ZA200705017B - Liposomal formulation of bortezomib (PS-341) - Google Patents

Liposomal formulation of bortezomib (PS-341)

Info

Publication number
ZA200705017B
ZA200705017B ZA200705017A ZA200705017A ZA200705017B ZA 200705017 B ZA200705017 B ZA 200705017B ZA 200705017 A ZA200705017 A ZA 200705017A ZA 200705017 A ZA200705017 A ZA 200705017A ZA 200705017 B ZA200705017 B ZA 200705017B
Authority
ZA
South Africa
Prior art keywords
bortezomib
liposomal formulation
liposomal
formulation
Prior art date
Application number
ZA200705017A
Other languages
English (en)
Inventor
Zalipsky Samuel
Martin Francis
Original Assignee
Alza Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alza Corp filed Critical Alza Corp
Publication of ZA200705017B publication Critical patent/ZA200705017B/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7024Esters of saccharides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Liposomes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Liposomes
    • A61K9/1271Non-conventional liposomes, e.g. PEGylated liposomes, liposomes coated with polymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Dispersion Chemistry (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Dermatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
ZA200705017A 2004-11-05 2007-06-04 Liposomal formulation of bortezomib (PS-341) ZA200705017B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US62521604P 2004-11-05 2004-11-05

Publications (1)

Publication Number Publication Date
ZA200705017B true ZA200705017B (en) 2008-09-25

Family

ID=35947260

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200705017A ZA200705017B (en) 2004-11-05 2007-06-04 Liposomal formulation of bortezomib (PS-341)

Country Status (21)

Country Link
US (2) US20060159736A1 (xx)
EP (2) EP1807053A1 (xx)
JP (2) JP2008519041A (xx)
KR (2) KR20070085644A (xx)
CN (2) CN101094649A (xx)
AR (1) AR051759A1 (xx)
AU (2) AU2005304881A1 (xx)
BR (2) BRPI0517061A (xx)
CA (2) CA2586354A1 (xx)
CR (1) CR9168A (xx)
EA (1) EA200701005A1 (xx)
IL (1) IL182967A0 (xx)
MX (2) MX2007005497A (xx)
NI (1) NI200700120A (xx)
NO (1) NO20072830L (xx)
NZ (2) NZ554950A (xx)
PE (1) PE20061135A1 (xx)
TW (1) TW200618820A (xx)
UY (1) UY29191A1 (xx)
WO (2) WO2006052733A1 (xx)
ZA (1) ZA200705017B (xx)

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RU2599791C2 (ru) 2010-08-10 2016-10-20 Ремпекс Фармасьютикэлз, Инч. Циклические бороновые кислотно-эфирные производные и их использование в терапии
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Also Published As

Publication number Publication date
KR20070085644A (ko) 2007-08-27
CN101094648A (zh) 2007-12-26
AR051759A1 (es) 2007-02-07
AU2005304880A1 (en) 2006-05-18
NZ554951A (en) 2010-12-24
MX2007005497A (es) 2007-09-21
EA200701005A1 (ru) 2007-10-26
EP1807053A1 (en) 2007-07-18
CN101094649A (zh) 2007-12-26
KR20070085642A (ko) 2007-08-27
CA2586348A1 (en) 2006-05-18
WO2006052734A1 (en) 2006-05-18
AU2005304881A1 (en) 2006-05-18
JP2008519041A (ja) 2008-06-05
UY29191A1 (es) 2006-01-31
EP1807052A1 (en) 2007-07-18
JP2008519040A (ja) 2008-06-05
IL182967A0 (en) 2007-08-19
WO2006052733A1 (en) 2006-05-18
NI200700120A (es) 2008-05-15
CR9168A (es) 2008-11-24
NZ554950A (en) 2010-12-24
BRPI0517668A (pt) 2008-10-14
PE20061135A1 (es) 2006-10-20
US20060159736A1 (en) 2006-07-20
MX2007005499A (es) 2007-09-21
NO20072830L (no) 2007-07-24
TW200618820A (en) 2006-06-16
BRPI0517061A (pt) 2008-09-30
CA2586354A1 (en) 2006-05-18
US20060153907A1 (en) 2006-07-13

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