003-09-30 | Astrazeneca Ab | Amorphous compound |
| US6987123B2 (en) | 2001-07-26 | 2006-01-17 | Cadila Healthcare Limited | Heterocyclic compounds, their preparation, pharmaceutical compositions containing them and their use in medicine |
| WO2004000823A1 (en) * | 2002-06-21 | 2003-12-31 | Dr. Reddy's Laboratories Limited | Amorphous form of(-)-}2-}4-}(4-chlorophenyl)-phenyl methyl}-1-piperazinyl] ethoxy] acetic acid dihydrochloride (levocetririzine dihydrochloride) |
| HRP20020614A2 (en) * | 2002-07-22 | 2004-06-30 | PLIVA-ISTRAŽIVAČKI INSTITUT d.o.o. | Rhombic pseudopolymorph of 9-deoxo-9a-aza-9a-methyl-9a-homoerythromycin a |
| WO2004067512A1 (en) * | 2003-01-27 | 2004-08-12 | Hanmi Pharm. Co., Ltd. | Stable amorphous amlodipine camsylate, process for preparing same and composition for oral administration thereof |
| US20040266787A1 (en) * | 2003-03-25 | 2004-12-30 | Dr. Reddy's Laboratories Limited | Novel amorphous form of [2-[4-[(4-chlorophenyl)-phenyl methyl]-1-piperazinyl]ethoxy]acetic acid and process for the preparation thereof |
| CN1874771A (zh) * | 2003-09-03 | 2006-12-06 | 惠氏公司 | 3－羟基－2－(羟甲基)－2－甲基丙酸的非晶态雷帕霉素42－酯及其包含相同化合物的药用组合物 |
| AR052918A1 (es) * | 2005-02-25 | 2007-04-11 | Recordati Ireland Ltd | Clorhidrato de lercanidipina amorfo |
| US10532028B2 (en) * | 2005-07-28 | 2020-01-14 | Isp Investments Llc | Method to improve characteristics of spray dried powders and granulated materials, and the products thereby produced |
| US20080085315A1 (en) * | 2006-10-10 | 2008-04-10 | John Alfred Doney | Amorphous ezetimibe and the production thereof |
| CA2825456C (en) * | 2011-01-31 | 2016-01-05 | Cadila Healthcare Limited | Treatment for lipodystrophy |
| PH12015502667B1 (en) | 2013-05-30 | 2023-10-18 | Zydus Lifesciences Ltd | A process for preparation of pyrroles having hypolipidemic hypocholesteremic activities |
-
2014
- 2014-08-28 US US14/915,457 patent/US9951009B2/en active Active
- 2014-08-28 WO PCT/IN2014/000551 patent/WO2015029066A1/en not_active Ceased
- 2014-08-28 EP EP14802513.3A patent/EP3039011A1/en not_active Withdrawn
- 2014-08-28 IN IN2828MU2013 patent/IN2013MU02828A/en unknown
- 2014-08-28 MX MX2016002612A patent/MX371021B/es active IP Right Grant
-
2016
- 2016-02-29 PH PH12016500394A patent/PH12016500394A1/en unknown
- 2016-03-03 ZA ZA2016/01461A patent/ZA201601461B/en unknown
-
2018
- 2018-04-06 US US15/947,044 patent/US20180297945A1/en not_active Abandoned
- 2018-04-06 US US15/947,049 patent/US20180297946A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US9951009B2 (en) | 2018-04-24 |
| US20160207884A1 (en) | 2016-07-21 |
| US20180297945A1 (en) | 2018-10-18 |
| EP3039011A1 (en) | 2016-07-06 |
| MX2016002612A (es) | 2016-10-04 |
| IN2013MU02828A (OSRAM) | 2015-07-03 |
| MX371021B (es) | 2020-01-13 |
| WO2015029066A1 (en) | 2015-03-05 |
| US20180297946A1 (en) | 2018-10-18 |
| PH12016500394A1 (en) | 2016-05-16 |
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