ZA200703022B - N-benzenesulfonyl substituted anilino-pyrimidine analogs - Google Patents
N-benzenesulfonyl substituted anilino-pyrimidine analogsInfo
- Publication number
- ZA200703022B ZA200703022B ZA200703022A ZA200703022A ZA200703022B ZA 200703022 B ZA200703022 B ZA 200703022B ZA 200703022 A ZA200703022 A ZA 200703022A ZA 200703022 A ZA200703022 A ZA 200703022A ZA 200703022 B ZA200703022 B ZA 200703022B
- Authority
- ZA
- South Africa
- Prior art keywords
- pyrimidine analogs
- substituted anilino
- benzenesulfonyl substituted
- benzenesulfonyl
- anilino
- Prior art date
Links
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- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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US6949544B2 (en) * | 2001-03-29 | 2005-09-27 | Vertex Pharmaceuticals Incorporated | Inhibitors of c-Jun N-terminal kinases (JNK) and other protein kinases |
MXPA03009257A (es) | 2001-04-10 | 2004-01-29 | Vertex Pharma | Derivados de isoxaxol como inhibidores de src y otras proteinas cinasas. |
JP2004535381A (ja) * | 2001-04-13 | 2004-11-25 | バーテックス ファーマシューティカルズ インコーポレイテッド | c−JunN末端キナーゼ(JNK)および他のプロテインキナーゼのインヒビター |
JP4316893B2 (ja) * | 2001-05-16 | 2009-08-19 | バーテックス ファーマシューティカルズ インコーポレイテッド | Srcおよび他のプロテインキナーゼのインヒビター |
CN100480242C (zh) * | 2001-05-29 | 2009-04-22 | 舍林股份公司 | Cdk抑制性嘧啶化合物、其制备方法以及作为药物的应用 |
ES2274035T3 (es) | 2001-06-01 | 2007-05-16 | Vertex Pharmaceuticals Incorporated | Compuestos de tiazol utiles como inhibidores de proteina quinasas. |
CA2450769A1 (fr) * | 2001-06-15 | 2002-12-27 | Vertex Pharmaceuticals Incorporated | 5-(2-aminopyrimidine-4-yl) benzisoxazoles en tant qu'inhibiteurs de proteine kinases |
US6939874B2 (en) * | 2001-08-22 | 2005-09-06 | Amgen Inc. | Substituted pyrimidinyl derivatives and methods of use |
US6703414B2 (en) | 2001-09-14 | 2004-03-09 | Arizona Board Of Regents On Behalf Of The University Of Arizona | Device and method for treating restenosis |
EP1472233A1 (fr) * | 2002-02-08 | 2004-11-03 | SmithKline Beecham Corporation | Composes de pyrimidine |
US7338959B2 (en) * | 2002-03-01 | 2008-03-04 | Smithkline Beecham Corporation | Diamino-pyrimidines and their use as angiogenesis inhibitors |
US7442697B2 (en) | 2002-03-09 | 2008-10-28 | Astrazeneca Ab | 4-imidazolyl substituted pyrimidine derivatives with CDK inhibitory activity |
GB0215844D0 (en) * | 2002-07-09 | 2002-08-14 | Novartis Ag | Organic compounds |
JP2006512314A (ja) * | 2002-11-01 | 2006-04-13 | バーテックス ファーマシューティカルズ インコーポレイテッド | Jakインヒビターおよび他のプロテインキナーゼインヒビターとしての組成物の使用 |
WO2004041810A1 (fr) * | 2002-11-05 | 2004-05-21 | Vertex Pharmaceuticals Incorporated | Composes utiles comme inhibiteurs de proteines jak et autres proteines kinase |
GB0226583D0 (en) * | 2002-11-14 | 2002-12-18 | Cyclacel Ltd | Compounds |
GB0226582D0 (en) * | 2002-11-14 | 2002-12-18 | Cyclacel Ltd | Anti-viral compounds |
-
2005
- 2005-10-13 KR KR1020077010445A patent/KR20070084067A/ko not_active Application Discontinuation
- 2005-10-13 JP JP2007536838A patent/JP2008515986A/ja active Pending
- 2005-10-13 TW TW094135620A patent/TW200626559A/zh unknown
- 2005-10-13 EP EP05812654A patent/EP1799652A1/fr not_active Withdrawn
- 2005-10-13 CN CNA2005800349350A patent/CN101039919A/zh not_active Withdrawn
- 2005-10-13 PA PA20058649401A patent/PA8649401A1/es unknown
- 2005-10-13 BR BRPI0516597-0A patent/BRPI0516597A/pt not_active IP Right Cessation
- 2005-10-13 AU AU2005295788A patent/AU2005295788A1/en not_active Abandoned
- 2005-10-13 WO PCT/US2005/036674 patent/WO2006044457A1/fr active Application Filing
- 2005-10-13 CA CA002580913A patent/CA2580913A1/fr not_active Abandoned
- 2005-10-13 US US11/248,495 patent/US7799915B2/en not_active Expired - Fee Related
- 2005-10-13 MX MX2007004488A patent/MX2007004488A/es unknown
- 2005-10-13 RU RU2007114080/04A patent/RU2007114080A/ru not_active Application Discontinuation
- 2005-10-13 PE PE2005001207A patent/PE20060582A1/es not_active Application Discontinuation
- 2005-10-13 GT GT200500286A patent/GT200500286A/es unknown
- 2005-10-13 AR ARP050104293A patent/AR051387A1/es not_active Application Discontinuation
-
2007
- 2007-03-28 NO NO20071642A patent/NO20071642L/no not_active Application Discontinuation
- 2007-03-29 IL IL182316A patent/IL182316A0/en unknown
- 2007-04-11 CR CR9048A patent/CR9048A/es unknown
- 2007-04-12 ZA ZA200703022A patent/ZA200703022B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
PA8649401A1 (es) | 2006-09-22 |
IL182316A0 (en) | 2007-07-24 |
KR20070084067A (ko) | 2007-08-24 |
BRPI0516597A (pt) | 2008-09-16 |
WO2006044457A1 (fr) | 2006-04-27 |
US7799915B2 (en) | 2010-09-21 |
GT200500286A (es) | 2006-06-13 |
TW200626559A (en) | 2006-08-01 |
PE20060582A1 (es) | 2006-08-17 |
CR9048A (es) | 2007-08-28 |
MX2007004488A (es) | 2007-09-11 |
RU2007114080A (ru) | 2008-11-27 |
JP2008515986A (ja) | 2008-05-15 |
US20060079543A1 (en) | 2006-04-13 |
AR051387A1 (es) | 2007-01-10 |
CN101039919A (zh) | 2007-09-19 |
EP1799652A1 (fr) | 2007-06-27 |
AU2005295788A1 (en) | 2006-04-27 |
CA2580913A1 (fr) | 2006-04-27 |
NO20071642L (no) | 2007-06-01 |
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